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2016年5月24日星期二

May 24, New compounds

Below is new Compounds we have finished.

Any interesting, welcome to my booth to have a meet.


2016 Shanghai CPHI, W5C47, Welcome!
EOS Med ChemMedchem is Big
執大象,天下往,往而無害,安平泰
網址www.eosmedchem.com 
辦公室: 0086-531-69905422-806(直通)
攜帶番號 & WhatsApp: +8618653174435

Skype: willgutian


1  4-Chloro-1H-pyrrolo[2,3-b]pyridine 55052-28-3 690/100g 1150/250g 1850/kg Stock
2 4-​Chloro-​1-​(phenylsulfonyl)​-1H-​Pyrrolo[2,​3-​b]​pyridine 744209-63-0 780/100g 1150/250g 2700/kg 4 Weeks
3 4-Chloro-5-nitro-1H-pyrrolo[2,3-b]pyridine 1245645-97-9 3050/100g 3850/250g 7700/kg 5 weeks
4 4-​Chloro-​5-​nitro-​1-​(phenylsulfonyl)​-1H-​pyrrolo[2,​3-​b]​pyridine 1245649-52-8 3050/100g 3850/250g 7700/kg 5 Weeks
5 5-​Nitro-1H-​Pyrrolo[2,​3-​b]​pyridine-​4-​carbonitrile 1401447-80-0 3050/100g 3850/250g 7700/kg 5 Weeks
6 3-Pyrrolidinecarboxylic acid 59378-87-9 1050/100g 1350/250g 3700/kg 6 Weeks
7 1-​(Phenylmethyl)​-3-​pyrrolidinecarboxyli​c acid 5731-18-0 1260/100g 1460/250g 1850/kg 3 Weeks
8 1-​Acetyl-3-​Pyrrolidinecarboxyli​c acid  712270-40-1 1550/100g 2550/250g 4150/kg 5-6 Weeks
9 1-​Benzoyl-3-​Pyrrolidinecarboxyli​c acid  113558-92-2 1180/100g 1850/250g 3030/kg 5-6 Weeks
10 5-Oxo-3-pyrrolidinecarboxylic acid 7268-43-1 1180/100g 1850/250g 3030/kg 5-6 Weeks
11 5-Oxo-1-benzylpyrrolidine-3-carboxylic acid 5733-86-8 780/100g 1180/250g 1850/kg 5-6 Weeks
12 3-Nitromethyl-1-phenylmethylpyrrolidine 1369148-11-7 1550/100g 2050/250g 4350/kg 5-6 Weeks
13 1-​Pyrrolidinecarboxyli​c acid, 3-​(nitromethyl)​-​, 1,​1-​dimethylethyl ester 1369237-63-7 2180/100g 2700/250g 4700/kg 5-6 Weeks
14 1-​Pyrrolidinecarboxyli​c acid, 4-​(nitromethyl)​-​2-​oxo-​, 1,​1-​dimethylethyl ester 1026779-31-6 1550/100g 2050/250g 4350/kg 5-6 Weeks
15 1-​(Phenylmethyl)​-2-​Pyrrolidinone 5291-77-0 550/100g 620/250g 690/kg Stock

2016年5月23日星期一

Pass Trial, will commercial production



2016, May - July new project will start.

Below API and Intermediates, we have finished Trial Production.

2016 China CPHI, welcome to my booth to talk about.

2016 Shanghai CPHI, W5C47, Welcome!
EOS Med ChemMedchem is Big
執大象,天下往,往而無害,安平泰
網址www.eosmedchem.com 
辦公室: 0086-531-69905422-806(直通)
攜帶番號 & WhatsApp: +8618653174435

Skype: willgutian


Niraparib1038915-60-41038915-56-8 1038915-60-4
Lucitanib1058137-23-71058137-21-5
Tivozanib475108-18-01072-67-9 1885-14-9 286371-44-6
Baricitinib1187594-09-71146629-75-5 1029716-44-6 1187595-85-2 941685-26-3 1146627-77-7
Talazoparib1207456-01-61207454-56-5 1207456-00-5 1373329-52-2 1322616-40-9 1322616-38-5 1322616-37-4 1322616-36-3
Ertugliflozin1210344-57-21210763-25-9 1210344-57-2 1233482-00-2
Abemaciclib1231929-97-71231930-82-7
Venetoclax1257044-40-81235865-75-41228780-72-0 1235865-77-6 1228779-96-1 685514-01-6 1228837-05-5
Duvelisib1201438-56-31350643-72-9
87694-49-3
1350643-73-0
Rociletinib1374640-70-61374507-23-9 1021426-42-5 68621-88-5 
Osimertinib1421373-66-11421372-67-9 1421372-94-2 1421372-66-8
Olaparib763113-22-0218301-22-5 61260-15-9 763114-25-6 1021298-68-9 763114-26-7 1021298-67-8 763111-47-3
Plecainide Flecainide 54143-55-435480-52-5 66300-61-6 610-71-9
Pimavanserin706779-91-1359878-47-0 4734-09-2 955997-89-4
Velpatasvir1377049-84-738533-38-9 334769-80-1 1335316-40-9 37074-40-1 1438383-92-6 1335316-40-9 1438383-89-1 1377604-63-1 74844-91-0 487048-28-2 50890-96-5 113400-36-5 38533-38-9 1335316-40-9
Filgotinib1206161-97-839093-93-1 1206163-59-8
Rucaparib283173-50-2459868-92-9 283173-80-8
Obeticholic acid459789-99-24651-67-6 10538-59-7 77341-09-4 863239-59-2 1516887-33-4 915038-26-5 1352328-67-6 1352328-66-5 1352328-65-4 1352328-64-3 111992-94-0
Selexipag475086-01-2475086-75-0 42042-71-7 41270-66-0
Lenvatinib417716-92-8491-11-2 17609-80-2 796848-80-1 796848-79-8 52671-64-4
Neratinib698387-09-6524955-09-7848133-76-6 848139-78-6 915942-01-7 915941-95-6 149586-32-3 524955-09-7 848133-76-6
Veliparib912444-00-963399-77-9 42856-71-3 166170-15-6 63399-74-6
Masitinib790299-79-5660837-08-1 314268-40-1 148077-69-4106261-48-7
Momelotinib1056634-68-4945749-71-3 6011-14-9
Panabinostat404950-80-7960058-93-9 441741-66-8
Aripiprazole lauroxil1259305-29-7
Cinitapride96623-56-2
Etelcalcetide1262780-97-1
ZS-9 (Sodium Zirconium cyclosilicate)242800-27-7
Fovista*
Ozanimod1306760-87-1
GED - 0301
Velcalcetide1334237-71-6, 1262780-97-1
Roxadustat808118-40-3
Naldemedine916072-89-4
Orantinib252916-29-3
CVT 301
Nusinersen1258984-36-9
Volanesorsen1573402-50-2
Custirsen903916-27-8
Alicaforsen185229-68-9
SAGE-547516-54-1
Acalabrutinib1420477-60-6
Crisaborole906673-24-3 
Patisiran
Motesanib453562-69-1

2016年5月20日星期五

Stock List



Below is some Intermediates, one of my Japan market supplier have stock list.

Most in sotck.

99% HPLC, NMR, MS is ok.


2016 Shanghai CPHI, W5C47, Welcome!
EOS Med ChemMedchem is Big
執大象,天下往,往而無害,安平泰
網址www.eosmedchem.com 
辦公室: 0086-531-69905422-806(直通)
攜帶番號 & WhatsApp: +8618653174435
Skype: willgutian


419572-18-2tert-Butyl (1R,5S,6R)-6-(hydroxymethyl)-3-azabicyclo[3.1.0]hexane-3-carboxylate500g in stock
 868733-71-54-(4-amino-2-fluorophenoxy)-picolinamide2kg in stock
1016636-76-26--2--8-环戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-2kg in stock
1031890-09-1benzyl (S)-2-carbamoyl-2-methylpyrrolidine-1-carboxylate500g in stock
103336-06-7(S)-1-(tert-butoxycarbonyl)-2-methylpyrrolidine-2-carboxylic acid
(S)-1-(tert-butoxycarbonyl)-2-methylpyrrolidine-2-carboxylic acid
100g in stock
105141-61-52-Piperidinecarboxylicacid,2-methyl-,(2R)2kg in stock
1064721-10-3[1-Benzyl-2-(3-bromo-phenoxy)-ethyl]-carbamic Acid Tert-Butyl Ester2kg in stock
1093865-09-81,1-dimethylethyl {(1R)-2-amino-1-[(3S)-tetrahydro-2H-pyran-3-ylmethyl]ethyl}methylcarbamate100g in stock
109772-27-22-Piperidinecarboxylicacid,2-methyl-,methylester,(S)2kg in stock
109-82-0亚甲氨基乙腈2kg in stock
1194-18-91,3-环庚二酮2.5kg in stock
1256039-44-7tert-butyl (3aR,5s,6aS)-5-cyanohexahydrocyclopenta[c]-pyrrole-2(1H)-carboxylate2.5kg in stock
1256240-40-0(3aR,5r,6aS)-octahydrocyclopenta[c]pyrrol-5-ol hydrochloride2kg in stock
1271145-38-0(3S*,4R*)-tetrahydro-3,4-ethylenedioxythiophene2.5kg in stock
1383481-11-57-chloroimidazo[1,2-b]pyridazine2kg in stock
146231-54-1cis-5-Oxohexahydrocyclopenta[c]pyrrole-2(1H)-carboxylic acid tert-butyl ester2kg in stock
170730-06-07-乙酰基-2,3-二氢苯并呋喃2kg in stock
19235-89-34--2-氰基吡啶2.5kg in stock
19524-67-5Ethyl (2E)-3-(piperidin-1-yl)acrylate100g in stock
26228-68-24-aminomethyl-4-hydroxy-1-methylpiperidine500g in stock
271-63-67-氮杂吲哚2.5kg in stock
275386-75-91,3-dihydro-5-fluoro-4-iodo-2H-indol-2-one2.5kg in stock
2854-16-21-AMino-2-Methylpropan-2-ol2.5kg in stock
289037-48-5(1R,5S,6R)-3-Azabicyclo[3.1.0]hexan-6-ylmethanol500g in stock
35700-40-42,3-二氢苯并呋喃-7-羧酸2kg in stock
486460-21-33-(三氟甲基)-5,6,7,8-四氢-[1,2,4]三唑并[4,3-a]吡嗪2.5kg in stock
5025-59-22-iodo-6-methoxy-Benzaldehyde2.5kg in stock
51207-66-0(S)-(+)-1-(2-Pyrrolidinylmethyl)pyrrolidine500g in stock
51411-49-51-aMino-2-Methylbutan-2-ol2.5kg in stock
5451-09-25-氨基乙酰丙酸盐酸盐100g in stock
55052-28-34--7-氮杂吲哚2.5kg in stock
552331-16-55--3-甲基-1H-吲唑2.5kg in stock
573762-62-6 5-Amino-3-(trifluromethyl) picolinonitrile 2kg in stock
60419-23-0(R)-1-(2-Pyrrolidinylmethyl)pyrrolidine2kg in stock
63399-74-6R-N-CBZ-2-Methylproline  D-500g in stock
63399-77-9(R)-2-Methylproline   D-100g in stock
65921-41-71-[(2S)-Pyrrolidinylmethyl]piperidine500g in stock
706806-60-2 (R)-2-benzyl-pyrrolidine-1,2-dicarboxylic acid 1-tert-butyl ester 100g in stock
7149-42-0C-(1-methyl-piperidin-4-yl)-methylamine500g in stock
747399-23-12-Azetidinecarboxylicacid,2-methyl-,methylester 100g in stock
749927-69-3N-甲基-4--2--苯甲酰胺2kg in stock
7568-93-62-AMINO-1-PHENYLETHANOL2.5kg in stock
76411-80-8 (S)-(-)-1-[(1-Methyl-2-pyrrolidinyl)methyl]pyrrolidine500g in stock
84466-85-3 (S)-(-)-1-[(1-Methyl-2-pyrrolidinyl)methyl]piperidine500g in stock
86116-84-9(R)-2-benzyl-pyrrolidine-2-carboxylic acid 100g in stock
868171-67-9 3-Pyridinecarboxylic acid, 1-(4-fluorophenyl)-1,2-dihydro-2-oxo-2kg in stock
876861-32-41-BroMo-2-Methoxy-3-nitro-benzene2.5kg in stock
89115-95-72-Piperidinecarboxylicacid,2-methyl-,(2S)100g in stock
915087-25-1N-甲基-4-氨基-2--苯甲酰胺2kg in stock
91790-91-94-[(2S)-Pyrrolidinylmethyl]morpholine500g in stock