EOS MED CHEM Stock List---2017.09.29

2017 China CPHI: E1M35

EOS Med Chem, Medchem is Big

執大象，天下往，往而無害，安平泰

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ABT-263 (Navitoclax),923564-51-6,ABT-263 (Navitoclax) is a potent inhibitor of Bcl-xL, Bcl-2 and Bcl-w with Ki of ≤ 0.5 nM, ≤1 nM and ≤ 1 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ABT-737,852808-04-9,ABT-737 is a BH3 mimetic inhibitor of Bcl-xL, Bcl-2 and Bcl-w with EC50 of 78.7 nM, 30.3 nM and 197.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Linifanib (ABT-869),796967-16-3,Linifanib (ABT-869) is a novel, potent ATP-competitive RTK inhibitor for KDR, CSF-1R, Flt-1, Flt-3 and PDGFRβ with IC50 of 4 nM, 3 nM, 3 nM, 3 nM, and 66 nM respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ABT-888 (Veliparib),912444-00-9,ABT-888 (Veliparib, NSC 737664) is a potent inhibitor of PARP1 and PARP2 with Ki of 5.2 nM and 2.9 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Axitinib,319460-85-0,Axitinib (AG-013736) is a multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFRβ and c-Kit with IC50 of 0.1 nM, 0.2 nM, 0.1-0.3 nM, 1.6 nM and 1.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Saracatinib (AZD0530),379231-04-6,Saracatinib (AZD0530) is a Src inhibitor for c-Src and v-Abl with IC50 of 2.7 nM and 30 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
FG-4592,808118-40-3,FG-4592 is an HIF α prolyl hydroxylase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD6244 (Selumetinib),606143-52-6,AZD6244 (Selumetinib, ARRY-142886) is highly potent to inhibit MEK1 with IC50 of 14 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BEZ235 (NVP-BEZ235),915019-65-7,BEZ235 (NVP-BEZ235) is a dual ATP-competitive PI3K and mTOR inhibitor of p110α, p110γ, p110δ and p110β with IC50 of 4 nM, 5 nM, 7 nM and 75 nM, respectively, and also inhibits ATR with IC50 of 21 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIBF1120 (Vargatef),656247-17-5,BIBF1120 (Vargatef) is a potent inhibitor of VEGFR1/2/3, FGFR1/2/3 and PDGFRα/β with IC50 of 34 nM/13 nM/13 nM, 69 nM/37 nM/108 nM and 59 nM/65 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Afatinib (BIBW2992),439081-18-2,BIBW2992 (Afatinib, Tomtovok, Tovok) irreversibly  inhibits EGFR/HER2 including EGFRwt, EGFRL858R, EGFRL858R/T790M and HER2 with IC50 of 0.5 nM, 0.4 nM, 10 nM and 14 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bortezomib (Velcade),179324-69-7,Bortezomib is a potent 20S proteasome inhibitor with Ki of 0.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bosutinib (SKI-606),380843-75-4,Bosutinib (SKI-606) is a novel, dual Src/Abl inhibitor with IC50 of 1.2 nM and 1 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cediranib (AZD2171),288383-20-0,Cediranib (AZD2171) is a highly potent VEGFR2 inhibitor with IC50 of 0.5 nM, also inhibits Flt1/4 with IC50 of 5 nM/≤3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dovitinib (TKI-258),405169-16-6,Dovitinib (TKI258, CHIR258) is a novel multi-target inhibitor for Flt3, c-Kit, FGFR1/3, VEGFR1/2/3, PDGFRα/β with IC50 of 1 nM, 2 nM, 8 nM/9 nM and 10 nM/13 nM/8 nM, 210 nM/27 nM respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CI-1033 (Canertinib),267243-28-7,CI-1033 is a potent inhibitor of EGFR and ErbB2 with IC50 of 1.5 nM and 9.0 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CI-1040 (PD184352),212631-79-3,CI-1040 (PD 184352) is an ATP non-competitive MEK1/2 inhibitor with IC50 of 17 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dasatinib (BMS-354825),302962-49-8,Dasatinib (BMS-354825, Sprycel) is a novel, potent and multi-targeted inhibitor that targets Abl, Src and c-Kit, with IC50 of ＜1 nM, 0.5 nM and 79 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Deforolimus (Ridaforolimus),572924-54-0,Deforolimus (Ridaforolimus, AP23573, MK-8669) is a selective mTOR inhibitor with IC50 of 0.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Erlotinib HCl,183319-69-9,Erlotinib HCl is an HER1/EGFR inhibitor with IC50 of 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gefitinib (Iressa),184475-35-2,Gefitinib (Iressa, ZD-1839) is an EGFR inhibitor for Tyr1173, Tyr992, Tyr1173 and Tyr992 in the NR6wtEGFR and NR6W cells with IC50 of 37 nM, 37nM, 26 nM and 57 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Imatinib Mesylate,220127-57-1,Imatinib Mesylate is orally bioavailability mesylate salt of Imatinib, which is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC50 of 0.6 μM, 0.1 μM and 0.1 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lapatinib Ditosylate (Tykerb),388082-77-7,Lapatinib Ditosylate (GW572016, GW2016, Tykerb, Tyverb) is a potent EGFR and ErbB2 inhibitor with IC50 of 10.8 and 9.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lenalidomide (Revlimid),191732-72-6,Lenalidomide (Revlimid, CC-5013) is a TNF-α secretion inhibitor with IC50 of 13 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Motesanib Diphosphate (AMG-706),857876-30-3,Motesanib Diphosphate (AMG-706) is a potent ATP-competitive inhibitor of VEGFR1/2/3, PDGFR, c-Kit and Ret with IC50 of 2 nM/3 nM/6 nM, 84 nM, 8 nM and 59 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nilotinib (AMN-107),641571-10-0,Nilotinib (AMN-107, Tasigna) is a Bcr-Abl inhibitor with IC50 less than 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-AEW541,475489-16-8 ,NVP-AEW541 is a potent inhibitor of IGF-1R with IC50 of 86 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pazopanib HCl,635702-64-6,Pazopanib Hydrochloride (GW786034, Votrient, Armala) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD0325901,391210-10-9,PD0325901 (PD325901) is selective and non ATP-competitive MEK inhibitor with IC50 of 0.33 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PI-103,371935-74-9,PI-103 is a potent, ATP-competitive PI3K inhibitor of DNA-PK, p110α, mTORC1, PI3KC2β, p110δ, mTORC2, p110β, and p110γ with IC50 of 2 nM, 8 nM, 20 nM, 26 nM, 48 nM, 83 nM, 88 nM and 150 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rapamycin (Sirolimus),53123-88-9,Rapamycin (Sirolimus, AY-22989, WY-090217) is a specific mTOR inhibitor with IC50 of ~0.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sorafenib (Nexavar),475207-59-1,Sorafenib Tosylate (Bay 43-9006, Nexavar) is a multikinase inhibitor of Raf-1, B-Raf and VEGFR-2 with IC50 of 6 nM, 22 nM and 90 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
STF-62247,315702-99-9,STF-62247 is selectively toxic and growth inhibitory to renal cells lacking VHL,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sunitinib Malate (Sutent),341031-54-7,Sunitinib Malate (Sutent, SU11248) is a multi-targeted RTK inhibitor targeting VEGFR2 (Flk-1) and PDGFRβ with IC50 of 80 nM and 2 nM, and also inhibits c-Kit.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tandutinib (MLN518),387867-13-2,Tandutinib (MLN518, CT53518) is an ATP-competitive and highly selective inhibitor of Flt3, PDGFRβ and c-Kit with IC50 of 0.22 μM, 0.20 μM and 0.17 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Temsirolimus (Torisel),162635-04-3,Temsirolimus (CCI-779, Torisel) is a specific mTOR inhibitor with IC50 of 1.76 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Trichostatin A (TSA),58880-19-6,Trichostatin A (TSA) is an HDAC inhibitor with IC50 of ~1.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vandetanib (Zactima),443913-73-3,Vandetanib (Zactima, ZD6474) is a potent inhibitor of VEGFR2 with IC50 of 40 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vorinostat (SAHA),149647-78-9,Vorinostat (suberoylanilide hydroxamic acid, SAHA, Zolinza) is an HDAC inhibitor with IC50 of ~10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VX-680 (MK-0457, Tozasertib),639089-54-6,VX-680 (MK-0457, Tozasertib) is a pan-Aurora inhibitor of Aurora A, Aurora B and Aurora C with Kiapp of 0.6 nM, 18 nM and 4.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Y-27632 2HCl,129830-38-2,Y-27632 2HCl is a selective ROCK1 (p160ROCK) inhibitor with Ki of 140 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Elesclomol,488832-69-5,Elesclomol (STA-4783) is a novel potent oxidative stress inducer that illicits pro-apoptosis events among tumor cells..,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Entinostat (MS-275, SNDX-275),209783-80-2,MS-275 is an HDAC inhibitor of HDAC1 and HDAC3 with IC50 of 0.51 μM and 1.7 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Enzastaurin (LY317615),170364-57-5,Enzastaurin (LY317615) is a potent PKC inhibitor for PKCβ, PKCα, PKCγ and PKCε with IC50 of 6 nM, 39 nM, 83 nM and 110 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS-599626 (AC480),714971-09-2,BMS-599626 (AC480) is a selective and efficacious inhibitor of HER1 and HER2 with IC50 of 20 nM and 30 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Obatoclax mesylate (GX15-070),803712-79-0,Obatoclax (GX15-070) is an inhibitor of Bcl-2 with Ki of 0.22 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Olaparib (AZD2281),763113-22-0,Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1 and PARP2 with IC50 of 5 nM and 1 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nutlin-3,890090-75-2,Nutlin-3 is a potent and selective Mdm2 (RING finger-dependent ubiquitin protein ligase for itself and p53) antagonist with IC50 of 90 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Masitinib (AB1010),790299-79-5,Masitinib is a novel tyrosine kinases inhibitor for Kit and PDGFRα/β with IC50 of 200 nM and 540 nM/800 nM, resectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GDC-0941,957054-30-7,GDC-0941 is a potent inhibitor of PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ with IC50 of 3 nM, 33 nM, 3 nM and 75 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SL327,305350-87-2,SL327 is a selective inhibitor for MEK1 and MEK2 with IC50 of 0.18 μM and 0.22 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 431542,301836-41-9,SB 431542 is a potent and selective inhibitor of ALK5 with IC50 of 94 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Crizotinib (PF-02341066),877399-52-5,PF-2341066 (Crizotinib) is a potent inhibitor of c-Met and ALK with IC50 of 11 nM and 24 nnM, respectivley.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AUY922 (NVP-AUY922),747412-49-3,NVP-AUY922 (VER-52296) is a highly potent HSP90 inhibitor for HSP90α and HSP90β with IC50 of 13 nM and 21 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PHA-665752,477575-56-7,PHA-665752 is a potent, selective and ATP-competitive c-Met inhibitor with IC50 of 9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
HA14-1,65673-63-4,HA14-1 is a nonpeptidic ligand of a Bcl-2 surface pocket with IC50 of~9 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZSTK474,475110-96-4,ZSTK474 is a potent pan-class I PI3K inhibitor with IC50 of 37 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 216763,280744-09-4,SB 216763 is a potent and selective GSK-3α inhibitor with IC50 of 34.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 203580,152121-47-6,SB203580 is a p38 MAPK inhibitor with IC50 of 0.3-0.5 μM and blocks PKB phosphorylation with IC50 of 3-5 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 202190,152121-30-7,SB 202190 (FHPI) is a potent p38 MAPK inhibitor targeting p38α and p38β with IC50 of 50 nM and 100 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-2206 2HCl,1032350-13-2,MK-2206 2HCl is a highly selective inhibitor of Akt1, Akt2 and Akt3 with IC50 of 8 nM, 12 nM and 65 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD153035 HCl,183322-45-4,PD153035 is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SU11274,658084-23-2,SU11274 is a selective Met inhibitor with IC50 of 10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vismodegib (GDC-0449),879085-55-9,GDC-0449 (Vismodegib, HhAntag691) is a potent, novel and specific hedgehog inhibitor with IC50 of 3 nM and also inhibits P-gp with IC50 of 3.0 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Brivanib (BMS-540215),649735-46-6,Brivanib is an ATP-competitive inhibitor against human VEGFR2 and FGFR with IC50 of 25 nM and 148 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Belinostat (PXD101),414864-00-9,Belinostat (PXD101) is a novel HDAC inhibitor with IC50 of 27 nM in HeLa cell extracts.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Iniparib (BSI-201),160003-66-7,BSI-201 (Iniparib, SAR240550) is a PARP1 inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-ADW742,475488-23-4,NVP-ADW742 is an IGF-1R inhibitor with IC50 of 0.17 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PCI-24781,783355-60-2,PCI-24781 (CRA-024781) is a novel broad spectrum HDAC inhibitor targeting HDAC1, HDAC2, HDAC3, HDAC6, HDAC8 and HDAC10 with Ki of 7 nM, 19 nM, 8.2 nM, 17 nM, 280 nM, 24 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Linsitinib (OSI-906),867160-71-2,OSI-906 (Linsitinib) is a selective inhibitor of IGF-1R and IR with IC50 of 35 nM and 75 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KU-55933,587871-26-9,KU-55933 is a potent and specific ATM inhibitor with IC50 and Ki of 13 nM and 2.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1904529A,1089283-49-7,GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-04217903,956905-27-4,PF-04217903 is a selective ATP-competitive c-Met inhibitor with IC50 of 4.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LAQ824 (NVP-LAQ824, Dacinostat),404951-53-7,LAQ824 (NVP-LAQ824) is a novel HDAC inhibitor with IC50 of 32 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ-26481585,875320-29-9,JNJ-26481585 (Quisinostat) is an HDAC inhibitor for HDAC1, HDAC2, HDAC4, HDAC10 and HDAC11 with IC50 of 0.11 nM, 0.33 nM, 0.64 nM, 0.46 nM and 0.37 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BTZ043 racemate,957217-65-1,BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2'-epimerase (DprE1) inhibitor acting as a new antimycobacterial agent that kill Mycobacterium tuberculosis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rucaparib (AG-014699 , PF-01367338),459868-92-9,Rucaparib (AG-014699, PF-01367338) is an inhibitor of PARP with Ki of 1.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MLN8054,869363-13-3,MLN8054 is a potent and selective inhibitor of Aurora A with IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vatalanib 2HCl (PTK787),212141-51-0,Vatalanib (PTK787) is an inhibitor of VEGFR2/KDR, Flt-1 and c-Kit with IC50 of 37 nM, 77 nM and 730 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
U0126-EtOH,1173097-76-1,U0126-EtOH is a highly selective inhibitor of MEK1 and MEK2 with IC50 of 0.07 μM and 0.06 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZM-447439,331771-20-1,ZM-447439 is a selective and ATP-competitive inhibitor for Aurora A and Aurora B with IC50 of 110 nM and 130 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GDC-0879,905281-76-7,GDC-0879 is a novel potent, selective B-Raf inhibitor for B-RafV600E with IC50 of 0.13 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY294002,154447-36-6,LY294002 is a PI3K inhibitor for p110α, p110δ and p110β with IC50 of 0.5 μM, 0.57 μM and 0.97 μM, and also blocks autophagosome formation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
OSU-03012 (AR-12) ,742112-33-0,OSU-03012 is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Danusertib (PHA-739358),827318-97-8,Danusertib (PHA-739358) is an Aurora inhibitor for Aurora A/B/C, Bcr-Abl, c-RET and FGFR with IC50 of 13 nM/79 nM/61 nM, 25 nM, 31 nM and 47 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAE684 (NVP-TAE684),761439-42-3,TAE684 is a potent and selective ALK inhibitor with IC50 of 3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BI 2536,755038-02-9,BI 2536 is a potent Plk1 inhibitor with IC50 of 0.83 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Varespladib (LY315920),172732-68-2,LY315920 (Varespladib) is a potent and selective secretory phospholipase A2 (sPLA) inhibitor with IC50 of 7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Foretinib (GSK1363089, XL880),849217-64-7,XL880 (GSK1363089, EXEL-2880) is an ATP-competitive inhibitor of MET and KDR with IC50 of 0.4 nM and 0.9 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SGX-523,1022150-57-7,SGX-523 is a selective Met inhibitor with IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK690693,937174-76-0,GSK690693 is a pan-Akt inhibitor targeting Akt1, Akt2 and Akt3 with IC50 of 2 nM, 13 nM, and 9 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ-38877605,943540-75-8,JNJ-38877605 is an ATP-competitive inhibitor of c-Met with IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Odanacatib (MK 0822),603139-19-1,Odanacatib (MK 0822) is a potent, selective, and neutral inhibitor of human and rabbit cathepsin K with IC50 of 0.2 nM and 1 nM , respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD 0332991 (Palbociclib) HCl,827022-32-2,PD 0332991 is a highly selective inhibitor of CDK4/cyclin D1 and CDK6/cyclin D2 with IC50 of 11 nM and 16 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Triciribine (Triciribine phosphate),35943-35-2,Triciribine (TCN, API-2) is a DNA synthesis inhibitor and also inhibits Akt and HIV-1 with IC50 of 130 nM and 20 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
XL147,956958-53-5,XL147 (SAR245408) is a selective and reversible class I PI3K inhibitor for wild type and mutant p110α with IC50 of 40 nM and 40 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
XL-184 (Cabozantinib),849217-68-1,XL184 (Cabozantinib) is a potent VEGFR2 inhibitor with IC50 of 0.035 nM and also inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, and AXL with IC50 of 1.3 nM, 4 nM, 4.6 nM, 12 nM/11.3 nM/6 nM, 14.3 nM and 7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Everolimus (RAD001),159351-69-6,Everolimus (RAD001) is an mTOR inhibitor of FKBP12 with IC50 of 1.6-2.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TW-37,877877-35-5,TW-37 is a novel nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 with Ki of 0.29 μM, 1.11 μM and 0.26 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mocetinostat (MGCD0103),726169-73-9,MGCD0103 (Mocetinostat) is a potent HDAC inhibitor for HDAC1, HDAC2 and HDAC3 with IC50 of 0.15 μM, 0.29 μM and 1.66 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Abiraterone (CB-7598),154229-19-3,Abiraterone (CB-7598) is a potent CYP17 inhibitor with IC50 of 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SRT1720,1001645-58-4,SRT1720 is a selective SIRT1 activator with EC1.5 of 0.16 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
YM155,781661-94-7,YM155 is a potent IAP (inhibitor of apoptosis protein via E3 ubiquitin ligase) inhibitor for survivin with IC50 of 0.54 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
INO-1001,3544-24-9,INO-1001 is a potent inhibitor of PARP with IC50 of 50 nM and a mediator of oxidant-induced myocyte dysfunction during reperfusion.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MLN8237 (Alisertib),1028486-01-2,MLN8237 (Alisertib) is a selective Aurora A inhibitor with IC50 of 1.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT9283,896466-04-9,AT9283 is a potent pan-Aurora inhibitor for Aurora A, Aurora B, JAK3, JAK2 and Abl with IC50 of 3 nM, 3 nM, 1.1 nM, 1.2 nM and 4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pemetrexed (Alimta),150399-23-8,Pemetrexed disodium (Alimta) is a novel antifolate and antimetabolite for TS, DHFR and GARFT with Ki of 1.3 nM, 7.2 nM and 65 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Brivanib alaninate (BMS-582664),649735-63-7,BMS-582664 is an oral VEGFR/FGFR inhibitor for VEGFR2, Flk1, VEGFR1 and FGFR1 with IC50 of 25 nM, 89 nM, 380 nM and 148 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ADL5859 HCl,850173-95-4,ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Andarine (GTX-007),401900-40-1,Andarine (GTX-007) is a selective nonsteroidal androgen receptor (AR) agonist with Ki of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
17-AAG (Tanespimycin),75747-14-7,17-AAG (Tanespimycin) is a potent HSP90 inhibitor with IC50of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
17-DMAG HCl (Alvespimycin),467214-21-7,17-DMAG (Alvespimycin, KOS-1022, NSC 707545) is a potent HSP90 inhibitor with IC50 of 62 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AG-490,133550-30-8 ,AG-490 (Tyrphostin B42) is an inhibitor of EGFR, ErbB2 and JAK2 with IC50 of 0.1 μM, 13.5 μM, and ~10 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ivacaftor (VX-770),873054-44-5,Ivacaftor (VX-770, Kalydeco) is a potentiator of CFTR targeting G551D-CFTR and F508del-CFTR with EC50 of 100 nM and 25 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SNS-032 (BMS-387032),345627-80-7,SNS-032 is a novel, potent and selective CDK inhibitor of CDK2, CDK7 and CDK9 with IC50 of 38 nM, 62 nM and 4 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cyclopamine,4449-51-8,Cyclopamine is a specific Hedgehog (Hh) signaling pathway antagonist of Smoothened (Smo) with IC50 of 46 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Barasertib (AZD1152-HQPA),722544-51-6,AZD1152-HQPA (Barasertib) is a highly selective Aurora B inhibitor with IC50 of 0.37 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Docetaxel (Taxotere),114977-28-5,Docetaxel, an analog of taxol, is an inhibitor of depolymerisation of microtubules through binding to stabilized microtubules.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gemcitabine HCl (Gemzar),122111-03-9,Gemcitabine Hydrochloride (Gemzar) is a DNA synthesis inhibitor with IC50 of 50 nM, 40 nM, 18 nM and 12 nM in PANC1, MIAPaCa2, BxPC3 and Capan2 cells, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Paclitaxel (Taxol),33069-62-4,Paclitaxel (Taxol, Onxol, Nov-Onxol) is a microtubule polymer stabilizer with IC50 of 0.1 pM in human endothelial cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PLX-4720,918505-84-7,PLX-4720 is a potent and selective inhibitor of B-RafV600E and c-Raf-1Y340D/Y341D with IC50 of 13 nM and 6.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Roscovitine (Seliciclib, CYC202) ,186692-46-6 ,Roscovitine (Seliciclib, CYC202, R-roscovitine) is a potent and selective CDK inhibitor for Cdc2/cyclin B, CDK2/cyclin A, CDK2/cyclin E and CDK5/p53 with IC50 of 0.65 μM, 0.7 μM, 0.7 μM and 0.16 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SNS-314 Mesylate,1146618-41-8,SNS-314 Mesylate is a potent and selective inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 9 nM, 31 nM, and 3.4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NSC 74859 (S3I-201),501919-59-1,S3I-201 (NSC 74859) is a Stat3 inhibitor with IC50 of 86 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Capecitabine (Xeloda),154361-50-9,Capecitabine is a tumor-selective fluoropyrimidine carbamate which achieves higher intratumoral 5-FU level with lower toxicity than 5-FU.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-8245,1030612-90-8,MK-8245 is an inhibitor of stearoyl-CoA desaturase (SCD) which targets the liver with IC50 of 1 nM for human SCD1 and 3 nM for both rat SCD1 and mouse SCD1.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ganetespib (STA-9090),888216-25-9,Ganetespib is an HSP90 inhibitor with IC50 of 4 nM in OSA 8 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TRAM-34,289905-88-0,TRAM-34 is a selective and potent inhibitor of the intermediate-conductance Ca2+-activated K+ channel (IKCa1, KCa3.1) with Kd of 20 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT13387,912999-49-6,AT13387 is a selective potent Hsp90 inhibitor with IC50 of 18 nM in A375 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
E7080 (Lenvatinib),417716-92-8,E7080 (Lenvatinib) is a multi-target inhibitor of VEGFR2 and VEGFR3 with IC50 of 4 nM and 5.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ABT-751,141430-65-1,ABT-751 (E7010) binds to the colchicine site on β-tubulin and inhibits polymerization of microtubules.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cisplatin,15663-27-1,Cisplatin is an inorganic and water-soluble platinum complex, which is able to inhibit DNA synthesis by conforming DNA adducts. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CP-724714,537705-08-1,CP-724,714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM and also inhibits EGFR with IC50 of 6.4 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Valproic acid sodium salt (Sodium valproate),1069-66-5,Valproic acid sodium salt (Sodium valproate) is a HDAC inhibitor with IC50 of 0.4 mM and also inhibits GABA-transaminase or succinic
semialdehyde dehydrogenase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
TGX-221,663619-89-4,TGX-221 is a potent, selective PI3K inhibitor for p110β with IC50 of 8.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WZ3146,1214265-56-1,WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM and 2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CYC116,693228-63-6,CYC116 is a potent inhibitor of Aurora A/B and VEGFR with Ki of 8.0 nM/9.2 nM and 44 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ 26854165 (Serdemetan),881202-45-5,JNJ 26854165 (Serdemetan) is an orally bioavailable HDM2 (an E3 ligase) antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WZ4002,1213269-23-8,WZ4002 is a novel, mutant-selective EGFR inhibitor for EGFRL858R and EGFRL858R/T790M with IC50 of 2 nM and 8 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ostarine (MK-2866),841205-47-8,Ostarine (GTx-024, MK-2866, Enobosarm, S-22) is a selective androgen receptor modulator (SARM) with Ki of 3.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIIB021,848695-25-0,BIIB021 is a novel inhibitor of HSP90 with Ki and EC50 of 1.7 nM and 38 nM, respectivley.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD98059,167869-21-8,PD98059 is a non-ATP competitive MEK inhibitor with IC50 of 2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Regorafenib (BAY 73-4506),755037-03-7,Regorafenib (BAY 73-4506, Fluoro-Sorafenib) is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WZ8040,1214265-57-2,WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
XAV-939,284028-89-3,XAV-939 is a selective Wnt β-catenin-mediated transcription inhibitor for TNKS1 and TNKS2 with IC50 of 11 nM and 4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ENMD-2076,934353-76-1,ENMD-2076 is a selective inhibitor of Aurora A and Aurora B with IC50 of 14 nM and 350 nM and also inhibits Flt3, Flt4 and VEGFR2 with IC50 of 1.86 nM/15.9 nM and 58.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Danoprevir,850876-88-9,Danoprevir is a peptidomimetic inhibitor of the NS3/4A protease of hepatitis C virus (HCV) with IC50 of 0.2-3.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ritonavir,155213-67-5,Ritonavir is an inhibitor of HIV protease used to treat HIV infection and AIDS.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIBR 1532,321674-73-1,BIBR 1532 is a potent and selective telomerase inhibitor with IC50 of 100 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PIK-90,677338-12-4,PIK-90 is a potent and cell permeable inhibitor of p110α, p110β, p110γ and p110δ with IC50 of 11 nM, 350 nM, 18 nM and 58 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Anastrozole,120511-73-1,Anastrozole inhibits the enzyme aromatase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aprepitant (MK-0869),170729-80-3,Substance P antagonists (SPA). ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bicalutamide (Casodex),90357-06-5,Bicalutamide (Casodex, Cosudex, Calutide, Kalumid) is an androgen receptor (AR) antagonist with IC50 of 0.16 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fulvestrant (Faslodex),129453-61-8,Fulvestrant is an estrogen receptor (ER) antagonist with IC50 of 0.094 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Raltitrexed (Tomudex),112887-68-0,Raltitrexed (Tomudex) is a thymidylate synthase inhibitor with an IC50 of 9 nM for the inhibition of L1210 cell growth.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Thalidomide,50-35-1,Thalidomide was introduced as a sedative drug,immunomodulatory agent and also is investigated for treating symptoms of many cancers.Thalidomide inhibits an E3 ubiquitin ligase， which is a CRBN-DDB1-Cul4A complex.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CUDC-101,1012054-59-9,CUDC-101 is a potent multi-target inhibitor targeting HDAC, EGFR and HER2 with IC50 of 4.4 nM, 2.4 nM, and 15.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-700 (Orteronel),426219-18-3,TAK-700 (Orteronel) is a potent and highly selective rat and human 17,20-lyase inhibitor with IC50 of 54 nM and 38 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Exemestane,107868-30-4,Exemestane is an aromatase inhibitor, inhibits human placental and rat ovarian aromatase with IC50 of 30 nM and 40 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Finasteride,98319-26-7,Finasteride is an inhibitor of steroid Type II 5α-reductase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Irinotecan,97682-44-5,Irinotecan (Camptosar, Campto, CPT-11) is a topoisomerase I inhibitor for LoVo cells and HT-29 cells with IC50 of 15.8 μM and 5.17 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cladribine,4291-63-8,Cladribine (Leustatin, Litak, 2CDA) is an adenosine deaminase inhibitor for U266, RPMI8226, and MM1.S cells with IC50 of approximately 2.43 μM, 0.75 μM, and 0.18 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Decitabine,2353-33-5,Decitabine is a potent inhibitor of DNA methylation with IC50 of 438 nM and 4.38 nM in HL-60 and KG1a cells, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dimesna,16208-51-8,Dimesna is an uroprotective agent used to decrease urotoxicity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dutasteride,164656-23-9,Dutasteride is a 5-alpha-reductase inhibitor ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PIK-75,372196-77-5,PIK-75 is a selective and competitive inhibitor of p110α with IC50 of 5.8 nM and also potently inhibits DNA-PK with IC50 of 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bisoprolol,104344-23-2,Bisoprolol is a selective type β1 adrenergic receptor blocker,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Tivozanib (AV-951),475108-18-0,AV-951 (Tivozanib, KRN-951) is a potent and selective VEGFR inhibitor for VEGFR1/2/3 with IC50 of 0.21 nM/0.16 nM/0.24 nM and also inhibits PDGFR and c-Kit with IC50 of 1.72 nM and 1.63 nM, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Doxorubicin (Adriamycin),25316-40-9,Doxorubicin (Adriamycin) is an antibiotic agent that inhibits DNA topoisomerase II and induces DNA damage and apoptosis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Adrucil (Fluorouracil),51-21-8,Adrucil (Fluorouracil) is an DNA/RNA synthesis inhibitor, which interrupts nucleotide synthetic by inhibiting thymidylate synthase (TS).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Abitrexate (Methotrexate),59-05-2,Abitrexate (Methotrexate) is an antimetabolite and antifolate agent with antineoplastic and immunosuppressant activities.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bendamustine HCL,3543-75-7,Bendamustine HCL (Ribomustin, Treanda, SDX-105) is a DNA-damaging agent with IC50 of 50 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nelarabine (Arranon),121032-29-9,Nelarabine (Arranon, 506U78) is a purine nucleoside analog and DNA synthesis inhibitor with IC50 from 0.067-2.15 μM in tumor cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bleomycin sulfate,9041-93-4,Bleomycin sulfate (Blenoxane) is a glycopeptide antibiotic and an anticancer agent for squamous cell carcinomas (SCC) with IC50 of 4 nM in UT-SCC-19A cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carboplatin,41575-94-4,Carboplatin is a DNA synthesis inhibitor by binding to DNA and interfering with the cell's repair mechanism.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PFI-1,1403764-72-6,PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clafen (Cyclophosphamide),50-18-0,This agent inhibited cell proliferation of NCI-H727 with IC50 at 9.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clofarabine,123318-82-1,Clofarabine inhibits the enzymatic activities of ribonucleotide reductase (IC50 = 65 nM) and DNA polymerase,HPLC 99%, NMR, LCMS is OK, stock more than 20g
YM201636,371942-69-7,YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
OSI-930,728033-96-3,OSI-930 is a potent inhibitor of Kit, KDR, Flt, CSF-1R, c-Raf and Lck with IC50 of 80 nM, 9 nM, 8 nM, 15 nM, 41 nM and 22 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dacarbazine (DTIC-Dome),4342-03-4,Dacarbazine(DTIC-Dome) is an antineoplastic chemotherapy drug used in the treatment of various cancers.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Epirubicin HCl,56390-09-1,Epirubicin HCl, a semisynthetic L-arabino derivative of doxorubicin, is an antineoplastic agent by inhibiting Topoisomerase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oxaliplatin (Eloxatin),61825-94-3,Oxaliplatin inhibits DNA synthesis by conforming DNA adducts.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Etoposide (VP-16),33419-42-0,Etoposide is a semisynthetic derivative of podophyllotoxin, which inhibits DNA synthesis via topoisomerase II  inhibition activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ku-0063794,938440-64-3,KU-0063794 is a potent and highly specific mTOR inhibitor for both mTORC1 and mTORC2 with IC50 ~10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Evista (Raloxifene HCl),82640-04-8,Raloxifene is estrogen antagonists, inhibits human cytosolic aldehyde oxidase-catalyzed phthalazine oxidation activity with IC50 of 5.7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Idarubicin HCl,57852-57-0,Idarubicin HCl (Idamycin, Zavedos, 4-demethoxydaunorubicin) is a hydrochloride salt form of Idarubicin which is an anthracycline antibiotic and a DNA topoisomerase II (topo II) inhibitor for MCF-7 cells with IC50 of 3.3 ng/mL.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fludarabine Phosphate (Fludara),75607-67-9,Fludarabine Phosphate is an analogue of adenosine and deoxyadenosine, which is able to compete with dATP for incorporation into DNA and inhibit DNA synthesis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Topotecan HCl,119413-54-6,Topotecan (Hycamtin, NSC 609699) is a topoisomerase I inhibitor for MCF-7 Luc cells and DU-145 Luc cells with IC50 of 13 nM and 2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
2-Methoxyestradiol,362-07-2,2-Methoxyestradiol is a tubulin polymerization inhibitor and also decreases HIF-1 activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AG-1024 ,65678-07-1,AG-1024 (Tyrphostin) is a specific IGF-1R and IR inhibitor with IC50 of 0.4 μM and 0.1 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Letrozole,112809-51-5,Letrozole is a third generation inhibitor of aromatase with IC50 of 0.07-20 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Temozolomide,85622-93-1,Methazolastone (Temozolomide, Temodar, Temodal) is a DNA damage inducer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vincristine,2068-78-2,Vincristine is an inhibitor of polymerization of microtubules by binding to tubulin with IC50 of 32 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Agomelatine,138112-76-2,Agomelatine is classified as a norepinephrine-dopamine disinhibitor (NDDI) due to its antagonism of the 5-HT2C receptor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amuvatinib (MP-470),850879-09-3,MP-470 (Amuvatinib) is a potent and multi-targeted inhibitor of c-KitD816H, PDGFαV561D and Flt3D835Y with IC50 of 10 nM, 40 nM and 81 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vinblastine,57-22-7,Vinblastine inhibits microtubule formation and supresses nAChR activity with IC50 of 8.9 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ-7706621,443797-96-4,JNJ-7706621 is a potent and multi-target inhibitor for CDK1/cyclin B, CDK2/cyclin A, CDK2/cyclin E, Aurora A and Aurora B with IC50 of 9 nM, 4 nM, 3 nM, 11 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MDV3100 (Enzalutamide),915087-33-1,MDV3100 is an androgen-receptor (AR) antagonist with IC50 of 36 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dienogest,65928-58-7,Dienogest is an orally active synthetic progesterone (or progestin). ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rufinamide (Banzel),106308-44-5,Rufinamide, a triazole derivative, is an anticonvulsant medication.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Posaconazole,171228-49-2,Posaconazole (Noxafil) is a sterol C14ɑ demethylase inhibitor with an IC50 of 0.25 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Prasugrel (Effient),150322-43-3,A novel platelet inhibitor ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ramelteon (TAK-375),196597-26-9,Ramelteon (TAK-375) is a novel melatonin receptor agonist for human MT1 and MT2 receptors and chick forebrain melatonin receptors with Ki of 14 pM, 112 pM and 23.1 pM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AMG-073 HCl (Cinacalcet HCl),364782-34-3,AMG-073 HCl (Cinacalcet hydrochloride) represents a new class of compounds for the treatment of hyperparathyroidism.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Celecoxib,169590-42-5,Celecoxib is a selective COX-2 inhibitor with IC50 of 40 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS-708163 (Avagacestat),1146699-66-2,BMS-708163 is a potent, selective γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD173074,219580-11-7,PD173074 is a potent FGFR1 inhibitor with IC50 of ~25 nM and also inhibits VEGFR2 with IC50 of 100-200 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WYE-354,1062169-56-5,WYE-354 is a potent, specific and ATP-competitive inhibitor of mTOR with IC50 of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vemurafenib (PLX4032),918504-65-1,PLX4032 (Vemurafenib, RG7204, Zelboraf, RO5185426) is a novel and potent inhibitor of B-RafV600E with IC50 of 31 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
IC-87114,371242-69-2,IC-87114 is a selective inhibitor of PI3Kδ with IC50 of 0.5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BX-795,702675-74-9,BX795 is a potent and specific TBK1, IKKε and PDK-1 inhibitor with IC50 of 6 nM, 41 nM and 111 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BX-912,702674-56-4,BX912 is a selective potent PDK1 inhibitor with IC50 of 12 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amisulpride,71675-85-9,Amisulpride is an atypical antipsychotic used to treat psychosis in schizophrenia and episodes of mania in bipolar disorder.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aniracetam,72432-10-1,Aniracetam is a nootropics and neuroprotective drug.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Asenapine,85650-56-2,Asenapine ihibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Benazepril HCl,86541-74-4,Benazepril is a medication used to treat high blood pressure.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Biperiden HCl,1235-82-1,Biperiden is an antiparkinsonian agent of the anticholinergic type.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Camptothecin,7689-03-4,Camptothecin (Camptohecine, 20-(S)-Camptothecin, CPT, NSC100880) is a specific inhibitor of DNA topoisomerase I (Topo I) with IC50 of 0.68 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carmofur,61422-45-5,Carmofur (INN) is a pyrimidine analogue used as an antineoplastic agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Celastrol,34157-83-0,Celastrol is a potent proteasome inhibitor for the chymotrypsin-like activity of a purified 20S proteasome with IC50 of 2.5 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cetirizine DiHCl,83881-52-1,Cetirizine Dihydrochloride is an antihistamine.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cilnidipine,132203-70-4,Cilnidipine is a calcium channel blocker.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cilostazol,73963-72-1,Cilostazol is a potent cyclic nucleotide phosphodiesterase type 3 (PDE3) inhibitor with IC50 of 0.2 μM and inhibitor of adenosine uptake.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Epothilone A,152044-53-6,Epothilone A is a Taxol-like microtubule-stabilizing agent with EC0.01 of 2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Floxuridine (Fludara),50-91-9,Floxuridine (Fludara) is a prodrugs of floxuridine and an oncology agent with an GI50 of 5.1 μM for the inhibition of MDCK/PEPT1.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ftorafur,17902-23-7,Ftorafur is a substance being used in the treatment of some types of cancer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ifosfamide,3778-73-2,Ifosfamide is a nitrogen mustard alkylating agent used in the treatment of cancer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Megestrol Acetate,595-33-5,Megestrol Acetate is a synthetic progesteronal agent with an IC50 of 260 μM for the inhibition of HegG2.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mercaptopurine,50-44-2,Mercaptopurine is a widely used antileukemic agent and immunosuppressive drug that inhibits de novo purine synthesis through incorporation of thiopurine methyltransferase metabolites into DNA and RNA.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zoledronic Acid (Zoledronate),118072-93-8,A potent nitrogen-containing bisphosphonates.It inhibited proliferation of human foetal osteoblastic cell line (hFOB) with an IC50 of 40 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ki16425,355025-24-0 ,Ki16425 is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AMG-208,1002304-34-8 ,AMG-208 is a highly selective c-Met inhibitor with IC50 of 9.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Costunolide,553-21-9,Costunolide inhibits FPTase with IC50 of 20 μM and also inhibits telomerase with IC50 of 90 μM and 65 μM in MCF-7 and MDA-MB-231 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dexamethasone,50-02-2,Dexamethasone is an anti-inflammatory and immunosuppressant.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Doxazosin mesylate,77883-43-3,Doxazosin mesylate is an alpha-1 adrenergic receptor blocker.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ellagic acid,476-66-4,Ellagic acid has antiproliferative and antioxidant property.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Etodolac (Lodine),41340-25-4,Etodolac (Lodine) is a COX inhibitor with an IC50 of 53.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Etomidate,33125-97-2,Etomidate is a GABAA receptors agonist at GABAA receptors.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flumazenil,78755-81-4,Flumazenil is a benzodiazepine antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fluoxetine  HCl,56296-78-7,Fluoxetine  HCl is an antidepressant of the selective serotonin reuptake inhibitor (SSRI)class.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flupirtine maleate,75507-68-5,Flupirtine maleate is the salt form of Flupirtine, which is a non-opioid, centrally acting analgesia, muscle relaxation and neuroprotection.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fluvoxamine maleate,61718-82-9,Fluvoxamine maleate is a selective serotonin (5-HT) reuptake inhibitor (SSRI).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gabapentin HCl,60142-95-2,Gabapentin Hydrochloride is a GABA analogue.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Galanthamine HBr,1953-04-4,Galanthamine (Razadyne, Reminyl) is an AChE inhibitor with IC50 of 14 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Genistein,446-72-0 ,Genistein, a phytoestrogen found in soy products, is a highly specific inhibitor of protein tyrosine kinase (PTK)  which blocks the mitogenic effect mediated by EGF on NIH-3T3 cells with IC50 of 12μM or by insulin with IC50 of 19 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Glimepiride,93479-97-1,Glimepiride is a medium-to-long acting sulfonylurea anti-diabetic compound with an ED50 of 182 μg/kg.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Granisetron HCl,107007-99-8,Granisetron HCl is a serotonin 5-HT3 receptor antagonist,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TG100-115,677297-51-7,TG100-115 is a potent and dual selective inhibitor for PI3Kγ and PI3Kδ with IC50 of 83 nM and 235 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ketoconazole,65277-42-1,Ketoconazole inhibits cyclosporine oxidase and testosterone 6 beta-hydroxylase with IC50 of 0.19 mM and 0.22 mM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lansoprazole,103577-45-3,Lansoprazole is a proton-pump inhibitor (PPI) which prevents the stomach from producing gastric acid.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lidocaine (Alphacaine),137-58-6,Lidocaine (Alphacaine) is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Loratadine,79794-75-5,Loratadine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Losartan potassium,124750-99-8,Losartan is an angiotensin II receptor antagonist, competes with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1059615,958852-01-2,GSK1059615 is a novel and dual inhibitor of PI3Kα, PI3Kβ, PI3Kδ, PI3Kγ and mTOR with IC50 of 0.4 nM, 0.6 nM, 2 nM, 5 nM and 12 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MGCD-265,875337-44-3,MGCD-265 is a potent, multi-target and ATP-competitive inhibitor of c-Met, VEGFR1, VEGFR2, VEGFR3, Ron, and Tie2 with IC50 of 1 nM, 3 nM, 3 nM, 4 nM, 2 nM and 7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rigosertib (ON-01910),1225497-78-8,Rigosertib (Estybon, Novonex, ON-01910) is a non-ATP-competitive inhibitor of PLK1 (Polo-like kinase 1) with IC50 of 9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ki8751,228559-41-9,Ki8751 is a potent and selective inhibitor of VEGFR2, PDGFRα and c-Kit with IC50 of 0.9 nM, 67 nM and 40 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Epothilone B (EPO906),152044-54-7,Epothilone B is a Taxol-like microtubule-stabilizing agent with EC0.01 of 1.8 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS-707035,729607-74-3,BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amonafide,69408-81-7,Amonafide (NSC-308847) is a selective topoisomerase II inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dorzolamide HCl,130693-82-2,Dorzolamide HCl is a carbonic anhydrase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gestodene,60282-87-3,Gestodene is a progestogen hormonal contraceptive.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Drospirenone,67392-87-4,Drospirenone is a synthetic progestin that is an analog to spironolactone.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ruxolitinib (INCB018424),941678-49-5,INCB018424 is a JAK family inhibitor for JAK1, JAK2 and JAK3 with IC50 of 2.7 nM, 4.5 nM and 322 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Isotretinoin,4759-48-2,It was developed to be used as a chemotherapy medication for the treatment of brain cancer, pancreatic cancer and more.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lopinavir (ABT-378),192725-17-0,Lopinavir (ABT-378) is a potent HIV protease inhibitor with Ki of 1.3 pM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mianserin HCl,21535-47-7,Mianserin is a psychoactive agent of the tetracyclic antidepressant.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Minoxidil,38304-91-5,Minoxidil is a vasodilator medication known for its ability to slow or stop hair loss and promote hair regrowth.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mizoribine (Bredinin),50924-49-7,Mizoribine (Bredinin) is an imidazole nucleoside and an immunosuppressive agent with an IC50 of approximately 100 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mosapride citrate,112885-42-4,Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nafamostat mesylate,82956-11-4,Nafamostat is an anticoagulant.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naftopidil DiHCl,57149-08-3,Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Omeprazole (Prilosec),73590-58-6,Omeprazole(Prilosec) is a proton pump inhibitor used in the treatment of dyspepsia.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ondansetron HCl (Zofran),99614-01-4,Ondansetron is a serotonin 5-HT3 receptor antagonist. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oxcarbazepine,28721-07-5,Oxcarbazepine inhibits the binding of [3H]BTX to sodium channels with IC50 of 160 μM and also inhibits the influx of 22Na+ into rat brain synaptosomes with IC50 about 100 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pelitinib (EKB-569),257933-82-7,Pelitinib (EKB-569) is a potent EGFR inhibitor with IC50 of 38.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Resveratrol,501-36-0,Resveratrol is a phytoalexin produced naturally by several plants with anti-cancer, anti-inflammatory, blood-sugar-lowering and other beneficial cardiovascular effects.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rocuronium bromide,119302-91-9,Rocuronium is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Stavudine,3056-17-5,Stavudine is a nucleoside analog reverse transcriptase inhibitor (NARTI) active against HIV. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tenofovir Disoproxil Fumarate,202138-50-9,Tenofovir disoproxil fumarate belongs to nucleotide analogue reverse transcriptase inhibitors (nRTIs). ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tenofovir (Viread),147127-20-6,Tenofovir blocks reverse transcriptase and hepatitis B virus infections.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Trilostane,13647-35-3,Trilostane is an inhibitor of 3 β-hydroxysteroid dehydrogenase used in the treatment of Cushing’s syndrome.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Alfuzosin HCl (Uroxatral),81403-68-1,Alfuzosin(Uroxatral) is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AS-605240,648450-29-7,AS-605240 is a novel, potent and selective PI3Kγ inhibitor with IC50 of 8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clopidogrel (Plavix),120202-66-6,Clopidogrel (Plavix) is an oral, thienopyridine class antiplatelet agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Staurosporine,62996-74-1,Staurosporine (AM-2282) is a potent PKC inhibitor with IC50 of 2.7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Droxinostat,99873-43-5,Droxinostat (CMH, 5809354) is a selective inhibitor of HDAC3, HDAC6 and HDAC8 with IC50 of 16.9 μM, 2.47μM and 1.46 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ranolazine 2HCl,95635-56-6,Ranolazine(Ranexa), is an antianginal medication.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Repaglinide,135062-02-1,Repaglinide is for the treatment of type II diabetes.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rolipram,61413-54-5,Rolipram is a PDE4-inhibitor and an anti-inflammatory agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sildenafil citrate,171599-83-0,Sildenafil citrate is an agent used to treat erectile dysfunction and pulmonary arterial hypertension (PAH).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sumatriptan succinate,103628-48-4,Sumatriptan succinate is a triptan sulfa drug containing a sulfonamide group for the treatment of migraine headaches.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tianeptine sodium,30123-17-2,Tianeptine is a selective serotonin reuptake enhancer (SSRE) compound used for treating major depressive episodes.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tizanidine HCl,64461-82-1,Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Topiramate,97240-79-4,Topiramate is an anticonvulsant compound.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Varenicline tartrate,375815-87-5,Varenicline is a prescription medication used to treat smoking addiction.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Venlafaxine,99300-78-4,Venlafaxine is an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Voriconazole,137234-62-9,Voriconazole (VFEND) is a triazole antifungal medication that is generally used to treat serious, invasive fungal infections.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zileuton,111406-87-2,Zileuton (ZYFLO) is an orally active inhibitor of 5-lipoxygenase, and thus inhibits leukotrienes (LTB4, LTC4, LTD4, and LTE4) formation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aurora A Inhibitor I,1158838-45-9,Aurora A Inhibitor I is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ispinesib (SB-715992),336113-53-2,Ispinesib (SB-715992, CK0238273) is a potent, specific and reversible inhibitor of KSP (HsEg5) with Ki of 1.7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tipifarnib (Zarnestra),192185-72-1,Tipifarnib (Zarnestra, R115777) is a potent and specific farnesyltransferase (FTase) inhibitor with IC50 of 0.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PHA-680632,398493-79-3,PHA-680632 is potent inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 27 nM, 135 nM and 120 nM, repectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cilomilast (SB-207499),153259-65-5,Cilomilast (SB-207499) is a potent LPDE4 and HPDE4 inhibitor with IC50 of 100 nM and 120 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zibotentan (ZD4054),186497-07-4,Zibotentan (ZD4054) is a specific Endothelin A (ETA) antagonist with IC50 of 21 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Atazanavir sulfate,229975-97-7,Atazanavir is a HIV protease inhibitor with Ki of 2.66 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Thiazovivin,1226056-71-8,Thiazovivin (Tzv) is a novel ROCK inhibitor with IC50 of ~0.5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SP600125,129-56-6,SP600125 is a broad-spectrum JNK inhibitor for JNK1, JNK2 and JNK3 with IC50 of 40 nM, 40 nM and 90 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ofloxacin (Floxin),82419-36-1,Ofloxacin is a synthetic broad-spectrum antimicrobial agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Moxifloxacin HCl,186826-86-8,Moxifloxacin(Avelox, Avalox) is a fourth generation synthetic fluoroquinolone antibacterial agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Alfacalcidol,41294-56-8,Alfacalcidol is a non-selective VDR activator medication.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TSU-68 (SU6668),252916-29-3,TSU-68  (SU6668, Orantinib) is a potent inhibitor of Flk-1/KDR, FGFR1 and PDGFRβ with Ki of 2.1 μM, 1.2 μM, and 8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Safinamide Mesylate (FCE28073),202825-46-5,Safinamide Mesylate is mesylate salt of Safinamide, which selectively and reversibly inhibits MAO-B with IC50 of 0.45 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK429286A,864082-47-3,GSK429286A is a selective inhibitor of ROCK1 and ROCK2 with IC50 of 14 nM and 63 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AS703026 (pimasertib),1236699-92-5,AS703026 is a highly selective and potent non-competitive inhibitor of MEK1/2 with IC50 of 5-11 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 525334,356559-20-1,SB 525334 is a potent and selective inhibitor of TGF-β1 (ALK5) with IC50 of 14.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Oligomycin A,579-13-5,Oligomycin A is a specific inhibitor of complex V (ATP synthase) of the electron transport chain.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
VX-222,1026785-55-6,VX-222 (VCH-222) is a novel, potent and selective inhibitor of HCV polymerase with IC50 of 0.94-1.2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY335979 (Zosuquidar 3HCl),167465-36-3,LY335979 (Zosuquidar) is a potent modulator of P-glycoprotein-mediated multidrug resistance with Ki of 60 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Daclatasvir （BMS-790052）,1009119-64-5,BMS-790052 is a highly selective inhibitor of HCV NS5A with EC50 of 9-50 pM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MC1568,852475-26-4,MC1568 is a selective HDAC inhibitor with IC50 of 220 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
HMN-214,173529-46-9 ,HMN-214 (IVX-214) is a potent inhibitor of Polo-like kinase (Plk)1 with IC50 of 118 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AEE788 (NVP-AEE788),497839-62-0,AEE788 is a potent inhibitor of EGFR and HER2/ErbB2 with IC50 of 2 nM and 6 nM and also inhibits VEGFR2 and Flt with IC50 of 77 nM and 59 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PHA-793887,718630-59-2,PHA-793887 is a novel and potent inhibitor of CDK2, CDK5 and CDK7 with IC50 of 8 nM, 5 nM and 10 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naratriptan HCl,143388-64-1,Naratriptan (Amerge) is a triptan agent that is used for the treatment of migraine headaches.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PIK-93,593960-11-3,PIK-93 is a novel and potent inhibitor of PI3Kγ and PI4KIIIβ with IC50 of 16 nM and 19 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ponatinib (AP24534),943319-70-8,AP24534 is a novel, potent multi-target inhibitor of Abl, PDGFRα, VEGFR2, FGFR1 and Src with IC50 of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM and 5.4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fludarabine (Fludara),21679-14-1,Fludarabine (Fludara, F-ara-A, NSC 118218) is a STAT1 activation inhibitor and a DNA synthesis inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2228820,862507-23-1,LY2228820 is a novel and potent inhibitor of p38 MAPK with IC50 of 7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pralatrexate (Folotyn),146464-95-1,Pralatrexate(Folotyn) is an antifolate, and structurally a folate analog. Its IC50 is < 300 nM in some cell lines.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-BEP800,847559-80-2,NVP-BEP800 is a novel, fully synthetic HSP90β inhibitor with IC50 of 58 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mycophenolate mofetil (CellCept),128794-94-5,Mycophenolate mofetil is a non-competitive, selective and reversible inhibitor of inosine monophosphate dehydrogenase I/II with IC50 of 39 nM and 27 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dyphylline (Dilor),479-18-5,Dyphylline(Dilor, Lufyllin, diprophylline) is a xanthine derivative with bronchodilator and vasodilator effects.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Perindopril Erbumine (Aceon),107133-36-8,Perindopril Erbumine (Aceon) is a potent ACE) inhibitor with IC50 of 1.05 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Irbesartan (Avapro),138402-11-6,Irbesartan (Avapro, SR-47436, BMS-186295) is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist with IC50 of 1.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tadalafil (Cialis),171596-29-5,Tadalafil is a PDE-5 inhibitor with IC50 of 1.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB939 (Pracinostat),929016-96-6,SB939 is a potent HDAC inhibitor with IC50 of 40-140 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ibuprofen Lysine (NeoProfen),57469-77-9,Ibuprofen Lysine(Motrin) is a non-steroidal anti-inflammatory drug.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CCT129202,942947-93-5,CCT129202 is an ATP-competitive pan-Aurora inhibitor for Aurora A, Aurora B and Aurora C with IC50 of 0.042 μM, 0.198 μM and 0.227 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tosedostat (CHR2797),238750-77-1,CHR-2797 is an aminopeptidase inhibitor for LAP, PuSA and Aminopeptidase N with IC50 of 100 nM, 150 nM and 220 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
XL765 (SAR245409),1349796-36-6,XL765 is a dual inhibitor of mTOR/PI3k for mTOR, p110α, p110β, p110γ and p110δ with IC50 of 157 nM, 39 nM, 113 nM, 9 nM and 43 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT7519,844442-38-2,AT7519 is a novel multi-CDK inhibitor for CDK1/cyclin B, CDK2/Cyclin A, CDK3/Cyclin E, CDK4/Cyclin D1, CDK5/p35 and CDK6/Cyclin D3 with IC50 of 210 nM, 47 nM, 360 nM, 100 nM, 13 nM and 170 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-1775,955365-80-7,MK-1775 is a potent and selective Wee1 inhibitor with IC50 of 5.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Quizartinib (AC220),950769-58-1,AC220 (Quizartinib) is a potent and selective inhibitor of Flt3ITD and Fltwt with IC50 of 1.1 nM and 4.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2811376,1194044-20-6,LY2811376 is a non-peptidic BACE1 inhibitor with IC50 of 239 nM/249 nM and also decreases the Aβ secretion with EC50 of ~300 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hesperadin,422513-13-1,Hesperadin inhibits Aurora B and  T. brucei Aurora kinase-1 (TbAUK1) with IC50 of 250 nM and 40 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIX 02188,1094614-84-2,BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIX 02189,1094614-85-3,BIX02189 is a selective inhibitor of MEK5 with IC50 of 1.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD7762,860352-01-8,AZD7762 is a novel CHK1 and CHK2 inhibitor with IC50 of 5 nM and <10 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
R406 (free base),841290-80-0,R406 (free base) is a Syk inhibitor with IC50 of 41 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CP 673451,343787-29-1,CP 673451 is a potent PDGFR-β inhibitor with an IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
DMXAA (ASA404),117570-53-3,DMXAA (ASA404) is a vascular disrupting agents (VDA) and competitive inhibitor of DT-diaphorase with Ki of 20 μM and IC50 of 62.5 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Telaprevir (VX-950),402957-28-2,Telaprevir (VX-950) is an HCV NS3-4A serine protease inhibitor with IC50 of 0.35 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Saxagliptin (BMS-477118,Onglyza),361442-04-8,Saxagliptin (BMS-477118, Onglyza) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
EX 527,49843-98-3,EX 527 is a potent and selective SIRT1 inhibitor with IC50 of 38 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AM-1241,444912-48-5,AM-1241 is a selective CB2 agonist with Ki of 3.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB-408124,288150-92-5,SB-408124 (Tocris-1963) is a non-peptide antagonist for OX1 with Ki of 57 nM and  27 nM in both whole cell and membrane, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dapagliflozin,461432-26-8,Dapagliflozin is a potent and selective hSGLT2 inhibitor with EC50 of 1.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nebivolol (Bystolic),152520-56-4,Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pimobendan (Vetmedin),74150-27-9,Pimobendan is a selective inhibitor of PDE3 with IC50 of 0.32 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD8055,1009298-09-2,AZD8055 is a novel ATP-competitive inhibitor of mTOR with IC50 of 0.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PHT-427,1191951-57-1,PHT-427 is a dual Akt and PDPK1 inhibitor with Ki of 2.7 μM and 5.2 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KRN 633,286370-15-8,KRN 633 is an ATP-competitive inhibitor of VEGFR1/2/3 with IC50 of 170 nM/160 nM/125 nM and also inhibits PDGFRα/β with IC50 of 965 nM/9850 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT7867,857531-00-1,AT7867 is a potent ATP-competitive inhibitor of Akt1/2/3 and S6K with IC50 of 32 nM/17 n/47 nM and 85 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS 777607,1025720-94-8,BMS-777607 is a Met-related inhibitor for c-Met, Axl, Ron and Tyro3 with IC50 of 3.9 nM, 1.1 nM, 1.8 nM and 4.3 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VX-809,936727-05-8,VX-809 is a CFTR modulator with EC50 of 0.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pomalidomide,19171-19-8,Pomalidomide inhibits LPS-induced TNF-α release with IC50 of 13 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD318088,391210-00-7 ,PD318088 is a non-ATP competitive allosteric MEK1/2 inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KU-60019,925701-49-1,KU-60019 is a potent and specific ATM inhibitor with IC50 of 6.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BS-181 HCl,1397219-81-6,BS-181 is a highly selective CDK inhibitor for CDK7 with IC50 of 21 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fasudil HCl (HA-1077),105628-07-7,Fasudil is a potent inhibitor of ROCK-II, PKA,  PKG,  PKC, and MLCK with Ki of 0.33 μM, 1.6 μM, 1.6 μM, 3.3 μM and 36 μM, respectively.  ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIRB 796 (Doramapimod),285983-48-4,BIRB 796 (Doramapimod) is a highly selective p38α MAPK inhibitor with Kd of 0.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tie2 kinase inhibitor,948557-43-5,Tie2 kinase inhibitor is a potent and selective Tie2 inhibitor with IC50 of 0.25 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Candesartan (Atacand),139481-59-7,Candesartan is an angiotensin II receptor antagonist with IC50 of 0.26 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD 0332991 (Palbociclib) Isethionate,827022-33-3,PD 0332991 (Palbociclib) Isethionate is the isethionate of PD 0332991, a highly specific inhibitor of CDK4 and CDK6 with IC50 of 11 nM and 16 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
H 89 2HCl,130964-39-5,H 89 2HCl is a mutiple-targeted inhibitor for S6K1, MSK1, PKA, ROCKII, PKBα and MAPKAP-K1b with IC50 of 80 nM, 120 nM, 135 nM, 270 nM, 2600 nM and 2800 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TWS119,601514-19-6,TWS119 is a GSK-3β inhibitor with IC50 of 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ubenimex (Bestatin),58970-76-6,Ubenimex is a competitive aminopeptidase B inhibitor with an IC50 of 100 mg/ml for K562 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apixaban,503612-47-3,Apixaban is a highly selective, reversible inhibitor of Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbit, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Semagacestat (LY450139),425386-60-3,Semagacestat (LY450139) is a γ-secretase blocker for Aβ42, Aβ40 and Aβ38 with IC50 of 10.9 nM, 12.1 nM and 12.0 nM, respectively. Semagacestat also inhibits Notch signaling with IC50 of 14.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Olmesartan medoxomil (Benicar),144689-63-4,Olmesartan medoxomil (Benicar) is a compound which is hydrolyzed to olmesartan that is a selective AT1 subtype angiotensin II receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rizatriptan Benzoate (Maxalt),145202-66-0,Rizatriptan Benzoate(Maxalt) is a 5-HT1 agonist triptan drug for the treatment of migraine headaches.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pyridostigmine Bromide (Mestinon),101-26-8,Pyridostigmine Bromide(Mestinon) is a parasympathomimetic and a reversible cholinesterase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cefoperazone (Cefobid),62893-19-0,Cefoperazone is a cephalosporin antibiotic for inhibition of rMrp2-mediated [3H]E217βG uptake with IC50 of 199 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Silodosin (Rapaflo),160970-54-7,Silodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Riluzole (Rilutek),1744-22-5,Riluzole(Rilutek) is a drug used to treat amyotrophic lateral sclerosis. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Risperidone (Risperdal),106266-06-2,Risperidone(Risperdal) is an atypical antipsychotic used to treat schizophrenia.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Acetylcysteine,616-91-1,Acetylcysteine is a pharmaceutical drug and nutritional supplement used primarily as a mucolytic agent and in the management of paracetamol (acetaminophen) overdose. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Alendronate (Fosamax),121268-17-5,Alendronate (Fosamax) is a farnesyl diphosphate synthase inhibitor with IC50 of 460 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naproxen (Aleve),26159-34-2,Naproxen (Aleve, Anaprox) is a COX inhibitor for COX-1 and COX-2 with IC50 of 8.7 μM and 5.2 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nitazoxanide (Alinia, Annita),55981-09-4,Nitazoxanide(Alinia, Annita) is a synthetic nitrothiazolyl-salicylamide derivative and an antiprotozoal agent. (IC50 for canine influenza virus ranges from 0.17 to 0.21 μM),HPLC 99%, NMR, LCMS is OK, stock more than 20g
Orlistat (Alli, Xenical),96829-58-2,Orlistat is a general lipase inhibitor with IC50 of 122 ng/ml for PL from human duodenal juice.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Allopurinol (Zyloprim),315-30-0,Allopurinol (Zyloprim) is a xanthine oxidase inhibitor with an IC50 of 7.82±0.12 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Allopurinol Sodium (Aloprim),17795-21-0,Allopurinol Sodium(Aloprim) is a xanthine oxidase inhibitor with an IC50 of 7.82±0.12 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zafirlukast (Accolate),107753-78-6,Zafirlukast is a leukotriene receptor antagonist (LTRA). (IC50=0.6μM, IC50=7.0 µM for CYP2C9),HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ibuprofen (Advil),15687-27-1,Ibuprofen (Advil, Dolgesic) is an anti-inflammatory inhibitor targeting COX-1 and COX-2 with IC50 of 13 μM and 370 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amprenavir (Agenerase),161814-49-9,Amprenavir is a HIV protease inhibitor with IC50 of 14.6 ng/mL in wild-type HIV isolates.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Methyldopa (Aldomet),555-30-6,Methyldopa (Aldomet) is a DOPA decarboxylase competitive inhibitor with an ED50 of 21.8 mg/kg.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ketoprofen (Actron),22071-15-4,Ketoprofen (Actron) is a non-selective NSAID with IC50 of 0.5 μM and 2.33 μM for human recombinant COX-1 and COX-2, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ketorolac (Toradol),74103-07-4,Ketorolac (Ketorolac tromethamine, Toradol) is a non-selective COX inhibitor of COX-1 and COX-2 with IC50 of 1.23 μM and 3.50 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cytarabine,147-94-4,Cytarabine (Cytosine arabinoside, AraC) is an antimetabolic agent and DNA synthesis inhibitor with IC50 of 16 nM in wild-type CCRF-CEM cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zolmitriptan (Zomig),139264-17-8,Zolmitriptan(Zomig) is a selective serotonin receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Enalaprilat dihydrate,84680-54-6 ,Enalaprilat is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 1.94 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Isradipine (Dynacirc),75695-93-1,Isradipine(Dynacirc) is a calcium channel blocker with an IC50 of 34±8 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Estrone,53-16-7 ,Estrone is an estrogenic hormone.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flucytosine (Ancobon),2022-85-7,Flucytosine (5-Fluorocytosine, 5-FC, Ancobon) is an antifungal drug with IC50 of 0.93 μM in C. albicans.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aminoglutethimide (Cytadren),125-84-8,Aminoglutethimide (AMG, Cytadren) is an aromatase inhibitor with IC50 of 10 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aminophylline (Truphylline),317-34-0 ,Aminophylline(Phyllocontin, Truphylline) is a competitive nonselective phosphodiesterase inhibitor with an IC50 of 0.12 mM and also a nonselective adenosine receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carbamazepine (Carbatrol),298-46-4,Carbamazepine (Carbatrol) is a sodium channel blocker with IC50 of 131 μM in rat brain synaptosomes.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Torsemide (Demadex),56211-40-6,Torsemide(Demadex) is a pyridine-sulfonyl urea type loop diuretic with an IC50 of 2.7 ± 0.17 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Didanosine (Videx),69655-05-6,Didanosine(Videx, Videx EC) is a reverse transcriptase inhibitor with an IC50 of 0.49 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Divalproex sodium,76584-70-8,Divalproex sodium consists of a compound of sodium valproate and valproic acid in a 1:1 molar relationship in an enteric coated form.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Emtricitabine (Emtriva),143491-57-0 ,Emtricitabine (Emtriva) is a nucleoside reverse transcriptase inhibitor with an IC50 of 27.7 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lamivudine (Epivir),134678-17-4,Lamivudine(Epivir) is a potent nucleoside analog reverse transcriptase inhibitor with an IC50 of 2.7 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Eplerenone,107724-20-9,Eplerenone is an aldosterone antagonist with an IC50 of 0.36 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Piroxicam (Feldene),36322-90-4,Piroxicam (Feldene) is a non-selective COX inhibitor with an IC50 of 6 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gemcitabine (Gemzar),95058-81-4 ,Gemcitabine(Gemzar) belongs to the group of medicines called antimetabolites.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Adefovir Dipivoxil (Preveon, Hepsera),142340-99-6,Adefovir Dipivoxil(Preveon, Hepsera) works by blocking reverse transcriptase, an enzyme that is crucial for the hepatitis B virus (HBV) to reproduce in the body.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zalcitabine,7481-89-2,Zalcitabine is a nucleoside analog HIV reverse transcriptase inhibitor (NARTI).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Paliperidone (Invega),144598-75-4,Paliperidone(Invega) is an atypical antipsychotic.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Telmisartan (Micardis),144701-48-4,Telmisartan (Micardis) is an angiotensin II receptor antagonist (ARB) used in the management of hypertension.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nevirapine (Viramune),129618-40-2,Nevirapine(Viramune) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used to treat HIV-1 infection and AIDS.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Esomeprazole magnesium (Nexium),161973-10-0 ,Esomeprazole magnesium(Nexium) is a proton pump inhibitor to reduce gastric acid secretion.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nimodipine (Nimotop),66085-59-4,Nimodipine(Nimotop) is a dihydropyridine derivative and an analogue of the calcium channel blocker nifedipine, with antihypertensive activity.Nimodipine decreases intracellular free Ca2+,Beclin-1 and autophagy.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nisoldipine (Sular),63675-72-9,Nisoldipine (Sular) is a calcium channel blocker belonging to the dihydropyridines class, specific for L-type Cav1.2 with IC50 of 10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oxybutynin (Ditropan),5633-20-5,Oxybutynin(Ditropan) is an anticholinergic medication used to relieve urinary and bladder difficulties.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Quetiapine fumarate (Seroquel),111974-72-2,Quetiapine fumarate(Seroquel) is an atypical antipsychotic used in the treatment of schizophrenia, bipolar I mania, bipolar II depression, bipolar I depression.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Chlorprothixene,113-59-7,Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Thioguanine,154-42-7,Thioguanine is a purine antimetabolite widely used in the treatment of acute lymphoblastic leukemia, autoimmune disorders (e.g., Crohn's disease, rheumatoid arthritis) and organ transplant recipients.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Toremifene Citrate (Fareston, Acapodene),89778-27-8,Toremifene Citrate(Fareston, Acapodene) is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azacitidine (Vidaza),320-67-2,Azacitidine is a nucleoside analogue of cytidine that specifically inhibits DNA methylation by trapping DNA methyltransferases.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bacitracin zinc,1405-89-6,Bacitracin zinc is a dephosphorylation of the C55-isoprenyl pyrophosphate interference for inhibition of cleavage of Tyr from Met-enkephalin with IC50 of 10 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Simvastatin (Zocor),79902-63-9,Simvastatin (Zocor) is a competitive inhibitor of HMG-CoA reductase with Ki of 0.1-0.2 nM .,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ramipril (Altace),87333-19-5,Ramipril (Altace) is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ranitidine (Zantac),66357-59-3,Ranitidine (Zantac) is a histamine H2-receptor antagonist with IC50 of 3.3 ± 1.4 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Acadesine,2627-69-2,Acadesine results in accumulation of ZMP, which mimics both activating effects of AMP on AMPK and AMPKK.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Acetylcholine chloride,60-31-1 ,The chemical compound acetylcholine (ACh) is a neurotransmitter in both the peripheral nervous system (PNS) and central nervous system (CNS) in many organisms including humans. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nifedipine (Adalat),21829-25-4,Nifedipine(Adalat), a potent vasodilator agent with calcium antagonistic action.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amlodipine besylate (Norvasc),111470-99-6,Amlodipine (Norvasc) is a long-acting calcium channel blocker with an IC50 of 1.9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Chlorpheniramine Maleate,113-92-8,Chlorpheniramine (Chlorpheniramine maleate, Chlorphenamine) is an histamine H1 receptor antagonist with IC50 of 12 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Betaxolol HCl (Betoptic),63659-19-8,Betaxolol hydrochloride (Betoptic) is a β1 adrenergic receptor blocker with IC50 of 6 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Proparacaine HCl,5875-06-9,Proparacaine HCl is a voltage-gated sodium channels antagonist with ED50 of 3.4 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pranlukast,103177-37-3,Pranlukast is a selective cysteinyl leukotriene receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carvedilol,72956-09-3,Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Butoconazole nitrate,64872-77-1,Butoconazole nitrate is an anti-fungal agent for IL-2, TNFα, IFN and GM-CSF with IC50 of 7.2 μg/mL, 14.4 μg/mL, 7.36 μg/mL and 7.6 μg/mL, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Azithromycin (Zithromax),83905-01-5,Azithromycin (Zithromax) is an antibiotic for inhibition of parasite growth with IC50 of 8.4 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Flubendazole (Flutelmium),31430-15-6,Flubendazole (Flutelmium) is an anthelmintic agent for MDAY-D2 cells with IC50 of 3 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Lomustine (CeeNU),13010-47-4,Lomustine inhibits cancer cells by damaging the DNA and stops cells from dividing.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cimetidine (Tagamet),51481-61-9,Cimetidine(Tagamet), a histamine congener, competitively inhibits histamine binding to histamine H2 receptors.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clemastine Fumarate,14976-57-9,Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Bifonazole,60628-96-8,Bifonazole is an antifungal agent and a prostatic aromatase activity inhibitor with IC50 of 1.6 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Metoprolol tartrate,392-17-7,Metoprolol tartrate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Etidronate (Didronel),2809-21-4,Etidronate (Didronel) is a human protein tyrosine phosphatase inhibitor with IC50 of 0.2 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Dapoxetine HCl (Priligy),129938-20-1,Dapoxetine hydrochloride is a short-acting novel selective serotonin reuptake inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Tranexamic acid (Transamin),1197-18-8,Tranexamic acid (Transamin) is an antifibrinolytic for blocking lysine-binding sites of plasmin and elastase-derived plasminogen fragments with IC50 of 5 mM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Roxatidine acetate HCl,93793-83-0,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Felodipine (Plendil),72509-76-3,Felodipine (Plendil) is a selective L-type Ca2+ channel blocker with IC50 of 0.15 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nizatidine,76963-41-2,Nizatidine is a histamine H2-receptor antagonist with and IC50 of 6.7 nM for AChE.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carbidopa,28860-95-9,Carbidopa is an aromatic-L-amino-acid decarboxylase inhibitor with an IC50 of 29 ± 2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Valsartan (Diovan),137862-53-4,Valsartan (Diovan) is an angiotensin II receptor antagonist with IC50 of ranging from 39.5 to 116 μM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tropisetron,105826-92-4 ,Tropisetron hydrochloride is a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist with an IC50 of 70.1 ± 0.9 nM for 5-HT3 receptor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Diclofenac sodium,15307-79-6,Diclofenac is a non-selective COX inhibitor with IC50 of 60 and 220 nM for ovine COX-1 and -2, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amlodipine (Norvasc),88150-42-9,Amlodipine(Norvasc) is a long-acting calcium channel blocker with an IC50 of 1.9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flutamide (Eulexin),13311-84-7,Flutamide (Eulexin) is an oral nonsteroidal antiandrogen agent primarily used to treat prostate cancer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fluvastatin sodium (Lescol),93957-55-2,Fluvastatin sodium inhibits HMG-CoA reductase activity with IC50 of 8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Tropicamide,1508-75-4,Tropicamide is an anticholinergic and a muscarinic receptor subtype M4-preferring antagonist with IC50 of 8.0 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Pregnenolone,145-13-1,Pregnenolone is an endogenous steroid hormone for inhibition of M1 receptor- and M3 receptor-mediated currents with IC50 of 11.4 ¦ÌM and 6.0 ¦ÌM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sulfamethoxazole,723-46-6,Sulfamethoxazole is a sulfonamide bacteriostatic antibiotic with an IC50 of 2.7 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Irsogladine,57381-26-7,Irsogladine is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Enalapril maleate (Vasotec),76095-16-4,Enalapril maleate (Vasotec), the active metabolite of enalapril, competes with angiotensin I for binding at the angiotensin-converting enzyme, blocking the conversion of angiotensin I to angiotensin II.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Metformin HCl (Glucophage),1115-70-4,Metformin hydrochloride(Glucophage) is a biguanide hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary modification.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Tolfenamic acid,13710-19-5,Tolfenamic acid is a COX-2 inhibitor with IC50 of 0.2 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Pranoprofen,52549-17-4,Pranoprofen is a PGE2 inhibitor with IC50 of 7.5 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Nefiracetam (Translon),77191-36-7,Nefiracetam (Translon) is a GABAergic, cholinergic, and monoaminergic neuronal systems enhancer for Ro 5-4864-induced convulsions.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nicorandil (Ikorel),65141-46-0,Nicorandil(Ikorel) is potassium channel activator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tamoxifen Citrate (Nolvadex),54965-24-1,Tamoxifen Citrate is an antagonist of the estrogen receptor by competitive inhibition of estrogen binding.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Meglumine,6284-40-8,Meglumine is an amino sugar derived from sorbitol for THP-1 cells with IC50 of 22 μg/mL.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Aripiprazole (Abilify),129722-12-9,Aripiprazole is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Methscopolamine (Pamine),155-41-9,Methscopolamine (Pamine) is a muscarinic acetylcholine receptor blocker. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Amiodarone HCl,19774-82-4,Amiodarone HCl is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with IC50 of 19.1 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Adenine,73-24-5,Adenine is a purine derivative and a nucleobase with a variety of roles in biochemistry.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Adenine sulfate,321-30-2,Adenine sulfate is a sulfate salt form of adenine which is a purine derivative and a nucleobase with a variety of roles in biochemistry.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Adenine HCl,2922-28-3 ,Adenine hydrochloride is a hydrochloride salt form of adenine which is a purine derivative and a nucleobase with a variety of roles in biochemistry.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ticlopidine HCl,53885-35-1,Ticlopidine HCl is an P2 receptor inhibitor against ADP-induced platelet aggregation with IC50 of ~2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lacidipine (Lacipil, Motens),103890-78-4,Lacidipine (Lacipil, Motens) is a L-type calcium channel blocker. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Procarbazine HCl (Matulane),366-70-1,Procarbazine hydrochloride (Matulane) is a hydrochloride salt form of procarbazine which is a polyfunctional alkylating compound used as an antineoplastic agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ondansetron (Zofran),99614-02-5,Ondansetron (Zofran) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium orthovanadate,13721-39-6,Sodium orthovanadate is an alkaline phosphatase and (Na,K)-ATPase inhibitor with IC50 of 10 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Elvitegravir (GS-9137),697761-98-1,Elvitegravir (EVG, JTK-303/GS-9137) is a HIV integrase inhibitor for HIV-1 IIIB, HIV-2 EHO and HIV-2 ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Maraviroc,376348-65-1,Maraviroc (Selzentry, UK-427857, Celsentri) is a CCR5 antagonist for MIP-1α, MIP-1β and RANTES with IC50 of 3.3 nM, 7.2 nM and 5.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Raltegravir (MK-0518),518048-05-0,Raltegravir (MK-0518, Isentress) is a potent integrase (IN) inhibitor for WT and S217Q PFV IN with IC50 of 90 nM and 40 nM, respectivly.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pyrimethamine,58-14-0,Pyrimethamine is a dihydrofolate reductase(DHFR) inhibitor with an IC50 of 15.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pramipexole 2HCl monohydrate ,191217-81-9,Pramipexole is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PCI-34051,950762-95-5,PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF 573228,869288-64-2,PF 573228 is a inhibitor of FAK with IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS-265246,582315-72-8,BMS265246 is a potent and selective CDK inhibitor for CDK1/cyclin B and CDK2/cyclin E with IC50 of 6 nM and 9 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Suplatast tosylate,94055-76-2,Suplatast tosilate is a novel capsular anti-asthmatic agent that suppresses both IgE production, IL-4 and IL-5 synthesis with IC50 above 100 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ENMD-2076 L-(+)-Tartaric acid,1291074-87-7,ENMD-2076 L-(+)-Tartaric acid is the tartaric acid of ENMD-2076, a selective inhibitor of Aurora A and Aurora B with IC50 of 14 nM and 350 nM and also inhibits Flt3, Flt4 and VEGFR2 with IC50 of 1.86 nM, 15.9 nM and 58.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Formoterol hemifumarate,43229-80-7,Formoterol hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist to β2 and β1 receptors with pKd of 8.12 and 5.58, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ketotifen fumarate (Zaditor),34580-14-8,Ketotifen fumarate (Zaditor) is a fumaric acid salt of ketotifen which is a H1-antihistamine and mast cell stabilizer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Urapidil HCl,64887-14-5,Urapidil hydrochloride is a hydrochloride salt form of urapidil which is α1-adrenoceptor antagonist and 5-HT1A receptor agonist with pIC50 of 6.13 and 6.4 respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Ginkgolide A,15291-75-5,Ginkgolide A is an extract from in Ginkgo biloba and a g-aminobutyric acid (GABA) antagonist with a Ki of 14.5 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Uridine,58-96-8,Uridine is a nucleoside, contains a uracil attached to a ribose ring via a β-N1-glycosidic bond.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Flunarizine 2HCl,30484-77-6,Flunarizine dihydrochloride is a dihydrochloride salt form which is a calcium channel blocker with a Ki of 68 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Rebamipide,90098-04-7,Rebamipide is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [125I]BH-CCK-8S with IC50 of 37.7 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Epalrestat,82159-09-9,Epalrestat is an aldose reductase inhibitor with IC50 of 72 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Candesartan cilexetil (Atacand),145040-37-5,Candesartan cilexetil (Atacand) is a specific nonpeptide Ang II receptor (ATR)  antagonist and the prodrug of candesartan which is an ATR antagonist with an IC50 of 15 μg/kg,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Phentolamine mesilate,65-28-1,Phentolamine mesilate is a nonselective alpha-adrenergic antagonist with IC50 of 0.1 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Nimesulide,51803-78-2,Nimesulide is a relatively COX-2 selective inhibitor with IC50 of 26 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Cyproterone acetate,427-51-0,Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Memantine HCl (Namenda),41100-52-1,Memantine hydrochloride (Namenda) is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Cyproheptadine HCl (Periactin),969-33-5 ,Cyproheptadine hydrochloride (Periactin) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist for 5-HT2 receptor with IC50 of 0.6 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Doxifluridine,3094-09-5,Doxifluridine is a thymidine phosphorylase activator for PC9-DPE2 cells with IC50 of 0.62 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Pioglitazone HCl (Actos),112529-15-4,Pioglitazone hydrochloride (Actos) is a hydrochloride salt form of pioglitazone which is a cytochrome P450 (CYP)2C8 and CYP3A4 enzymes inhibitor for CYP2C8, CYP3A4 and CYP2C9 with Ki of 1.7 μM, 11.8 μM and 32.1 μM, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Lornoxicam (Xefo),70374-39-9,Lornoxicam (Xefo) is a COX-1 and COX-2 inhibitor with IC50 of 5 nM and 8 nM, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Strontium ranelate (Protelos),135459-87-9,Strontium ranelate (Protelos) is a strontium(II) salt of ranelic acid for (-)-desmethoxyverapamil binding to calcium channel with IC50 of 0.5 mM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Captopril (Capoten),62571-86-2,Captopril (Capoten) is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Orphenadrine citrate (Norflex),4682-36-4,Orphenadrine citrate is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Gimeracil,103766-25-2,Gimeracil is an inhibitor of dihydropyrimidine dehydrogenase, which inhibits the early step in homologous recombination for double strand breaks repair.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Terazosin HCl (Hytrin),70024-40-7,Hytrin (terazosin) is an alpha-adrenergic blocker used to treat high blood pressure and enlarged prostate.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Lovastatin (Mevacor),75330-75-5,Lovastatin is an inhibitor of HMG-CoA reductase with IC50 of 3.4 nM, used for lowering cholesterol (hypolipidemic agent).
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Lafutidine,118288-08-7,Lafutidine, a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Moxonidine,75438-57-2,Moxonidine is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Ozagrel HCl,78712-43-3,Ozagrel hydrochloride is a selective thromboxane A2 synthetase enzyme inhibitors with IC50 of 11 nM, used as antiasthmatic agent.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Mitiglinide calcium,145525-41-3,Mitiglinide is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-cells.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Rosiglitazone HCl,302543-62-0,Rosiglitazone is a blood glucose-lowering drugs, stimulating insulin secretion by binding to the PPAR receptors in fat cells.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Lisinopril (Zestril),83915-83-7,Lisinopril is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks, and also in preventing renal and retinal complications of diabetes.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Atorvastatin calcium (Lipitor),134523-03-8,Atorvastatin (Lipitor) is an inhibitor of HMG-CoA reductase used as a cholesterol-lowering medication that blocks the production of cholesterol.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Famotidine (Pepcid),76824-35-6,Famotidine is a histamine H2–receptor antagonist with IC50 of 0.6 mM, commonly used to treat heartburn, GERD, ulcers, and other digestive conditions.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Moexipril HCl,82586-52-5,Moexipril hydrochloride is a potent orally active non-sulfhydryl angiotensin converting enzyme inhibitor (ACE) with IC50 of 0.041 ¦ÌM, which is used for the treatment of hypertension and congestive heart failure.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Cleviprex (Clevidipine),167221-71-8,Cleviprex (Clevidipine) is a dihydropyridine calcium channel blocker use as agent for the reduction of blood pressure.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Cilazapril monohydrate (Inhibace),92077-78-6,Cilazapril is a angiotensin-converting enzyme (ACE) inhibitor used for the treatment of hypertension and congestive heart failure.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Adiphenine HCl,50-42-0,Adiphenine is a nicotinic receptor inhibitor with IC50 of 15 ¦ÌM, used as an antispasmodic drug.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Duloxetine HCl (Cymbalta),136434-34-9 ,Duloxetine is a serotonin-norepinephrine reuptake inhibitor with Ki of 4.6 nM, used for treatment of major depressive disorder and generalized anxiety disorder (GAD).
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Trimebutine,39133-31-8,Trimebutine is an agonist of peripheral mu, kappa and delta opiate receptors, used as spasmolytic agent for treatment of both acute and chronic abdominal pain.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Ivabradine HCl (Procoralan),148849-67-6,Ivabradine, a new If inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Rivastigmine tartrate (Exelon),129101-54-8,Rivastigmine, a cholinesterase inhibitor with IC50 of 5.5 μM, ues as a parasympathomimetic or cholinergic agent for the treatment of mild to moderate Alzheimer disease.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Dexmedetomidine HCl (Precedex),145108-58-3,Dexmedetomidine is a highly selective and potent alpha-2 adrenoceptor agonist, which reduces anesthetic requirements for patients by providing significant sedation.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Betaxolol (Betoptic),659-18-7,Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Detomidine HCl,90038-01-0,Detomidine produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Fosinopril sodium (Monopril),88889-14-9,Fosinopril sodium (Monopril) is the ester prodrug of an angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension and some types of chronic heart failure.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Almotriptan malate (Axert),181183-52-8,Almotriptan malate (Axert) is a selective 5-hydroxytryptamine1B/1D (5-HT1B/1D) receptor agonist, used for the treatment of Migraine attacks in adults.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Ambrisentan,177036-94-1,Ambrisentan, a highly selective antagonist of the endothelin-1 type A receptor with IC50 of 18 nM, is indicated for the treatment of pulmonary arterial hypertension (PAH).
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Bexarotene,153559-49-0,Bexarotene is a retinoid specifically selective for retinoid X receptors, used as an oral antineoplastic agent in the treatment of cutaneous T-cell lymphoma.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Temocapril HCl,110221-44-8,Temocapril HCl is the hydrochloride of Temocapril, which is a long-acting angiotensin-converting enzyme (ACE) inhibitor, used for the treatment of hypertension.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Gabexate mesylate,56974-61-9,Gabexate is a serine protease inhibitor with IC50 of 0.19 μM which is used therapeutically in the treatment of pancreatitis and disseminated intravascular coagulation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Rasagiline mesylate,161735-79-1,Rasagiline mesylate is a new MAO-B inhibitor for the treatment of idiopathic Parkinson's disease.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Naltrexone HCl,16676-29-2,Naltrexone is an opioid receptor antagonist with IC50 of 8 nM used primarily in the management of alcohol dependence and opioid dependence.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Levosulpiride (Levogastrol),23672-07-3,Levosulpiride is a selective antagonist for D2 dopamine receptors used as an antipsychotic and prokinetic agent.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Azasetron HCl (Y-25130),123040-16-4,Azasetron HCl is a selective 5-HT3 receptor antagonist with IC50 of 0.33 nM used in the management of nausea and vomiting induced by cancer chemotherapy.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Mizolastine (Mizollen),108612-45-9,Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Flunixin meglumin,42461-84-7,Flunixin meglumine is a potent inhibitor of the enzyme cyclooxygenase used as analgesic agent with anti-inflammatory and antipyretic activity.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Vinpocetine (Cavinton),42971-09-5,Vinpocetine is a selectively inhibitor of voltage-sensitive sodium channel for the treatment of stroke, vascular dementia  and Alzheimer's disease.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Lapatinib,231277-92-2,Lapatinib, used in the form of Lapatinib Ditosylate, is a potent EGFR and ErbB2 inhibitor with IC50 of 10.8 and 9.2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Blonanserin (Lonasen),132810-10-7,Blonanserin is a novel atypical antipsychotic agent with potent dopamine D2 (Ki, 14.8 nM) and serotonin 5-HT2(Ki, 3.98 nM) receptors antagonist properties.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Cisatracurium besylate (Nimbex),96946-42-8,Cisatracurium besylate is a nondepolarizing neuromuscular blocking agent, antagonizing the action of acetylcholine by inhibiting neuromuscular transmission.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Ibutilide fumarate,122647-32-9,Ibutilide is a Class III antiarrhythmic agent that is indicated for acute cardioconversion of atrial fibrillation and atrial flutter of a recent onset to sinus rhythm by induction of slow inward sodium current, which prolongs action potential and refractory period of myocardial cells.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Naftopidil (Flivas),57149-07-2,Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
S- (+)-Rolipram,85416-73-5,S-(+)-Rolipram inhibits human monocyte cyclic AMP-specific PDE4 with IC50 of 0.75 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bazedoxifene HCl,198480-56-7,Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of  23 nM and 89 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Atropine,5908-99-6,Atropine sulfate monohydrate is a competitive muscarinic acetylcholine receptor antagonist with an IC50 of 2.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Roflumilast (Daxas),162401-32-3,Roflumilast (Daxas) is a selective inhibitor of PDE4 with IC50 of 0.2-4.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gabapentin (Neurontin),60142-96-3,Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analogue.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD8330,869357-68-6,AZD8330 (ARRY-424704) is a MEK 1/2 inhibitor with IC50 of 7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1292263,1032823-75-8,GSK-1292263 is a novel GPR119 agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Neratinib (HKI-272),698387-09-6,Neratinib (HKI-272) is a highly selective HER2 and EGFR inhibitor with IC50 of 59 nM and 92 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LDE225 (NVP-LDE225, Erismodegib),956697-53-3,LDE225 (NVP-LDE225) is a smoothened antagonist with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CGS 21680 HCl,124431-80-7,CGS 21680 hydrochloride is an A2A adenosine receptor agonist with an Ki of 27 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIBR-1048 (Dabigatran etexilate, Pradaxa),211915-06-9,BIBR-1048 (Dabigatran) is an anticoagulant from the class of the direct thrombin inhibitors. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2608204,1234703-40-2,LY2608204 activates glucokinase (GK) with EC50 of 42 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2886721,1262036-50-9,LY2886721 is an BACE inhibitor used for the treatment of Alzheimer's Disease.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2940680,1258861-20-9,LY2940680 binds to the Smo receptor and potently inhibits Hh signaling.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KW 2449,1000669-72-6,KW-2449 potently inhibits Flt3, Abl and Aurora A with IC50 of 6.6 nM, 14 nM and 48 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tebipenem pivoxil (L-084),161715-24-8,Tebipenem pivoxil(L-084) is a novel oral carbapenem antibiotic with an IC50 of 100 μg/ml for human CYP isoforms,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-4708671,1255517-76-0,PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) with Ki of 20 nM and IC50 of 160 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD 128907 HCl,112960-16-4,PD 128907 HCl is a potent and selective dopamine D2/D3 receptors agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rosuvastatin calcium (Crestor),147098-20-2,Rosuvastatin calcium is an competitive inhibitor of HMG-CoA reductase with IC50 of 11 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ITF2357 (Givinostat),732302-99-7,ITF2357 (Givinostat) is a potent inhibitor of HDAC with IC50 of 7.5-16 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AG14361,328543-09-5,AG14361 is a potent inhibitor of PARP1 with Ki of < 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2784544,1229236-86-5,LY2784544 is selective to V617F mutant JAK2 with IC50 of 55 nM in Ba/F3 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MLN2238,1072833-77-2,MLN2238 inhibits the chymotrypsin-like proteolytic (β5) site of the 20S proteasome with IC50 and Ki of 3.4 nM and 0.93 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MLN9708,1201902-80-8,MLN9708 is a selective inhibitor of chymotrypsin-like proteolytic (β5) site of the 20S proteasome with IC50 and Ki of 3.4 nM and 0.93 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 743921,940929-33-9,SB 743921 is a KSP inhibitor with IC50 of 0.2 nM, 0.07 nM, 1.7 nM, 0.06 nM and 14.4 nM in SKOV3, Colo205, MV522, MX1 and P388 cell lines, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BGJ398 (NVP-BGJ398),872511-34-7,BGJ398 (NVP-BGJ398) is a potent and selective inhibitor of FGFR1, FGFR2 and FGFR3 with IC50 of 0.9 nM, 1.4 nM and 1 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AST-1306,1050500-29-2,AST-1306 is a novel irreversible inhibitor of EGFR and ErbB4 with IC50 of 0.5 nM and 0.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB-505124,694433-59-5,SB505124 is a selective inhibitor of ALK4 and ALK5 with IC50 of 129 nM and 47 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Avasimibe (CI-1011),166518-60-1 ,Avasimibe inhibits ACAT and CYP2C9 with IC50 of 3.3 μM and 2.9 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD8931,848942-61-0,AZD8931 is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4 nM, 3 nM and 4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK461364,929095-18-1,GSK461364 inhibits purified Plk1 with Ki of 2 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
R406,841290-81-1,R406 is a potent Syk inhibitor with IC50 of 41 nM and also potently inhibits Flt3.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SGI-1776 free base,1025065-69-3,SGI-1776 is a novel ATP competitive inhibitor to Pim1, Pim2 and Pim3 with IC50 of 7 nM, 363 nM and 69 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aliskiren hemifumarate,173334-58-2,Aliskiren hemifumarate is a direct renin inhibitor with IC50 of 1.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS 794833,1174046-72-0,BMS794833 is a potent ATP competitive inhibitor of Met and VEGFR2 with IC50 of 1.7 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-BHG712,940310-85-0,NVP-BHG712 is a specific inhibitor of c-Raf, c-Src and c-Abl with IC50 of 0.395 μM, 1.266 μM and 1.667 μM and also inhibits EphB4 and VEGFR2 with ED50 of 25 nM and 4.2 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
OSI-420,183320-51-6,OSI-420 is an active metabolite of Erlotinib which is an orally active EGFR inhibitor for inhibition of human EGFR and EGFR autophosphorylation with IC50 of 2 nM and 20 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
R935788 (Fostamatinib disodium, R788 disodium),1025687-58-4,R935788 (Fostamatinib disodium, R788) is a Syk inhibitor with IC50 of 41 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PIK-293,900185-01-5 ,PIK-293 is a PI3-K inhibitor for p110α, p110β, p110δ and p110γ with IC50 of 100 μM, 25 μM, 0.24 μM and 10 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Formestane,566-48-3,Formestane(Lentaron(R)) is a second generation selective aromatase inhibitor with an IC50 of 80 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vinflunine Tartrate,1201898-17-0,Vinflunine is a new vinca alkaloid uniquely fluorinated with the properties of mitotic-arresting and tubulin-interacting activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZ 960,905586-69-8,AZ 960 is a novel ATP competitive JAK2 inhibitor with IC50 and Ki of <3 nM and 0.45 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
DAPT (GSI-IX),208255-80-5,DAPT (GSI-IX) is a novel γ-secretase inhibitor, which inhibits Aβ production with IC50 of 20 nM in HEK 293 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mubritinib (TAK 165),366017-09-6,Mubritinib (TAK 165) is a potent inhibitor of ErbB2 with IC50 of 6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Irinotecan HCl Trihydrate (Campto),136572-09-3,Irinotecan prevents DNA from unwinding by inhibition of topoisomerase 1.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PP242,1092351-67-1,PP242 is a selective mTOR inhibitor with IC50 of 8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cyt387,1056634-68-4,CYT387 is an ATP-competitive inhibitor of JAK1 and JAK2 with IC50 of 11 nM and 18 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB590885,405554-55-4 ,SB590885 is a potent B-Raf inhibitor with Ki of 0.16 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apatinib (YN968D1),811803-05-1,Apatinib (YN968D1) is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAME,901-47-3,Tosyl-L-Arginine Methyl Ester (TAME) is an APC inhibitor and also inhibits an E3 ubiquitin ligase called "anaphase-promoting complex/cyclosome (APC/C)".,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CAL-101 (GS-1101),870281-82-6,CAL-101 is a selective PI3K class I inhibitor of p110δ with IC50 of 2.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PIK-294,900185-02-6,PIK-294 is a highly potent and selective p110δ inhibitor with IC50 of 10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Eltrombopag (SB-497115-GR),496775-61-2,Eltrombopag (SB-497115-GR, Promacta, Revolade) is a small molecule agonist of the c-mpl (TpoR) receptor with an IC50 of 0.69 μM for the inhibition of hERG K+ channel tail current.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2157299,700874-72-2,LY2157299 is a potent TGFβ receptor I (TβRI) inhibitor with IC50  of 56 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Telatinib (BAY 57-9352),332012-40-5,Telatinib (BAY 57-9352) is a potent inhibitor of VEGFR2/3, c-Kit and PDGFRβ with IC50 of 6 nM/4 nM, 1 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ketanserin (Vulketan Gel),74050-98-9,Ketanserin (Vulketan Gel) is specific 5-HT2A serotonin receptor antagonist with a Ki of 2.5 nM for rat and human 5-HT2A.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Esomeprazole sodium (Nexium),161796-78-7,Esomeprazole sodium (Nexium) is a sodium salt of esomeprazole that is a potent proton pump inhibitor with an IC50 of 0.076 mg/kg.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BI6727 (Volasertib),755038-65-4,BI6727 (Volasertib) is a highly potent Plk1 inhibitor with IC50 of 0.87 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Palomid 529,914913-88-5,Palomid 529 (P529) is a PI3K/Akt/mTOR inhibitor for VEGF-A and bFGF with IC50 of 10 nM and 30 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fesoterodine fumarate (Toviaz),286930-03-8,Fesoterodine fumarate (Toviaz) is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WP1130,856243-80-6,WP1130 (degrasyn) is a selective deubiquitinase (DUB: USP5, UCH-L1,  USP9x, USP14, and UCH37) inhibitor and also inhibits Bcr/Abl with IC50 of 1.8 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AR-42 (HDAC-42),935881-37-1,AR-42 (HDAC-42, OSU-HDAC42) is a pan-HDAC inhibitor with IC50 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CP-466722,1080622-86-1,CP-466722 is an potent and reversible ATM inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Abiraterone Acetate (CB7630),154229-18-2,Abiraterone acetate (CB7630, CB 7630, CB-7630) is an acetate salt form of Abiraterone which is a steroidal cytochrome CYP17 inhibitor with IC50 of 72 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BKM120 (NVP-BKM120),944396-07-0,BKM120 is a selective PI3K inhibitor of p110α, p110β, p110δ and p110γ with IC50 of 52-99 nM, 166 nM, 116 nM and 262 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CX-4945 (Silmitasertib),1009820-21-6,CX-4945 is a potent and selective inhibitor of CK2α and CK2α' with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
(-)-Huperzine A,102518-79-6,(-)-Huperzine A is a potent, highly specific and reversible inhibitor of acetylcholinesterase (AChE) with Ki of 7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
4-Methylumbelliferone (4-MU),90-33-5,4-Methylumbelliferone is a hyaluronic acid (HA) synthesis inhibitor with an IC50 of 0.4 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aloe-emodin,481-72-1,Aloe-emodin is an interferon-inducing agent with IC50 of about 1 μg/mL for JEV and of about 0.33 μg/mL for EV71.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apigenin,520-36-5,Apigenin is a potent P450 inhibitor for CYP2C9 with IC50 of 23 pM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Arbutin (Uva, p-Arbutin),497-76-7,Arbutin(Uvasol, p-Arbutin) is a tyrosinase inhibitor with an IC50 of 1.09 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Artesunate,88495-63-0,Artesunate is a part of the artemisinin group of agents with an IC50 of < 5 μM for small cell lung carcinoma cell line H69.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Asiatic acid,464-92-6,Asiatic acid is the aglycone of asiaticoside isolated from the plant Centella asiatica, commonly used in wound healing. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Baicalein,491-67-8,Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Baicalin,21967-41-9,Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cryptotanshinone,35825-57-1,Cryptotanshinone (CPT) is a STAT3 inhibitor with IC50 of 4.6 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cytisine (Baphitoxine, Sophorine),485-35-8,Cytisine is a nicotinic acetylcholine receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hesperetin,520-33-2,Hesperetin is a bioflavonoid and, to be more specific, a flavanone.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Honokiol,35354-74-6,Honokiol is a biphyl neolignan present in the cones, bark, and leaves of Magnolia grandifloris that displays antiangiogenic, antiinflammatory, and antitumor properties due to the inhibitory effect on the PI3K/Akt pathway.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Icariin,489-32-7,Icariin is a flavonol and PDE5 inhibitor with IC50 of 1.0, 0.75, and 1.1 μM for PDE5A1, A2, and A3, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Luteolin,491-70-3 ,Luteolin is a PDE4 inhibitor and a general phosphodiesterase inhibitor, and an Interleukin 6 inhibitor. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Matrine ((+)-Matrine),519-02-8 ,Matrine((+)-Matrine) is an alkaloid found in plants from the Sophora family. It has a variety of pharmacological effects, including anti-cancer effects, and action as a kappa opioid receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Neohesperidin,13241-33-3 ,Neohesperidin is an antioxidant agent with an IC50 of 22.31 μg/ml in the 1,1-diphenyl-2-picryldydrazyl (DPPH) radical-scavenging assay.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Parthenolide ((-)-Parthenolide),20554-84-1,Parthenolide ((-)-Parthenolide) is a sesquiterpene lactone which occurs naturally in the plant feverfew(Tanacetum parthenium) and also promotes the ubiquitination of MDM2 and activates p53 cellular functions.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Puerarin (Kakonein),3681-99-0,Puerarin (Kakonein) is a 5-HT2C receptor and benzodiazepine site antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Salinomycin (Procoxacin),53003-10-4,Aminoglutethimide (Cytadren) is an anti-steroid drug which inhibits aromatase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Synephrine (Oxedrine),94-07-5,Synephrine (Oxedrine) is a compound commonly used for weight loss.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
5-hydroxytryptophan (5-HTP),56-69-9,5-Hydroxytryptophan(5-HTP) is decarboxylated to serotonin (5-hydroxytryptamine or 5-HT) by the enzyme aromatic-L-amino-acid decarboxylase with the help of Vitamin B6.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aloin (Barbaloin),1415-73-2 ,Aloin(Barbaloin) is a potent tyrosinase inhibitor with an IC50 of 97 μM for HeLaS3 cells,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dioscin (Collettiside III),19057-60-4 ,Dioscin(Collettiside III) is a saponin extracted and isolated from Polygonatum Zanlanscianense Pamp with IC50 of 2.6, 0.8, 7.5, and 4.5 μM for the inhibition of the growth of the MDA-MB-435, H14, HL60, and HeLa cell lines, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Indirubin,479-41-4 ,Indirubin is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 75 nM and 0.19 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Quercetin (Sophoretin),117-39-5,Quercetin (Sophoretin) is a PI3K and PKC inhibitor with IC50 of 3.8 μM and 15µg/ml. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naringenin,480-41-1,Naringenin is a flavonoid that is considered to have a bioactive effect on human health as antioxidant, free radical scavenger, anti-inflammatory, carbohydrate metabolism promoter, and immune system modulator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Salidroside (Rhodioloside),10338-51-9,Salidroside (Rhodioloside; Rhodosin) is a glucoside compound with an IC50 of 4.99 ± 0.23 μg/mL for the proliferation of SACC-2 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium Danshensu,67920-52-9,Sodium Danshensu is a mono sodium of danshensu which is a compound isolated from Salvia miltiorrhiza Bge.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tetrandrine (Fanchinine),518-34-3,Tetrandrine (Fanchinine; Hanfangchin A) is a calcium channel blocker with an IC50 of 38.23± 25.77 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Chrysophanic acid (Chrysophanol),481-74-3,Chrysophanic acid (Chrysophanol) is a EGFR/mTOR pathway inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Astragaloside A,83207-58-3,Astragaloside A is a pure small molecular compound isolated from Radix Astragali and is commonly used in the treatment of degenerative bone diseases such as osteoporosis. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
20-Hydroxyecdysone,5289-74-7,20-Hydroxyecdysone (Ecdysterone, 20E) is a naturally occurring ecdysteroid hormone which controls the ecdysis (moulting) and metamorphosis of arthropods.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
10-Hydroxycamptothecin,19685-09-7,10-Hydroxycamptothecin (10-HCPT, 10-hydroxy-CPT, OHCPT, NSC107124) is a DNA topoisomerase I inhibitor with potent anti-tumor activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apocynin (Acetovanillone),498-02-2,Apocynin (Acetovanillone) is a selective NADPH-oxidase inhibitor with IC50 of 10 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rotundine,483-14-7,Rotundine (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Synephrine HCl,5985-28-4,Synephrine HCl (Oxedrine, p-Synephrine) is a sympathomimetic α-adrenergic receptor (AR) agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tolbutamide,64-77-7,Tolbutamide is an inhibitor of cAMP with IC50 of 4 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Forskolin,66575-29-9,Forskolin is a ubiquitous activator of eukaryotic adenylyl cyclase (AC).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Equol,531-95-3,Equol is an isoflavandiol metabolized from daidzein by bacterial flora in the intestines.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amantadine HCl (Symmetrel),665-66-7,Amantadine hydrochloride(Symmetrel) is used to treat or prevent infections of the respiratory tract caused by a certain virus.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amfebutamone (Bupropion),31677-93-7,Amfebutamone (Bupropion) is a selective norepinephrine-dopamine reuptake inhibitor with IC50 of 6.5 and 3.4μM for the reuptake of dopamine and norepinephrine, respectively,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Benserazide,14919-77-8,Benserazide is a peripherally-acting aromatic L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bupivacaine HCl (Marcain),18010-40-7,Bupivacaine hydrochloride(Marcain) is a more potent cAMP production inhibitor with an IC50 of 2.3 μM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bethanechol chloride,590-63-6,Bethanechol chloride is a selective muscarinic receptor agonist without any effect on nicotinic receptors.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Chlorpromazine (Sonazine),69-09-0,Chlorpromazine (Sonazine) is a dopamine and potassium channel inhibitor with IC50 of 6.1 and 16 μM for nward-rectifying K+ currents and time-independent outward currents,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clonidine HCl (Catapres),4205-91-8,Clonidine hydrochloride(Catapres) is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clozapine (Clozaril),5786-21-0,Clozapine (Clozaril) is a potent 5-HT1C receptor antagonist with an IC50 of 110 nM for 5-HT-stimulated phosphoinositide hydrolysis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pramipexole (Mirapex),104632-26-0,Pramipexole (Mirapex) is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Domperidone (Motilium),57808-66-9,Domperidone(Motilium) is a dopamine blocker and an antidopaminergic reagent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Donepezil HCl (Aricept),120011-70-3,Donepezil is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM , respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Estriol,50-27-1,Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fluocinolone acetonide (Flucort-N),67-73-2,Fluocinolone(Flucort-N) acetonide is a corticosteroid that binds to the cytosolic glucocorticoid receptor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gallamine triethiodide (Flaxedil),65-29-2,Gallamine triethiodide(Flaxedil) is a cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hexestrol (Bibenzyl),84-16-2,Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Imatinib (Gleevec),152459-95-5,Imatinib is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC50 of 0.6 μM, 0.1 μM and 0.1 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Loperamide HCl,34552-83-5,Loperamide is an opioid-receptor agonist with an ED50 of 0.15 mg/kg.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Manidipine (Manyper),89226-50-6,Manidipine (Manyper) is a lipophilic, third-generation, highly vasoselective dihydropyridine calcium antagonist with an IC50 of 2.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Manidipine 2HCl (CV-4093),89226-75-5,Manidipine HCl is a HCl salt form of Manidipine which is a calcium channel blocker for Ca2+ current with IC50 of 2.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Milrinone (Primacor),78415-72-2,Milrinone(Primacor) is a a potent and selective phosphodiesterase 3 inhibitor with an IC50 of 0.42 μM for the inhibition of FIII PDE,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mitoxantrone HCl,70476-82-3,Mitoxantrone HCl is a classic folic acid antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nateglinide (Starlix),105816-04-4,Nateglinide(Starlix) is an insulin secretagog agent that lowers blood glucose levels by stimulating insulin secretion from the pancreas.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Neostigmine bromide (Prostigmin),114-80-7,Neostigmine bromide(Prostigmin) is a reversible acetylcholinesterase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nitrendipine,39562-70-4,Nitrendipine is a dihydropyridine calcium channel blocker with an IC50 of 95 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Olanzapine (Zyprexa),132539-06-1,Olanzapine(Zyprexa) is a high affinity for 5-HT2 serotonin and D2 dopamine receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Olopatadine HCl (Opatanol),140462-76-6,Olopatadine hydrochloride(Opatanol) is a histamine blocker and mast cell stabilizer with an IC50 of 559 μM for the release of histamine,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oxymetazoline HCl,2315-02-8,Oxymetazoline hydrochloride is an α1 and α2 adrenergic receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ozagrel,82571-53-7,Ozagrel is a potent and selective thromboxane A2 synthetase inhibitor with an IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pancuronium (Pavulon),15500-66-0,Pancuronium (Pavulon) is a competitive acetylcholine antagonist with an IC50 of 5.5 ¡À 0.5 nM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenoxybenzamine HCl,63-92-3,Phenoxybenzamine HCl is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Propafenone (Rytmonorm) HCl,34183-22-7,Propafenone(Rytmonorm) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial and ventricular arrhythmias.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Racecadotril (Acetorphan),81110-73-8,Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rosiglitazone maleate,155141-29-0,Rosiglitazone maleate (Avandia) is an anti-diabetic agent in the thiazolidinedione class of agents.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Salbutamol sulfate (Albuterol),51022-70-9,Salbutamol (Albuterol) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Scopolamine HBr,114-49-8,Scopolamine hydrobromide is a competitive muscarinic acetylcholine receptor with an IC50 of 55.3 ¡À 4.3 nM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sotalol (Betapace),959-24-0,Sotalol (Betapace) is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sulfadoxine (Sulphadoxine),2447-57-6,Sulfadoxine(Sulphadoxine) is an ultra-long-lasting sulfonamide with an IC50 of 249 μg/ml for P. vivax,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tenoxicam (Mobiflex),59804-37-4,Tenoxicam(Mobiflex) is a good HO. radicals scavenger with an IC50 of 56.7 μM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vardenafil Hydrochloride Trihydrate (Vivanza),224785-90-4,Vardenafil Hydrochloride Trihydrate (Vivanza) is a new type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Xylazine HCl,23076-35-9,Xylazine HCl is α2 class of adrenergic receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Maprotiline HCl,10347-81-6,Maprotiline hydrochloride (Deprilept, Ludiomil, Psymion) is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naphazoline HCl (Naphcon),550-99-2,Naphazoline hydrochloride (Naphcon) is an ocular vasoconstrictor and imidazoline derivative sympathomimetic amine.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Epinephrine bitartrate (Adrenalinium),51-42-3,Epinephrine bitartrate (D02149, Adrenalinium) is alpha- and beta-adrenergic receptor stimulator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
L-Adrenaline (Epinephrine),51-43-4,L-Adrenaline (Epinephrine) belongs to a group of the compounds known as catecholamines.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
DL-Adrenaline,329-65-7,DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenytoin sodium (Dilantin),630-93-3,Phenytoin sodium (Dilantin) is an inactive voltage-gated sodium channel stabilizer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenytoin (Lepitoin),57-41-0,Phenytoin (Lepitoin; NSC 8722; Phenytek; Phenytoine; Sodanton; Zentropi) is an inactive voltage-gated sodium channel stabilizer.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Alizarin,72-48-0,Alizarin strongly inhibits P450 isoform CYP1A1, CYP1A2 and CYP1B1 with IC50 of 6.2 μM, 10.0 μM and 2.7 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dopamine HCl (Inotropin),62-31-7,Dopamine hydrochloride (Inotropin) is a catecholamine neurotransmitter present in a wide variety of animals,And a dopamine D1-5 receptors agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Asaraldehyde (Asaronaldehyde),4460-86-0 ,Asaraldehyde (Asaronaldehyde) is natural COX-2 inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ritodrine HCl (Yutopar),23239-51-2,Ritodrine hydrochloride (DU 21220; Miolene; NSC 291565; Pre-Par) is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clomipramine HCl (Anafranil),17321-77-6,Clomipramine hydrochloride (Anafranil) is a hydrochloride salt of clomipramine which is a serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) blocker with Ki of 0.14, 54 and 3 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenformin HCl,834-28-6,Phenformin hydrochloride is a hydrochloride salt of phenformin that is an anti-diabetic drug from the biguanide class.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Scopine,498-45-3,Scopine is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Tiotropium Bromide hydrate,139404-48-1,Tiotropium Bromide hydrate is a monohydrate of tiotropium bromide (Spiriva; Tiova; BA 679BR; tiopropium) that is an anticholinergic and bronchodilator and a muscarinic receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Scopine HCl,85700-55-6,Scopine HCl is the hydrochloride of Scopine, which is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Trospium chloride (Sanctura),10405-02-4,Trospium chloride (Sanctura) is a competitive muscarinic cholinergic receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tolterodine tartrate (Detrol LA),124937-52-6,Tolterodine tartrate (Detrol LA) is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azelastine HCl (Astelin),79307-93-0,Azelastine hydrochloride (Astelin) is a potent, second-generation, selective, histamine antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Daphnetin,486-35-1,Daphnetin is an inhibitor of EGFR, PKA and PKC with IC50 of 7.67 μM, 9.33 μM and 25.01 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clarithromycin (Biaxin, Klacid),81103-11-9,Clarithromycin (Biaxin, Klacid) is a macrolide antibiotic and a CYP3A4 substrate and inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rosiglitazone (Avandia),122320-73-4,Rosiglitazone (Avandia) is a potent antihyperglycemic agent and a potent thiazolidinedione insulin sensitizer with IC50 of 12, 4 and 9 nM for rat, 3T3-L1 and human adipocytes, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amiloride HCl dihydrate,17440-83-4,Amiloride hydrochloride dihydrate is a potent epithelial sodium channel blocker.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clomifene citrate (Serophene),50-41-9,Clomifene citrate (Serophene) is a selective estrogen receptor modulator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hydralazine HCl,304-20-1,Hydralazine hydrochloride is a hydrochloride salt of hydralazine (Apresoline) that is a direct-acting smooth muscle relaxant with an IC50 of 1.9 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Isoprenaline HCl,51-30-9,Isoprenaline is a non-selective β-adrenoceptor, inhibits the 3H-inositol phosphate accumulation with IC50 of 0.08 μM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Medroxyprogesterone acetate,71-58-9,Medroxyprogesterone acetate is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenylephrine HCl,61-76-7,Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tetracaine HCl (Pontocaine),136-47-0,Tetracaine hydrochloride (Pontocaine) is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Phenacetin,62-44-2,Phenacetin is a non-opioid analgesic without anti-inflammatory properties.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zidovudine (Retrovir),30516-87-1,Zidovudine (Retrovir) is a reverse transcriptase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Quinapril HCl (Accupril),82586-55-8,Quinapril hydrochloride (Accupril) is the hydrochloride salt of quinapril that is an angiotensin-converting enzyme inhibitor with a Ki of 20 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Trazodone HCl (Desyrel),25332-39-2,Trazodone is an antidepressant belonging to the class of serotonin receptor antagonists and reuptake inhibitors for treatment of anxiety disorders.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Brompheniramine,980-71-2,Brompheniramine is a histamine H1 receptors antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pioglitazone (Actos),111025-46-8,Pioglitazone (Actos) is a selective peroxisome proliferator-activated receptor gamma stimulator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tolvaptan (OPC-41061),150683-30-0,Tolvaptan (OPC-41061) is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28¦ÌM for the inhibition of AVP-induced platelet aggregation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gliclazide (Diamicron),21187-98-4,Gliclazide (Diamicron) is a whole-cell beta-cell ATP-sensitive potassium currents blocker with an IC50 of 184 ¡À 30 nM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Acemetacin (Emflex),53164-05-9,Acemetacin (Emflex) is a non-steroidal anti-inflammatory drug and a glycolic acid ester of indometacin that is a cyclooxygenase inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tioxolone,4991-65-5,Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor with a Ki of 91 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dehydroepiandrosterone (DHEA),53-43-0,Dehydroepiandrosterone(DHEA) is a 19-carbon endogenous natural steroid hormone.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mifepristone (Mifeprex),84371-65-3,Mifepristone (Mifeprex, RU-486, RU-38486, Mifegyne) is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lonidamine,50264-69-2,Lonidamine is an orally administered small molecule hexokinase inactivator with an IC50 of 0.85 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Ethisterone,434-03-7,Ethisterone is a progestogen hormone being considered to treat prostate cancer.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Arecoline,300-08-3 ,Arecoline is a muscarinic acetylcholine receptor agonist. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Noradrenaline bitartrate monohydrate (Levophed),108341-18-0,Noradrenaline bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-733,1035555-63-5,TAK-733 is a potent, selective, non ATP-competitive MEK inhibitor with IC50 of 3.2 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LDN193189,1062368-24-4,LDN193189 is a selective inhibitor of ALK2 and ALK3 with IC50 of 5 nM and 30 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK256066,801312-28-7,GSK256066 is a selective PDE4B inhibitor with IC50 of 3.2 pM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD5438,602306-29-6 ,AZD5438 is a potent inhibitor of CDK1, CDK2 and CDK9 with IC50 of 16 nM, 6 nM, and 20 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PP-121,1092788-83-4,PP-121 is a multi-target inhibitor of PDGFR, Hck, mTOR, VEGFR2, Src and Abl with IC50 of 2 nM, 8 nM, 10 nM, 12 nM, 14 nM and 18 nM, respectively, and also inhibits DNA-PK with IC50 of 60 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
OSI-027,936890-98-1,OSI-027 is a selective and potent dual inhibitor of mTORC1 and mTORC2 with IC50 of 22 nM and 65 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
R788 (Fostamatinib),901119-35-5,R788 (Fostamatinib) is a Syk inhibitor with IC50 of 41 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2603618 (IC-83),911222-45-2,LY2603618 (IC-83) is a selective Chk1 inhibitor with potential anti-tumor activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tubastatin A HCl,1310693-92-5,Tubastatin A is a potent HDAC6 inhibitor with IC50 of 15 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-05212384 (PKI-587),1197160-78-3,PKI-587 is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PNU-120596,501925-31-1,PNU-120596 is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM in α7*-expressing SH-EP1 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW3965 HCl,405911-17-3,GW3965 is a potent, selective LXR agonist, which exhibits its potency in the LXRα/SRC1 LiSA and LXRα-GAL4 with EC50 of 125 nM and 190 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
URB597,546141-08-6 ,URB597 (KDS-4103) is a potent FAAH inhibitor with IC50 of 4.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMS-806 (BMS 378806),357263-13-9 ,BMS-806 (BMS 378806) selectively inhibitis the binding of HIV-1 gp120 to the CD4 receptor with EC50 of 0.85-26.5 nM in virus.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
DCC-2036 (Rebastinib),1020172-07-9,DCC-2036 is a conformational control inhibitor of Abl1 and Abl1(T315I) with IC50 of 0.8 nM and 4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CCT128930,885499-61-6,CCT128930 is a potent, ATP-competitive and selective inhibitor of Akt2 with IC50 of 6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A66,1166227-08-2 ,A66 is a potent and specific p110α inhibitor with IC50 of 32 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-875,1374598-80-7,TAK-875 is a selective GPR40 agonist with EC50 of 14 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NU7441 (KU-57788),503468-95-9 ,NU7441 is a highly potent and selective DNA-PK inhibitor with IC50 of 14 nM and also inhibits PI3K with IC50 of 5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SNX-2112,908112-43-6,SNX-2112 selectively binds to the ATP pocket of HSP90α and HSP90β with Ka of 30 nM and 30 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-04929113 (SNX-5422),908115-27-5,PF-04929113 (SNX-5422) is a potent and selective HSP90 inhibitor with Kd of 41 nM and also inhibits Her-2 degradation with IC50 of 37 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK2126458,1086062-66-9 ,GSK2126458 is a highly selective and potent inhibitor of p110α, p110β, p110γ, p110δ, mTORC1 and mTORC2 with Ki of 0.019 nM, 0.13 nM, 0.024 nM, 0.06 nM, 0.18 nM and 0.3 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
5-hydroxymethyl tolterodine (PNU 200577),207679-81-0,5-hydroxymethyl tolterodine (PNU 200577) is a new muscarinic receptor antagonist with Kb of 0.84 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-0752,471905-41-6 ,MK-0752 is a moderately potent γ-secretase inhibitor, which reduces Aβ40 production with IC50 of 5 nM in human SH-SY5Y cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WYE-125132,1144068-46-1,WYE-125132 is a highly potent, ATP-competitive and specific mTOR inhibitor with IC50 of 0.19 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WAY-100635 HCl,146714-97-8,WAY 100635 is a potent and selective 5-HT agonist with IC50 of 0.95 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clinofibrate,30299-08-2,Clinofibrate inhibits hydroxymethylglutaryl coenzyme A reductase (HMGCR) with IC50 of 0.47 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ciprofibrate,52214-84-3,Ciprofibrate is a peroxisome proliferator-activated receptor agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-3845,1196109-52-0,PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
S/GSK1349572 (GSK1349572),1051375-16-6,S/GSK1349572 (GSK1349572) is a two-metal-binding HIV integrase inhibitor with IC50 of 2.7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WYE-687,1062161-90-3,WYE-687 is an ATP-competitive and selective inhibitor of mTOR with IC50 of 7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY310762,192927-92-7,LY310762 is a 5-HT1D antagonist with Ki of ~0.2 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A-674563,552325-73-2,A-674563 inhibits Akt1, PKA and CDK2 with Ki of 11 nM, 16 nM and 46 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AS-252424,900515-16-4,AS-252424 is a novel, potent and selective inhibitor of PI3Kγ with IC50 of 33 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-00562271,939791-38-5,PF-00562271 is the benzenesulfonate salt of PF-562271, which is a potent, ATP-competitive, reversible inhibitor of FAK and Pyk2 with IC50 of 1.5 nM and 14 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1120212 (Trametinib),871700-17-3,GSK1120212 (JTP-74057, trametinib) is a highly specific and potent MEK1 and MEK2 inhibitor with IC50 of 0.92 nM and 1.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A 922500,959122-11-3,A 922500 is a DGAT-1 inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BRL-15572,193611-72-2,BRL-15572 is a 5-HT1D antagonist with pKi of 7.9.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NSC-207895 (XI-006),58131-57-0,NSC-207895 suppresses MDMX with IC50 of 2.5 ¦ÌM, leading to enhanced p53 stabilization/activation and DNA damage, and also regulate MDM2, an E3 ligase,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flavopiridol (Alvocidib) HCl,131740-09-5,Flavopiridol competes with ATP to inhibit CDKs including CDK1, CDK2, CDK4 and CDK6 with IC50 of ~ 40 nM, and CDK7 with IC50 of 300 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PCI-32765 (Ibrutinib),936563-96-1,PCI-32765 (Ibrutinib) is a potent and highly selective Btk inhibitor with IC50 of 0.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AS-604850,648449-76-7 ,AS-604850 is a selective, ATP-competitive PI3Kγ inhibitor with IC50 of 250 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CAY10505,1218777-13-9 ,CAY10505 is a PI3Kγ inhibitor with IC50 of 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CHIR-124,405168-58-3,CHIR-124 is a novel and potent Chk1 inhibitor with IC50 of 0.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CX-5461,1138549-36-6,CX-5461 selectively inhibits Pol I-driven transcription of rRNA with IC50 of 142 nM in HCT-116 cells. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KW-2478,819812-04-9,KW-2478 is a nonansamycin HSP90 inhibitor with IC50 of 3.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-BSK805 2HCl,1092499-93-8 (free base),NVP-BSK805 is a potent and selective ATP-competitive JAK2 inhibitor with IC50 of 0.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
R547,741713-40-6,R547 is a potent and selective CDK inhibitor with Ki and IC50 of 1-3 nM and 80 nM respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WAY-600,1062159-35-6 ,WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ADX-47273,851881-60-2,ADX47273 is a potent and specific mGlu5 antagonist with IC50 of 0.17μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BMY 7378,21102-95-4,BMY 7378 is a multiple inhibitors of α2C-adrenoceptor and α1D-adrenoceptor with pKi of 6.54 and 8.2, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TG101209,936091-14-4,TG101209 is a potent inhibitor of JAK2, Flt3 and RET with IC50 of 6 nM, 25 nM and 17 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WAY-362450,629664-81-9,WAY-362450 is a potent, selective FXR agonist with EC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GDC-0980 (RG7422),1032754-93-0,GDC-0980 (RG7422) is a potent, selective inhibitor of PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ with IC50 of 5 nM, 27 nM, 7 nM, and 14 nM, and also a mTOR inhibitor with Ki of 17 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A-769662,844499-71-4,A-769662 is a potent, reversible AMPK activator with EC50 of 0.8 μM and inhibits fatty acid synthesis with IC50 of 3.2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
RS-127445,199864-87-3,RS-127445 is a selective 5-HT2B antagonist with pKi of 9.5 and pIC50 of 10.4.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CH5132799,1007207-67-1,CH5132799 exhibits a strong inhibitory activity especially against PI3Kα with IC50 of 14 nM and also inhibits mTOR with IC50 of 1.6 µM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KX2-391,897016-82-9,KX2-391 (KX01) is a highly selective non ATP-competitive Src inhibitor with GI50 of 9-60 nM in cancer cell lines .,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1838705A,1116235-97-2,GSK1838705A is a potent inhibitor of IGF-1R, IR and ALK with IC50 of 2.0 nM, 1.6 nM and 0.5 nM, respectively,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2109761,700874-71-1 ,LY2109761 is a novel selective TGF-β receptor type I/II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
YO-01027,209984-56-5,YO-01027 (Dibenzazepine, DBZ) is a dipeptidic γ-secretase inhibitor with IC50 of 2.6 nM and 2.9 nM for APPL and Notch, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Geldanamycin,30562-34-6,Geldanamycin is a natural existing HSP90 inhibitor with Kd of 1.2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY411575,209984-57-6,LY-411575 is a potent γ-secretase inhibitor with IC50 of 0.078 nM and 0.082 nM for membrane- and cell-based γ-secretase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CP-91149,186392-40-5,CP-91149 is a selective glycogen phosphorylase (GP) inhibitor with IC50 of 0.13 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-901,934541-31-8,TAK-901 is a novel inhibitor of Aurora A and Aurora B with IC50 of 21 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AMG 900,945595-80-2,AMG 900 is a potent and highly selective pan-Aurora inhibitor for Aurora A, Aurora B and Aurora C with IC50 of 5 nM, 4 nM and 1 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZM 336372,208260-29-1,ZM 336372 is a potent and selective c-Raf inhibitor with IC50 of 70 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nilvadipine (ARC029),75530-68-6,Nilvadipine (ARC029) is a potent calcium channel blocker with an IC50 of 0.03 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JTC-801,244218-51-7,JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-03814735,942487-16-3,PF-03814735 is a novel, potent and reversible inhibitor of both Aurora A and Aurora B with IC50 of 0.8 nM and 5 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PH-797804,586379-66-0,PH-797804 is a novel pyridinone inhibitor of p38α with IC50 of 26 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dacomitinib (PF299804,PF-00299804),1110813-31-4,PF299804 is a potent, irreversible pan-ErbB inhibitor against ErbB1, ErbB2 and ErbB4 with IC50 of 6 nM, 45.7 nM and 73.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AG-1478 (Tyrphostin AG-1478),153436-53-4,AG-1478 (Tyrphostin AG-1478) is a selective EGFR inhibitor with IC50 of 3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 415286,264218-23-7,SB 415286 is a potent GSK3α and GSK3β inhibitor with IC50 of 78 nM and ~78 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Crenolanib (CP-868596),670220-88-9,Crenolanib (CP-868596) is a potent and selective inihibitor of PDGFRα with IC50 of 10 nM in PDGFRα over-expressed CHO cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZ 3146,1124329-14-1,AZ3146 is a selective Mps1 inhibitor with IC50 of ~35 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TG101348 (SAR302503),936091-26-8,TG-101348 (SAR302503) is a selective inhibitor of JAK2 with IC50 of 3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PAC-1,315183-21-2,PAC-1 is a potent procaspase-3 activator with EC50 of 0.22 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PKI-402,1173204-81-3,PKI-402 is a potent dual PI3K/mTOR inhibitor targeting PI3Kα, PI3Kβ, PI3Kγ, PI3Kδ and mTOR with IC50 of 2 nM, 7 nM, 16 nM, 14 nM, and 3 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK1070916,942918-07-2,GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B and Aurora C with IC50 of 3.5 nM and 6.5 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PHA-767491,845714-00-3,PHA-767491 is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and 34 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-04691502,1013101-36-4 ,PF-04691502 is an ATP-competitive, selective inhibitor of PI3K(α/β/δ/γ)/mTOR with Ki of 1.8 nM/2.1 nM/1.6 nM/1.9 nM and 16 nM, also inhibits Akt phosphorylation on T308/S473 with IC50 of 7.5 nM/3.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CCT137690,1095382-05-0,CCT137690 is a highly selective inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 15 nM, 25 nM and 19 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CHIR-98014,252935-94-7,CHIR-98014 is a potent and selective GSK-3 inhibitor for GSK-3ɑ and GSK-3β with IC50 of 0.65 nM and 0.58 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZ628,878739-06-1,AZ628 is a potent inhibitor for wild-type CRAF and BRAFV600E with IC50 of 29 nM and 34 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AMG458,913376-83-7 ,AMG 458 is a potent c-Met inhibitor of human c-Met and mouse c-Met with Ki of 1.2 nM or 2.0 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Anacetrapib (MK-0859),875446-37-0,Anacetrapib (MK0859) is a potent and selective rhCETP and mutant CETP(C13S) inhibitor with IC50 of 7.9 nM and 11.8 nM, respectively,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-BGT226,1245537-68-1,NVP-BGT226 is a novel dual PI3K/mTOR inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW788388,452342-67-5,GW788388 is a potent and selective inhibitor of ALK5 with IC50 of 18 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Milciclib (PHA-848125),802539-81-7,PHA-848125 is a potent, ATP-competitive cyclin A/CDK2 inhibitor with IC50 of 45 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Arry-380,937265-83-3,ARRY-380 is a potent and selective HER2 inhibitor with IC50 of 8 nM and also inhibits EGFR with IC50 of 4 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT-406,1071992-99-8,AT-406 is a potent IAP (inhibitor of apoptosis protein via E3 ubiquitin ligase) inhibitor of XIAP, cIAP1, and cIAP2 with Ki of 66.4 nM, 1.9 nM, and 5.1 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ARRY334543,845272-21-1,ARRY334543 is a selective and potent ErbB1 and ErbB2 inhibitor with IC50 of 7 nM and 2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Wortmannin,19545-26-7,Wortmannin is a multi-target inhibitor of MLCK and PI3K with IC50 of 170 nM and 3 nM, also blocks autophagosome formation and potently inhibits DNA-PK/ATM with IC50 of 16 nM and 150 nM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PI3K/HDAC Inhibitor I,1339928-25-4,PI3K/HDAC Inhibitor I is a dual PI3K and HDAC inhibitor for PI3Kɑ, HDAC1, HDAC2, HDAC3 and HDAC10 with IC50 of 19 nM, 1.7 nM, 5 nM, 1.8 nM and 2.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Canagliflozin,842133-18-0,Canagliflozin is a highly potent and selective SGLT2 inhibitor for CHO-hSGLT2, CHO-rSGLT2 and CHO-mSGLT2 with IC50 of 4.4 nM, 3.7 nM and 2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-BVU972,1185763-69-2,NVP-BVU972 is a selective and potent Met inhibitor with IC50 of 14 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CH5424802,1256580-46-7,CH5424802 is a potent and selective ALK inhibitor with IC50 of 1.9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-2048,869901-69-9,MK-2048 is an potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
3-Methyladenine,5142-23-4,3-Methyladenine (3-MA) is a selective PI3K inhibitor for Vps34 and PI3Kγ with IC50 of 25 μM and 60 μM and also blocks autophagosome formation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dinaciclib (SCH727965),779353-01-4,Dinaciclib (SCH727965) is a novel and potent CDK inhibitor for CDK2, CDK5, CDK1 and CDK9 with IC50 of 1 nM, 1 nM, 3 nM and 4 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dovitinib Dilactic acid (TKI258 Dilactic acid) ,852433-84-2,Dovitinib (TKI258, CHIR-258) is a multitargeted tyrosine kinase inhibitor of FLT3 and c-KIT with IC50 of 1 nM and 2 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-5108 (VX-689),1010085-13-8,MK-5108 (VX-689) is a highly selective Aurora A inhibitor with IC50 of 0.064 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dalcetrapib (JTT-705),211513-37-0,Dalcetrapib (JTT-705) is a rhCETP inhibitor with IC50 of 0.2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB705498,501951-42-4,SB705498 is a TRPV1 antagonist for hTRPV1 with pIC50 and pKi of 7.1 and 7.6 in HEK293 cells. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MK-2461,917879-39-1,MK-2461 is a potent inhibitor of c-Met, Ron, Flt1/3, PDGFRβ, Mer and FGFR1/2/3 with IC50 of 2.5 nM, 7 nM, 10 nM/22 nM, 22 nM, 24 nM and 65 nM/39 nM/50 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nocodazole,31430-18-9,Nocodazole inhibits Abl, Abl(E255K) and Abl(T315I) with IC50 of 0.21 μM, 0.53 μM and 0.64 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CPI-613,95809-78-2,CPI-613 inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-5274857,1373615-35-0,PF-5274857 is a potent and selective Smoothened (Smo) antagonist with IC50 and Ki of 5.8 nM and 4.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW842166X,666260-75-9,GW842166X is a potent and highly selective agonist of CB2 receptor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
M344,251456-60-7 ,M344 is a potent HDAC inhibitor with IC50 of 100 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
RITA (NSC 652287),213261-59-7,RITA (NSC 652287) is a DNA damaging agent with IC50 of 2 nM and 20 nM in A498 and TK-10 cells, and also inhibits MDM2-p53 interaction by targeting to p53.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW4064,278779-30-9,GW 4064 is an agonist of farnesoid X receptor (FXR) with EC50 of 65 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD2014,1009298-59-2,AZD2014 is a novel dual mTORC1 and mTORC2 inhibitor with potential antineoplastic activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-285,871026-44-7,TAK-285 is a novel dual HER2 and EGFR inhibitor with IC50 of 17 nM and 23 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A-803467,944261-79-4,A-803467 is a selective NaV1.8 channel blocker with IC50 of 8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
INCB28060,1029712-80-8,INCB28060 is a novel, ATP-competitive inhibitor of c-MET with IC50 of 0.13 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tofacitinib (CP-690550, Tasocitinib),477600-75-2,CP-690550 is a novel inhibitor of JAK3 with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Istradefylline (KW-6002),155270-99-8,Istradefylline (KW-6002) is a selective adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sotrastaurin (AEB071),425637-18-9,Sotrastaurin (AEB071) is a potent selective pan-PKC inhibitor and highly inhibits PKCθ with Ki of 0.22 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Torcetrapib (CP-529414),262352-17-0,Torcetrapib (CP-529414) is a CETP inhibitor with IC50 of 37 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VU 0357121,433967-28-3,VU0357121 is a novel allosteric modulator of mGlu5 with EC50 of 33 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WP1066,857064-38-1,WP1066 is a novel inhibitor of JAK2 and STAT3 with IC50 of 2.30 μM and 2.43 μM in HEL cells .,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lonafarnib (SCH66336),193275-84-2,Lonafarnib (SCH 66336) is a selectively FPTase inhibitor for H-ras, K-ras-4B and N-ras with IC50 of 1.9 nM, 5.2 nM and 2.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
APO866 (FK866),658084-64-1,APO866 effectively inhibits NAMPT with IC50 of 0.09 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD4547,1035270-39-3,AZD4547 is a novel selective FGFR inhibitor targeting FGFR1, FGFR2, and FGFR3 with IC50 of of 0.2 nM, 2.5 nM, and 1.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BAY80-6946,1032568-63-0,BAY 80-6946 is a potent and highly selective reversible PI3K inhibitor for PI3Kα and PI3Kβ with IC50 of 0.469 nM and 3.72 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Galeterone (TOK-001),851983-85-2,Galeterone (TOK-001, VN/124-1) is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sirtinol,410536-97-9,Sirtinol is a specific SIRT1 and SIRT2 inhibtor with IC50 of 131 μM and 38 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY364947,396129-53-6,LY364947 is a potent ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CEP33779,1257704-57-6,CEP33779 is a selective JAK2 inhibitor with IC50 of 1.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dabrafenib (GSK2118436),1195765-45-7,Dabrafenib (GSK2118436) is a potent ATP-competitive inhibitor of B-Raf, B-RafV600E and c-Raf with IC50 of 3.2 nM, 0.8 nM and 5.0 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GDC-0068,1001264-89-6,GDC-0068 is a highly selective pan-Akt inhibitor targeting Akt1, Akt2 and Akt3 with IC50 of 5 nM, 18 nM and 8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MPEP,96206-92-7,MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
INK 128 (MLN0128),1224844-38-5,INK 128 is a potent and selective mTOR inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AT101,90141-22-3,AT-101 is a BH3 mimetic known to be a potent inhibitor of antiapoptotic Bcl-2 family members.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ciproxifan,184025-19-2,Ciproxifan is a highly potent and selective H3-receptor antagonist with IC50 of 9.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BYL719,1217486-61-7,BYL719 strongly and selectively inhibits PI3Kα.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tyrphostin AG 879 (AG 879),148741-30-4,AG879 inhibits both ErbB2 and Flk-1 with IC50 of 1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Torin 2,1223001-51-1,Torin 2 is a highly potent and selective mTOR inhibitor with IC50 of 0.25 nM, and also exhibits potent cellular activity against ATM/ATR/DNA-PK with EC50 of 28 nM, 35 nM and 118 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CI994 (Tacedinaline),112522-64-2,CI994 (Tacedinaline) is an anti-cancer drug which inhibits HDAC1 with IC50 of 0.57 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AM251,183232-66-8,AM251 is a cannabinoid 1 receptor antagonist with IC50 of 8.9 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NVP-TAE226,761437-28-9,NVP-TAE226, a potent dual FAK/IGF-1R, inhibiting FAK and IGF-1R with IC50 of 5.5 nM and 0.14 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
RG108,48208-26-0,RG108 is an inhibitor of DNA methyltransferase with IC50 of 115 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tideglusib,865854-05-3 ,Tideglusib (NP031112, NP-12) is a potent non ATP-competitive inhibitor of GSK3 with IC50 of 60 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TPCA-1,507475-17-4,TPCA-1 is an inhibitor of IKK-2 with IC50 of 17.9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ML133 HCl,1222781-70-5,ML133 is a potent potassium channel inhibitor for Kir2.1 with IC50 of 1.8 μM (pH 7.4) and 290 nM (pH 8.5).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Desmethyl Erlotinib (CP-473420),183321-86-0,Desmethyl Erlotinib (CP-473420) is a free base of OSI-420, which is an active metabolite of Erlotinib which is an orally active EGFR inhibitor for human EGFR with IC50 of 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Torin 1,1222998-36-8,Torin1 is a potent inhibitor of mTOR with IC50 of 2-10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ 1661010,681136-29-8,JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Epiandrosterone (3β-androsterone),481-29-8,Epiandrosterone (3β-androsterone) is a steroid hormone with weak androgenic activity which acts as a L-type Ca2+ channel antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ARN-509,956104-40-8,ARN-509 is a selective androgen receptor inhibitor with IC50 of 16 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SAR131675,,SAR131675 is a VEGFR-3 inhibitor with IC50 of 20 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BI-D1870,501437-28-1,BI-D1870 is an ATP-competitive inhibitor of ribosomal S6 for RSK1, RSK2, RSK3 and RSK4 with IC50 of 31 nM, 24 nM, 18 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Semaxanib (SU5416),194413-58-6,Semaxanib (SU5416) is a potent and selective VEGFR (Flk-1/KDR) inhibitor with IC50 of 1.04 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cathepsin Inhibitor 1,225120-65-0,Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB-269970 HCl,261901-57-9,SB-269970 HCl is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with pKi of 8.3.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Baricitinib (LY3009104, INCB28050),1187594-09-7,Baricitinib is a selective JAK1 and JAK2 inhibitor with IC50 of 5.9 nM and 5.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BRL 54443,57477-39-1,BRL 54443 is a 5-HT1E and 5-HT1F receptor agonist with pKi of 8.7 and 9.25, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Carfilzomib (PR-171),868540-17-4,Carfilzomib (PR-171) is a proteasome inhibitor with IC50 less than 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BML-190,2854-32-2,BML-190 is a selective CB2 inverse agonist with Ki of 435 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
MRS 2578,711019-86-2,MRS2578 is a potent P2Y6 receptor with IC50 of 37 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SB 271046,209481-20-9,SB-271046 is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dizocilpine (MK 801),77086-21-6,Dizocilpine is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
StemRegenin 1,1227633-49-9,StemRegenin 1 is an AhR inhibitor with IC50 of 127 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Golvatinib (E7050),928037-13-2,E7050 is a dual c-Met and VEGFR-2 inhibitor with IC50 of 14 nM and 16 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
IEM 1754 dihydrobroMide,162831-31-4,IEM 1754 dihydrobroMide  is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CTEP,871362-31-1,CTEP is a selective allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
 VU 0364770,61350-00-3,VU 0364770 is a selective positive allosteric mGlu4 with EC50 of 1.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ML130,799264-47-4,ML130 is a potent and selective inhibitor of NOD1 with IC50 of 0.56 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
IMD 0354,978-62-1,IMD-0354 is an IKKβ inhibitor and blocks IκBα phosphorylation in NFκβ pathway.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VUF 10166,155584-74-0,VUF10166 is a novel, potent and competitive antagonist to 5-HT3A with Ki of 0.04 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
U-104,178606-66-1,U-104 is a potent carbonic anhydrase (CA) inhibitor for CA IX and CA XII with IC50 of 45.1 nM and 4.5 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WHI-P154,211555-04-3,WHI-P154 is a potent JAK3 inhibitor with IC50 of 1.8 μM and also inhibits EGFR with IC50 of 4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Alogliptin (SYR-322),850649-61-5,Alogliptin(SYR-322) is a potent, selective inhibitor of DPP-4 with IC50 of < 10 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
 TG 100713,925705-73-3,TG 100713 is a PI3K inhibitor for PI3Kγ, PI3Kδ, PI3Kα and PI3Kβ with IC50 of 50 nM, 24 nM, 165 nM and 215 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
T0070907,313516-66-4,T0070907 is a potent and selective PPARγ inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW5074,220904-83-6,GW5074 is a potent and selective c-Raf inhibitor with IC50 of 9 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Camostat Mesilate (FOY-305),59721-29-8,Camostat is a trypsin-like protease inhibitor, inhibiting matriptase and human neutrophil elastase with IC50 of 0.5 μM and 0.2 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Prucalopride,179474-81-8,Prucalopride is a selective, high affinity 5-HT receptor agonistfor 5-HT4a and 5-HT4b with Ki of 2.5 nM and 8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
(-)-MK 801 Maleate,121917-57-5,MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
L-NAME HCl,51298-62-5,L-NAME is a nonselective inhibitor of nitric oxide synthetases (NOS) for nNOS (bovine), eNOS (human), and iNOS (murine), with Ki of 15 nM, 39 nM and 4.4 μM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
IKK-16,873225-46-8,IKK 16 is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
A 205804,251992-66-2,A-205804 is a potent and selective inhibitor of E-selectin and ICAM-1 expression with IC50 of 20 nM and 25 nM respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-562271,717907-75-0,PF-562271 is a potent, ATP-competitive, reversible inhibitor of FAK and Pyk2 with IC50 of 1.5 nM and 14 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW441756,504433-23-2,GW 441756 is a potent, selective inhibitor of TrkA with IC50 of 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"VU 0361737,1161205-04-4,VU 0361737 is a selective positive allosteric modulator for mGlu4 receptor with EC50 of 240 nM and 110 nM at human and rat receptors, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
SB-742457,607742-69-8,SB-742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tyrphostin 9 (SF 6847),10537-47-0,SF 6847 is an inhibitor of EGFR with IC50 of 460 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZM 323881 HCl,193000-39-4,ZM-323881 is a potent and selective inhibitor of VEGFR2 with IC50 < 2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZM 306416,690206-97-4,ZM-306416 is a VEGFR inhibitor, inhibiting Src, VEGFR1 and Abl with IC50 of 0.33 μM, 0.33 μM and 1.3 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GNF-2,778270-11-4,GNF-2 is a highly selective non-ATP competitive inhibitor of Bcr-Abl, inhibiting the proliferation of the Bcr-Abl-expressing cells with IC50 of 138 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cobicistat (GS-9350),1004316-88-4,Cobicistat (GS-9350) is a potent and selective inhibitor of CYP3A with IC50 of 30-285 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CCG 50014,883050-24-6,CCG 50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
S-Ruxolitinib,941685-37-6,S-Ruxolitinib is a JAK family inhibitor for JAK1 and JAK2 with IC50 of 3.3 nM and 2.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lumiracoxib (COX-189),220991-20-8,Lumiracoxib (COX-189) is a novel, selective COX-2 inhibitor with Ki of 0.06 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF 477736,952021-60-2,PF 477736 is a ChK inhibitor against ChK1, ChK2, VEGFR2, Yes and Fms with IC50 of 0.49 nM, 47 nM, 8 nM, 14 nM and 10 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
JNJ-7777120,459168-41-3,JNJ-7777120 is a potent and selective non-imidazole histamine H4 receptor antagonist with Ki of 4.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ki16198,355025-13-7,Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pirfenidone,53179-13-8,Pirfenidone inhibits TGF-β bioactivity by affecting TGF-β2 mRNA expression and processing of pro-TGF-β in CCL-64 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Go 6983,133053-19-7,Go 6983 is a pan PKC inhibitor against PKCα, PKCβ, PKCγ, PKCδ, PKCζ with IC50 of 7 nM, 7 nM, 6 nM, 10 nM and 60 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WZ 811,55778-02-4,WZ811 is a highly potent competitive CXCR4 antagonist with EC50 of 0.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BAY 11-7082 (BAY 11-7821),19542-67-7,Bay 11-7082 inhibits TNFα-induced IκBα phosphorylation with IC50 of 10 μM and inactivates the E2-conjugating enzymes Ubc (ubiquitin conjugating) 13, UbcH7 and the E3 ligase LUBAC (linear ubiquitin assembly complex).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dapivirine,244767-67-7,Dapivirine is an nonnucleoside reverse transcriptase inhibitor for HIV reverse transcriptase with IC50 of 24 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW9662,22978-25-2,GW9662 is a selective PPAR antagonist, inhibiting PPARγ, PPARα and PPARδ with IC50 of 3.3 nM, 32 nM and 2 μM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
HC-030031,349085-38-7,HC-030031 is a selective TRPA1 channel blocker that antagonizes AITC- and formalin-evoked calcium influx with IC50 of 6.2 μM and 5.3 μM respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
IOX2,931398-72-0,IOX2 is a potent inhibitor of HIF-1α prolyl hydroxylase-2 (PHD2) with IC50 of 21 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mozavaptan,137975-06-5,Mozavaptan (OPC-31260) is a novel competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PF-4981517,1390637-82-7,PF-4981517 is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Icotinib,610798-31-7,Icotinib is a potent and specific epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) with IC50 of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Salubrinal,405060-95-9,Salubrinal is a selective inhibitor of eIF2α dephosphorylation and inhibits ER stress-mediated apoptosis with EC50 of ~15 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CHIR-99021 (CT99021) HCl,252917-06-9 (free base),CHIR-99021 HCl (CT99021) is hydrochloride of CHIR-99021, which is a GSK-3α and GSK-3β inhibitor with IC50 of 10 nM and 6.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Evacetrapib (LY2484595),1186486-62-3,LY2484595 is a potent and selective inhibitor of CETP with IC50 of 5.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TDZD-8,327036-89-5 ,TDZD-8 is a non-ATP competitive GSK-3β inhibitor with IC50 of 2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apoptosis Activator 2,79183-19-0,Apoptosis Activator 2 activates caspases in a cytochrome c-dependent manner and induces apoptosis in tumor cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK 715,303162-79-0,TAK 715 is a p38 MAPK inhibitor for p38α with IC50 of 7.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pifithrin-α,63208-82-2,Pifithrin-α is an inhibitor of p53, inhibiting p53-dependent transactivation of p53-responsive genes.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rivaroxaban (Xarelto),366789-02-8,Rivaroxaban (Xarelto, BAY 59-7939) is a direct inhibitor of Factor Xa with Ki and IC50 of 0.4 nM and  0.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Paroxetine HCl,78246-49-8,Paroxetine is an antidepressant drug of the SSRI type.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
"Zaltoprofen,74711-43-6,Zaltoprofen is an inhibitor of Cox-1 and Cox-2 for treatment of arthritis.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Pazopanib,444731-52-6,Pazopanib is a potent and selective multi-targeted receptor tyrosine kinase inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR-α/β, and c-Kit. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Plerixafor 8HCl (AMD3100 8HCl),155148-31-5,Plerixafor 8HCl (DB06809, Mozobil, AMD3100) is the hydrochloride of Plerixafor, a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aspirin (Acetylsalicylic acid),50-78-2,Aspirin is a salicylate drug, often used as an analgesic to relieve minor aches and pains, as an antipyretic to reduce fever, and as an anti-inflammatory medication.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Niflumic acid,4394-00-7,Niflumic acid is an inhibitor of cyclooxygenase-2 used for joint and muscular pain.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Ciclopirox ethanolamine,41621-49-2,Ciclopirox ethanolamine (Ciclopirox olamine, HOE 296) is a broad-spectrum antifungal agent working as an iron chelator.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rimonabant (SR141716),168273-06-1,Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bufexamac,2438-72-4,Bufexamac is a COX inhibitor for IFN-α release with EC50 of 8.9 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lamotrigine,84057-84-1,Lamotrigine is a novel anticonvulsant drug for inhibition of 5-HT with IC50 of 240 μM and 474 μM in human platelets and rat brain synaptosomes, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PMSF (Phenylmethylsulfonyl Fluoride),329-98-6,PMSF (Phenylmethyl sulfonyl fluoride) is an irreversible serine/cysteine protease inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Piceatannol,10083-24-6,Piceatannol is a selective Syk inhibitor with IC50 of ~10 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Niclosamide (Niclocide),50-65-7,Niclosamide can inhibit DNA replication and inhibit STAT with IC50 of 0.7 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Linagliptin (BI-1356),668270-12-0,Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bindarit ,130641-38-2,Bindarit exhibits selective inhibition against monocyte chemotactic proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vildagliptin (LAF-237),274901-16-5,Vildagliptin (LAF-237) inhibits DPP−4 with IC50 of 2.3 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sitaxentan sodium (TBC-11251),210421-74-2,Sitaxentan sodium (TBC-11251) is a selective endothelin receptor-A antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Daunorubicin HCl (Daunomycin HCl),23541-50-6,Daunorubicin HCl inhibits both DNA and RNA synthesis and inhibits DNA synthesis with Ki of 0.02 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pravastatin sodium,81131-70-6,Pravastatin sodium is an HMG-CoA reductase inhibitor against sterol synthesis with IC50 of 5.6 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bepotastine Besilate,190786-44-8,Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fosaprepitant dimeglumine,265121-04-8,Fosaprepitant (MK-0517, L-758,298) is a water-soluble phosphoryl prodrug for Aprepitant which is a NK1 antagonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rofecoxib (Vioxx),162011-90-7,Rofecoxib (Vioxx) is a COX-2 inhibitor with IC50 of 18 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lurasidone HCl,367514-88-3,Lurasidone is an atypical antipsychotic, inhibits Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C with IC50 of 1.68 nM, 2.03 nM, 0.495 nM, 6.75 nM and 10.8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azilsartan (TAK-536),147403-03-0,Azilsartan (TAK-536) is an angiotensin II type 1 (AT1) receptor antagonist with IC50 of 2.6 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Otilonium Bromide,26095-59-0,Otilonium bromide is an antimuscarinic.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Solifenacin succinate,242478-38-2,Solifenacin succinate is a urinary antispasmodic of the antimuscarinic class.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Palonosetron HCl,135729-62-3,Palonosetron HCl is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bosentan Hydrate,157212-55-0,Bosentan is an endothelin (ET) receptors antagonist for ET-A and ET-B with Ki of 4.7 nM and 95 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rupatadine Fumarate,182349-12-8,Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azelnidipine,123524-52-7,Azelnidipine is a dihydropyridine calcium channel blocker.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Miltefosine (Hexadecylphosphocholine),58066-85-6,Miltefosine inhibits PI3K/Akt activity with ED50 of 17.2 μM and 8.1 μM in carcinoma cell lines A431 and HeLa.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azilsartan Medoxomil (TAK-491),863031-21-4,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Medetomidine HCl,86347-15-1,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ambroxol HCl,23828-92-4,Ambroxol HCl is a potent inhibitor of the neuronal Na+ channels with IC50 of 35.2 μM and 22.5 μM for tonic and phasic block, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amikacin sulfate,39831-55-5,Amikacin sulfate binds to 16S rRNA (bacterial 30S ribosome), causing misreading of mRNA and supressing proteins synthesis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Naloxone HCl,357-08-4,Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Piracetam,7491-74-9,Piracetam is a cyclic derivative of the neurotransmitter  gamma-aminobutyric acid (GABA), used in treatment of a wide range of cognitive disorders.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
(R)-baclofen,69308-37-8,(R)-baclofen is a derivative of gamma-aminobutyric acid primarily used to treat spasticity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dexmedetomidine,113775-47-6,Dexmedetomidine is a sedative medication used by intensive care units and anesthetists.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Etravirine (TMC125),269055-15-4,Etravirine (TMC125) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used for the treatment of HIV.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ulipristal,126784-99-4,Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Indacaterol Maleate,753498-25-8,Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oxybutynin chloride,1508-65-2,Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Milnacipran HCl,101152-94-7,Milnacipran inhibits both norepinephrine transporter (NET) and norepinephrine transporter (SERT) with IC50 of 77 nM and 420 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Darifenacin HBr,133099-07-7,Darifenacin is a selective M3 muscarinic receptor antagonist with pKi of 8.9.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tripelennamine HCl,154-69-8,Tripelennamine is a widely used H1 antagonist, inhibiting PhIP glucuronidation with IC50 of 30 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Entacapone,130929-57-6,Entacapone inhibits catechol-O-methyltransferase(COMT) with IC50 of 151 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Estradiol valerate,979-32-8,Estradiol is a synthetic ester used to treat menopausal symptoms and hormone deficiencies.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Gliquidone,33342-05-1,Gliquidone is an ATP-sensitive K+ channel antagonist with IC50 of 27.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ethynodiol diacetate,297-76-7,Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Benztropine mesylate,132-17-2,Benztropine is a dopamine transporter (DAT) inhibitor with IC50 of 118 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Abacavir sulfate,188062-50-2,Abacavir is a commonly used nucleoside analogue with potent antiviral activity against HIV-1.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Altrenogest,850-52-2,Altrenogest is a progestogen structurally related to veterinary steroid trenbolone.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Anagrelide HCl ,58579-51-4,Anagrelide is a drug used for the treatment of essential thrombocytosis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Atomoxetine HCl,82248-59-7,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Betahistine 2HCl,5579-84-0,Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Brinzolamide,138890-62-7,Brinzolamide is a potent carbonic anhydrase II inhibitor with IC50 of 3.19 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flumequine,42835-25-6,Flumequine is a synthetic chemotherapeutic antibiotic, inhibiting topoisomerase II with IC50 of 15 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Amitriptyline HCl ,549-18-8,Amitriptyline inhibits serotonin receptor, norepinephrine receptor, 5-HT4, 5-HT2 and sigma 1 receptor with IC50 of 3.45 nM, 13.3 nM, 7.31 nM, 235 nM and 287 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Adrenalone HCl,62-13-5,Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Azatadine dimaleate,3978-86-7,Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ropinirole HCl,91374-20-8,Ropinirole a selective dopamine D2 receptors inhibitor with IC50 of 29 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Reboxetine mesylate,98769-84-7,Reboxetine is a norepinephrine reuptake inhibitor with Ki of 8.2 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Triflusal,322-79-2,Triflusal irreversibly inhibits the production of thromboxane-B2 in platelets by acetylating cycloxygenase-1.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Trifluoperazine 2HCl,440-17-5,Trifluoperazine is a dopamine D2 receptor inhibitor with IC50 of 1.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Catharanthine,2468-21-5,Catharanthine inhibits nicotinic receptor mediated diaphragm contractions with IC50 of 59.6 ¦ÌM,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Meptazinol HCl,59263-76-2,Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fexofenadine HCl,153439-40-8,Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Moclobemide,71320-77-9,Moclobemide is MAO-A (5-HT) inhibitor with IC50 of 6.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Betulinic acid,472-15-1,Betulinic acid is a naturally occurring pentacyclic triterpenoid which has antiretroviral, antimalarial, and anti-inflammatory properties.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pergolide mesylate,66104-23-2,Pergolide mesylate is an antiparkinsonian agent which functions as a dopaminergic agonist.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cabozantinib malate ,1140909-48-3,Cabozantinib malate is the malate of Cabozantinib, a potent VEGFR2 inhibitor with IC50 of 0.035 nM and also inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, and AXL with IC50 of 1.3 nM, 4 nM, 4.6 nM, 12 nM/11.3 nM/6 nM, 14.3 nM and 7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sitagliptin phosphate monohydrate,654671-77-9,Sitagliptin phosphate (MK-0431) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ethambutol HCl,1070-11-7,Ethambutol is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosyl transferases.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Doxycycline HCl,10592-13-9,Doxycycline HCL is a tetracycline antibiotic that commonly used to treat a variety of infections and MMP inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Clinafloxacin (PD127391),105956-97-6,Clinafloxacin (PD127391) is a fluoroquinolone that inhibits both DNA gyrase and topoisomerase IV dually in Streptococcus pneumoniae.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pentamidine HCl,50357-45-4,Pentamidine is an inhibitor of <i>PRL Phosphatases</i> and also inhibits synthesis of DNA, RNA and protein.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Pemirolast (BMY 26517) potassium,100299-08-9,Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mirabegron (YM178),223673-61-8,Mirabegron is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Acebutolol HCl,34381-68-5,Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ampiroxicam,99464-64-9,Ampiroxicam is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Desloratadine,100643-71-8,Desloratadine is a potent antagonist for  human histamine H1 receptor with IC50 of 51 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium Monofluorophosphate  ,10163-15-2,Monofluorophosphate is a competitive inhibitor of pyruvate kinase and alkaline phosphatase with Ki of 3.4 mM and 69 μM, respectively, which also irreversibly inhibits phosphorylase phosphatase with Ki of 0.5 mM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hyoscyamine (Daturine),101-31-5,Hyoscyamine (Daturine) is an AChR inhibitor with IC50 of 7.5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ouabain,11018-89-6,Ouabain is a selective Na+, K+-ATPase inhibitor, binds to α2 subunit and α3 subunit with Ki of 41 nM and 15 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Allylthiourea,109-57-9,Allylthiourea is a metabolic inhibitor that selective inhibits ammonia oxidation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Avanafil,330784-47-9,Avanafil is a highly selective PDE5 inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tolcapone,134308-13-7,Tolcapone is a selective, potent and reversible of catechol-O-methyl transferase (COMT) inhibitor with Ki of 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Probenecid (Benemid),57-66-9,Probenecid (Benemid) is a classical competitive inhibitor of organic anion transport, which is also a TRPV2 agonist and an inhibitor of TAS2R16.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
 Procaine (Novocaine) HCl,51-05-8,Procaine (Novocaine) HCl is an inhibitor of sodium channel, NMDA receptor and nAChR with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with KD of 1.7 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Homatropine Methylbromide,80-49-9,Homatropine Methylbromide is muscarinic AChR antagonist, inhibits endothelial and smooth muscle muscarinic receptors of WKY-E and SHR-E with IC50 of 162.5 nM and 170.3 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Homatropine Bromide,51-56-9,Homatropine Bromide is muscarinic AChR antagonist, inhibits endothelial and smooth muscle muscarinic receptors of WKY-E and SHR-E with IC50 of 162.5 nM and 170.3 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hydroxyzine 2HCl,2192-20-3,Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Flavoxate HCl,3717-88-2,Flavoxate is a muscarinic AChR antagonist with IC50 of 12.2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dexamethasone Sodium Phosphate,2392-39-4,Dexamethasone is an interleukin receptor inhibitor and also suppresses COX-2. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Aclidinium Bromide,320345-99-1,Aclidinium Bromide inhibits human muscarinic AChR M1, M2, M3, M4 and M5 with Ki of 0.1 nM, 0.14 nM, 0.14 nM, 0.21 nM and 0.16 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Bismuth Subsalicylate,14882-18-9,Bismuth Subsalicylate is the active ingredient in Pepto-Bismol and inhibits prostaglandin G/H Synthase 1/2.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Diphemanil Methylsulfate,62-97-5,Diphemanil Methylsulfate is a quaternary ammonium anticholinergic, it binds muscarinic acetycholine receptors (mAchR).,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Vitamin D2 (Ergocalciferol),50-14-6,Vitamin D2 is a selective inhibitors of mammalian DNA polymerase A (pol A) with IC50 of 123 mM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Doxapram HCl,7081-53-0,Doxapram HCl inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 410 nM, 37 μM, 9 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Dibucaine (Cinchocaine) HCl,61-12-1,Dibucaine (Cinchocaine) HCl is a local anesthetics.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Methazolamide,554-57-4,Methazolamide is a carbonic anhydrase inhibitor with Ki of 50 nM, 14 nM and 36 nM for hCA I, hCA II and bCA IV isoforms, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tetrahydrozoline HCl,522-48-5,Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Valdecoxib,181695-72-7,Valdecoxib is a potent and selective inhibitor of COX-2 with IC50 of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Nabumetone,42924-53-8,Nabumetone is a non-steroidal anti-inflammatory drug and its active metabolite inhibits the COX.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sertraline HCl,79559-97-0,Sertraline HCl is a 5-HT antagonist with Ki of 13 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Spironolactone,52-01-7,Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Ropivacaine HCl,98717-15-8,Ropivacaine HCl is an anaesthetic agent and blocks impulse conduction in nerve fibres through inhibiting sodium ion influx reversibly.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Erythromycin Ethylsuccinate,1264-62-6,Erythromycin Ethylsuccinate, an oral macrolide antibiotic produced by <i>Streptomyces erythreus</i>, reversibly binds to the 50S ribosome of bacteria, and inhibits protein synthesis.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vitamin D3 (Cholecalciferol),67-97-0,Vitamin D3 (Cholecalciferol) is a form of vitamin D, binds and activates a H305F/H397Y mutant vitamin D receptor (VDR) with EC50 of 300 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Escitalopram Oxalate,219861-08-2,Escitalopram Oxalate is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Guanabenz (WY-8678) Acetate,23256-50-0,Guanabenz (WY-8678) Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Dequalinium Chloride,522-51-0,Dequalinium Chloride is a PKC inhibitor with IC50 of 7-18 μM, and also a selective blocker of apamin-sensitive K+ channels with IC50 of 1.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Hexamethonium Bromide,55-97-0,Hexamethonium Bromide is a selective antagonist of neuronal-type nicotinic AChR in ganglia.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Decamethonium Bromide,541-22-0,Decamethonium Bromide is a nicotinic AChR partial agonist and neuromuscular blocking agent.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium 4-Aminosalicylate,6018-19-5,Sodium 4-Aminosalicylate is an antibiotic used to treat tuberculosis via NF-?oB inhibition and free radical scavenging.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium Nitrite,7632-00-0,Sodium nitrite is a myeloperoxidase inhibitor with IC50 of 1.3 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zinc Pyrithione,13463-41-7,Zinc pyrithione is an antifungal and antibacterial agent disrupting membrane transport by blocking the proton pump.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Propranolol HCl,318-98-9,Propranolol HCl is a competitive non-selective beta-adrenergic receptors inhibitor with IC50 of 12 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Mefenamic Acid,61-68-7,Mefenamic acid is a competitive inhibitor of COX-1 and COX-2.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Ticagrelor,274693-27-5,Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist, also inhibits CYP2C9 and 4-hydroxylation with IC50 of 10.5 μM and 8.2 μM respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Triamterene,396-01-0,Triamterene blocks epithelial Na+ channel (ENaC) in a voltage-dependent manner with IC50 of 4.5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sulfacetamide Sodium,127-56-0,Sulfacetamide Sodium is an anti-biotic.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Lorcaserin HCl,846589-98-8,Lorcaserin HCl is a selective full agonist of human 5-HT2C receptor with Ki of 15 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Estradiol Benzoate,50-50-0,Estradiol benzoate is an estradiol analog which binds to the human, murine and chicken ERα with IC50 of 22-28 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Desvenlafaxine Succinate,386750-22-7,Desvenlafaxine Succinate is a new serotonin (5-HT) transporter and norepinephrine (NE) transporter reuptake inhibitor with Ki of 40.2 nM and 558.4 nM respectively.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Desvenlafaxine,93413-62-8,Desvenlafaxine is a serotonin (5-HT) and norepinephrine (NE) reuptake inhibitor with Ki of 40.2 nM and 558.4 nM, respectively. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Histamine 2HCl,56-92-8,Histamine is an organic nitrogen compound, acts on target cells in mammalian brain via stimulation of Histamine 1/2.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Pefloxacin Mesylate Dihydrate,149676-40-4,Pefloxacin Mesylate Dihydrate is the third generation of fluoroquinolone class of antibacterials, which inhibits Topoisomerase II activity and DNA replication.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
Timolol Maleate,26921-17-5,Timolol Maleate is a non-selective, beta-adrenergic receptor antagonist for β1/β2 with Ki of 1.97 nM/2.0 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Sodium Phenylbutyrate,1716-12-7,Sodium Phenylbutyrate is a transcriptional regulators that act by altering chromatin structure via the modulation of HDAC activity. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Terbutaline Sulfate,23031-32-5 ,Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Deoxyarbutin,53936-56-4,DeoxyArbutin is a reversible tyrosinase inhibitor, inhibiting tyrosinase activity with IC50 of 50 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tofacitinib citrate (CP-690550 citrate),540737-29-9,Tofacitinib citrate (CP-690550) is a potent JAK3 inhibitor with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Fingolimod (FTY720),162359-56-0,FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
LY2140023 (LY404039),635318-55-7,LY404039 is a potent agonist of recombinant human mGlu2, mGlu3 receptors and rat neurons expressing native mGlu2/3 receptors with Ki of 149 nM, 92 nM and 88 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PTC124 (Ataluren),775304-57-9,PTC124 (Ataluren) is a potent nonsense mutation inhibitor with EC50 of ~0.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VX-702,745833-23-2,VX-702 is a highly selective inhibitor of p38 MAPKα with IC50 of 4-20 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PP2,172889-27-9,PP2 is Src kinase inhibitor, potently inhibits GST-Src activity with IC50 of 100 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Stattic,19983-44-9,Stattic inhibits STAT3 with IC50 of 5.1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Embelin,550-24-3,Embelin, from the Japanese Ardisia herb, is a fairly potent, nonpeptidic, cell-permeable inhibitor of XIAP and efficiently overcomes the protective effect of XIAP XLALP to apoptosis.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"
IPI-145 (INK1197),1201438-56-3,IPI-145 (INK1197) is a novel and selective PI3K δ/γ inhibitor with Ki and IC50 of 23 pM/243 pM and 1 nM/50 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD2461,1174043-16-3,AZD2461 is a poor P-glycoprotein substrate with lower affinity for Pgp than does olaparib.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PD168393,194423-15-9,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Brefeldin A ,20350-15-6,Brefeldin A is a lactone antibiotic and ATPase inhibitor for protein transport with IC50 of 0.2 μM in HCT 116 cells.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Oprozomib (ONX 0912),935888-69-0,Oprozomib (ONX 0912) selectively inhibits CT-L activity of 20S proteasome β5/LMP7 with IC50 of 36 nM/82 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VX-661,1152311-62-0,VX-661 is a second F508del CFTR corrector and is believed to help CFTR protein reach the cell surface.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK J4 HCl,1373423-53-0(free base),GSK J4 HCl is a cell permeable prodrug of GSK J1, which is the first selective inhibitor of the H3K27 histone demethylase JMJD3/UTX with IC50 of 60 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
(+)-Bicuculline,485-49-4,(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NMDA (N-Methyl-D-aspartic acid),6384-92-5,NMDA（N-Methyl-D-aspartic acid）is a specific agonist for NMDA receptor mimicking the action of L-glutamate.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Cilengitide (EMD 121974, NSC 707544),188968-51-6,Cilengitide (EMD 121974, NSC 707544) is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
KY02111,1118807-13-8,KY02111 promotes differentiation of hPSCs to cardiomyocytes by inhibiting Wnt signaling.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
(−)-Blebbistatin,856925-71-8,(-)-Blebbistatin is a selective cell-permeable inhibitor of non-muscle myosin II ATPases with IC50 from 0.5-5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Zebularine,3690-10-6,Zebularine is an inhibitor of cytidine deaminase and also inhibit DNA methylation.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AMG-517,659730-32-2,AMG 517 is a potent and selective transient receptor potential vanilloid-1 (TRPV1)  antagonist with IC50 of <10 nM. ,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tenovin-1,380315-80-0,Tenovin-1 protects against MDM2-mediated p53 degradation, which invloves ubiquitination, and acts through inhibition of protein-deacetylating activities of SirT1 and SirT2.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Rocilinostat (ACY-1215),1316214-52-4,Rocilinostat (ACY-1215) is a selective HDAC6 inhibitor with IC50 of 5 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK2636771,1372540-25-4,GSK2636771 is a potent, orally bioavailable, PI3Kβ-selective inhibitor.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PQ 401,196868-63-0,PQ 401 is an IGF-1R inhibitor with IC50 of <1 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ZM 39923 HCl,1021868-92-7,ZM39923 is an JAK inhibitor for JAK1, JAK3, EFGR and TGM2 with IC50 of 4.4 μM, 7.1 μM, 5.6 μM and 10 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
SMI-4a,438190-29-5,SMI-4a is a potent inhibitor of Pim1 with IC50 of 17 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
BIX01294,1392399-03-9,BIX01294 is an inhitor of G9a histone methyltransferase with IC50 of 2.7 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VE-821,1232410-49-9,VE-821 is a potent and selective ATP competitive inhibitor of ATR with Ki and IC50 of 13 nM and 26 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AG 18 (Tyrphostin 23),118409-57-7,AG 18 inhibits EGFR with IC50 of 35 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PRX-08066,866206-55-5,PRX-08066 is a selective 5-HT2B antagonist with IC50 of 3.4 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Otenabant (CP-945598) HCl ,686347-12-6,CP-945598 HCl is a potent and selective cannabinoid type 1 receptor antagonist with Ki of 0.7 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW9508,885101-89-3,GW9508 is a potent and selective agonist for FFA1 (GPR40) with pEC50 of 7.32.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
CEP-32496,1188910-76-0,CEP-32496 is a RAF inhibitor for BRAF(V600E), BRAF(WT), c-Raf, Abl-1 and CSF-1R with IC50 of 14 nM, 36 nM, 39 nM, 3 nM and 9 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TAK-438,1260141-27-2,TAK-438 is a novel potassium-competitive acid blocker (P-CAB) type antisecretory agent that reversibly inhibits gastric H+, K+-ATPase with IC50 of 19 nM at pH 6.5.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
AZD5363,1143532-39-1,AZD5363 is a potent Akt inhibitor for Akt1, Akt2 and Akt3 with IC50 of 3 nM, 8 nM and 8 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW0742,317318-84-6,GW0742 is a potent and highly selective PPARβ/δ agonist, binding to hPPARδ with IC50 of 1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Vortioxetine (Lu AA21004) hydrobromide,960203-27-4,Lu-AA21004 is an oral multimodal serotonergic agent, inhibits 5-HT(1A), 5-HT(1B), 5-HT(3A), 5-HT(7) and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Empagliflozin (BI10773),864070-44-0,Empagliflozin (BI-10773) is a potent and selective SGLT2 inhibitor with IC50 of 3.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
TCS 359,301305-73-7,TCS 359 is a potent FLT3 inhibitor with IC50 of 42 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tyrphostin AG 1296 (AG 1296),146535-11-7,Tyrphostin AG 1296 (AG 1296) is an inhibitor of PDGFR, FGFR and c-Kit with IC50 of < 1 μM, 12.3 μM and 1.8 μM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GSK3787,188591-46-0,GSK3787 is as a potent and selective antagonist of PPARδ with pIC50 of 6.6.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Tariquidar,206873-63-4,Tariquidar (XR9576) is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
WY 14643 (Pirinixic Acid),50892-23-4,WY 14643 (Pirinixic Acid) is a potent peroxisome proliferator and activator of PPARα with ED50 of 1.5 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Plerixafor (AMD3100),110078-46-1,Plerixafor is a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
NSC 23766,1177865-17-6,NSC 23766 is an inhibitor of Rac GTPase targeting Rac activation by guanine nucleotide exchange factors (GEFs) with IC50 of about 50 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
PRT062607 (P505-15, PRT2607, BIIB057) HCl,1370261-97-4,1370261-96-3(free base),,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Apremilast (CC-10004),608141-41-9,Apremilast (CC-10004) is a potent PDE4 and TNF-α inhibitor with IC50 of 74 nM and 77 nM, respectively.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
VU 0364439,1246086-78-1,,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Butein,487-52-5,Butein, a plant polyphenol isolated from <i>Rhus verniciflua</i>, inhibits EGFR tyrosine phosphorylation with IC50 of 8 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Necrostatin-1,4311-88-0,Necrostatin-1 is a specific RIP1 inhibitor and inhibits TNF-α-induced necroptosis with EC50 of 490 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
UPF 1069,1048371-03-4,UPF 1069 is a selective PARP2 inhibitor with IC50 of 0.3 μM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GDC-0349,1207360-89-1,GDC-0349, is a potent and selective ATP-competitive inhibitor of mTOR with Ki of 3.8 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
GW2580,870483-87-7,GW2580 is a selective inhibitor of human c-FMS with IC50 of 30 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
Scriptaid ,287383-59-9,Scriptaid is an inhibitor of histone deacetylase.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
ABT-199 (GDC-0199 ),1257044-40-8,ABT-199 is a Bcl-2-selective inhibitor with Ki of < 0.010 nM.,HPLC 99%, NMR, LCMS is OK, stock more than 20g
"Macitentan,441798-33-0,Macitentana (Actelion-1, ACT-064992) is an orally active, non-peptide dual endothelin (ET)A/B receptor antagonist with IC50 of 0.5 nM/391 nM.
,HPLC 99%, NMR, LCMS is OK, stock more than 20g"