Crisaborole; AN2728 906673-24-3 Inter:
1)
2-Bromo-5-hydroxy-benzaldehyde,CAS:2973-80-0,Appearance: white solid,HPLC,1H NMR 98%+;
2)
4-(4-Bromo-3-formyl-phenoxy)-benzonitrile,CAS: 906673-54-9,Appearance: white solid,HPLC,1H NMR 98%+;
3)
4-(4-Bromo-3-hydroxymethyl-phenoxy)-benzonitrile,CAS:906673-45-8,Appearance: white solid,HPLC,1H NMR 98%+;
4)
4-(4-bromo-3-(1,3-dioxolan-2-yl)phenoxy)benzonitrile,CAS#:1217366-74-9,外观:白色至类白色固体,HPLC,1H NMR 98%+;
1-萘酮-6-位衍生物
5)
6-Amino-3,4-dihydro-1(2H)-naphthalenone ;6-氨基-1,2,3,4-四氢-1-萘酮,CAS:3470-53-9;外观:浅黄棕色固体,HPLC,1H NMR 98%+
6)
6-Chloro-1-tetralone,6-氯-3,4-二氢-2H-1-萘酮,CAS: 26673-31-4;外观:浅黄色油状物,HPLC,1H NMR 97%+
7)
6-碘-3,4-二氢-2H-1-萘酮,CAS: 26673-31-4;外观:白色至类白色固体,HPLC,1H NMR 97%+
1)

2)

3)

4)

1-萘酮-6-位衍生物
5)

6)

7)

Carfilzomib,PR171中间体:
8)

CAS: 247068-81-1,Appearance: white solid,HPLC,1H NMR 99%+;
9)

CAS:247068-82-2,tert-butyl ((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-yl)carbamate,Appearance: white solid,HPLC,1H NMR 98%+;



10)
CAS:247068-85-5 ,Appearance: white solid,HPLC,1H NMR 98%+;
