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2017年11月18日星期六

Eos Med Chem, Product List--Small molecule inhibitors of Clinical---40029

Small molecule inhibitors of Clinical---40029

一种潜在治疗炎症性疼痛的大麻素受体2(CB2)拮抗剂。

AB-001;CAS号1345973-49-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一个潜在治疗慢性腰背痛的大麻素1和2受体激动剂。

Abacavir acetate;KM-133; CAS号1446418-48-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗斑块状银屑病的药物。

ABC-294640;CAS号915385-81-8(ABC 294640), 1185157-59-8(ABC 294640), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体瘤和B细胞淋巴瘤的鞘氨醇激酶2抑制剂。

Abediterol;AZD-0548; LAS-100977, CAS号915133-65-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗哮喘和慢性阻塞性肺疾病的长效β肾上腺素受体激动剂。

Abexinostat;CG-781; CRA-024781; PCI-24781; S-78454
CAS号783355-60-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗霍奇金淋巴瘤和非霍奇金淋巴瘤(NHL)的组蛋白去乙酰化酶(HDAC)抑制剂。

Glecaprevir;ABT-493, CAS号1365970-03-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙型肝炎的蛋白酶抑制剂。

ABT-494;CAS号1310726-60-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗风湿性关节炎的蛋白酪氨酸激酶(Jak1)抑制剂。

Pibrentasvir;ABT-530;CAS号1353900-92-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙型肝炎的蛋白酶抑制剂。

ABT-751; E-7010, CAS号141430-65-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌,肾细胞癌及非小细胞肺癌的微管蛋白聚合抑制剂。

ABX-464; SPL-464 CAS号1258453-75-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗HIV感染的病毒RNA复制抑制剂。

ATN-161;CAS号262438-43-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗恶性胶质瘤和肾细胞癌的整合素αVβ3(玻璃粘连蛋白)拮抗剂。

Acebilustat; CTX-4430; EP-501, CAS号943764-99-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗囊性纤维化的白三烯A4水解酶抑制剂。

EM-652; SCH-57068; EM-01538
CAS号182167-02-8(Acolbifene), 252555-01-4(Acolbifene Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的预防绝经前妇女高风险乳腺癌的选择性雌激素受体调节剂(SERM)。

Acumapimod;BCT-197, CAS号836683-15-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性阻塞性肺疾病(COPD)的p38丝裂原活化蛋白激酶(MAPK)抑制剂。

Aderbasib;INCB-7839; INCB-007839, CAS号791828-58-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗非霍奇金淋巴瘤、实体瘤的表皮生长因子受体抑制剂。

ADX-71149; JNJ-40411813, CAS号1127498-03-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗焦虑症与精神分裂症的代谢型谷氨酸受体2(mGluR2)阳性变构调节剂(PAM)。

NS-986; SMP-986
CAS号 877606-63-8(Afacifenacin) 877614-61-4(Afacifenacin Fumarate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗夜尿症的毒蕈碱受体拮抗剂。

Afimoxifene;4-OHT; 4OHT CAS号68392-35-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳房胀痛及其它良性乳腺疾病的雌性激素受体抑制剂。

AFN-1252; AFN-12520000; API-1252; Debio-1452
CAS号620175-39-5 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.

Afuresertib;GSK-2110183 CAS号1047644-62-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗卵巢癌,慢性淋巴细胞白血病和多发性骨髓瘤的蛋白激酶抑制剂。

AL-8176; ALS-008176; ALS-8176 CAS号1445385-02-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗呼吸道合胞体病毒感染的RNA聚合酶抑制剂。

Aladorian; ARM-036; S-36; S-44121; S-44121-1; S-441211 CAS号865433-00-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗心律失常的作用于ryanodine受体(RyR)的药物。

Albaconazole;UR-9825; W-0027, CAS号187949-02-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗真菌感染的三唑类抗真菌剂。

Alisertib;MLN-8237, CAS号1028486-01-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗小细胞肺癌的激光A型激酶抑制剂。

Alpelisib;BYL-719; NVP-BYL-719; NVPBYL-719
CAS号1217486-61-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗头颈部鳞状细胞癌,乳腺癌,非小细胞肺癌和实体肿瘤的磷脂酰肌醇-3-羟激酶抑制剂。

HL-275; HMR-1275; L-86-8275; MDL-107826A; NSC-649890; L-868275
CAS号 146426-40-6(Alvocidib), 131740-09-5(Alvocidib Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体肿瘤和淋巴瘤的细胞周期蛋白依赖性激酶抑制剂。

AMD-070; AMD-11070, CAS号558447-26-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗HIV感染的趋化因子受体4拮抗剂。

AMG-131; INT-131; T-0903131; T-131
CAS号315224-26-1(AMG-131 Free), 849738-78-9(AMG-131), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一个潜在治疗二型糖尿病和多发性硬化症的过氧化物酶体增殖物活化受体PPARγ激活剂。

AMG-232;CAS号1352066-68-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗黑色素瘤的MDM2抑制剂。

AMG-337;CAS号1173699-31-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗食道腺癌,胃食管交界腺癌和胃癌的肝细胞生长因子受体抑制剂。

Aminopterin;NSC-739; AMT, CAS号54-62-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗风湿性关节炎的二氢叶酸还原酶抑制剂。

Amiselimod;MT-1303
CAS号 942399-20-4(Amiselimod) ,942398-84-7(Amiselimod hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗复发缓解型多发性硬化、克罗恩氏病和斑块型银屑病的溶血磷脂质edg1(S1P1)配体。

AN-0128; CRM-0005; ONT-0001, CAS号872044-70-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗特应性皮炎的肿瘤坏死因子-α(TNF-α)抑制剂。

AN-2898;CAS号906673-33-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.

Ansofaxine Hydrochloride  (盐酸安舒法辛);LY-03005
CAS号916918-80-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗抑郁症的5-羟色胺-多巴胺-去甲肾上腺素再摄取抑制剂。

AP-1531; BGC-20-1531; BGC-201531
CAS号1186532-61-5(AP-1531), 736183-35-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.

APD-334;CAS号1206123-37-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗自身免疫疾病的1-磷酸鞘氨醇受体激动剂。

API-001; E-52862; S-1RA
CAS号878141-96-9, 1265917-14-3(API-001), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗多发性神经痛的Sigma1(σ1)受体拮抗剂。

Apitolisib;G-038390; GDC-0980; RG-7422; R-7422
CAS号1032754-93-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌,前列腺癌和非霍奇金淋巴瘤的磷脂酰肌醇3-激酶(PI3K)抑制剂。

APR-246; PRIMA-1MET CAS号5291-32-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗急性骨髓性白血病、卵巢癌与前列腺癌的p53基因激动剂。

AQ-13;CAS号32571-49-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗疟疾的氨基喹啉类抗生素。

AQW-051;CAS号669770-29-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗精神分裂症的α-7烟碱型受体激动剂。

(S)-HDAC-42; AR-42; NSC-736012; OSU-42; OSU-HDAC-42; OSUHDAC-42
CAS号935881-37-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体瘤、白血病和淋巴瘤的组蛋白去乙酰化酶(HDAC)抑制剂。

ASLAN-002; BMS-777607
CAS号1025720-94-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胃癌和乳腺癌的RON/MET/Flt3多靶点抑制剂。

ASM-024;CAS号1609534-88-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗哮喘与慢性阻塞性肺病(COPD)的烟碱受体激动剂。

AT-101;(R-(-)-醋酸棉酚)
CAS号90141-22-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非霍奇金淋巴瘤,前列腺癌和非小细胞肺癌的B细胞淋巴瘤蛋白-2抑制剂。

AT-406; Debio-1143; SM-406
CAS号,1071992-99-8(AT 406) 1071992-57-8(AT 406), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗头颈癌和实体瘤的凋亡抑制蛋白抑制剂。

AT-7519; AT-7519M
CAS号844442-38-2(AT 7519) 902135-91-5(AT 7519), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗慢性淋巴细胞白血病、套细胞淋巴瘤与多发性骨髓瘤的细胞周期蛋白依赖性激酶抑制剂。

AT-9283;CAS号896466-04-9(AT 9283), 896466-61-8(AT-9283), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的用于治疗多发性骨髓瘤的多靶向激酶抑制剂。

Ataciguat;HMR-1766 CAS号254877-67-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗主动脉瓣狭窄的鸟苷酸环化酶激活剂。

ATB-346;CAS号1226895-20-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗骨关节炎、类风湿性关节炎、强直性脊柱炎的环氧化酶(COX)抑制剂。

Atreleuton;VIA-2291; ABT-761; A-85761; Abbott-85761 CAS号154355-76-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗急性冠脉综合征的5-脂氧合酶抑制剂。

AUS-131; (S)-Equol; (S)Equol CAS号531-95-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗良性前列腺增生(BPH)与潮热(HF)的雌激素β受体(ER-β)激动剂。

AE-37; AVex-73; Anavex-2-73; Anavex-273 CAS号195615-83-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗阿尔茨海默病的毒蕈碱M1受体激动剂。

AZD-1775; AZ-1775; MK-1775 CAS号955365-80-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗卵巢癌的WEE1激酶抑制剂。

AZD-1981;CAS号802904-66-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗慢性特发性荨麻疹(CIU)的CRTH2抑制剂。

AZD-2624;CAS号941690-55-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的用于治疗精神分裂症的速激肽NK3受体拮抗剂。

AZD-3241 CAS号890655-80-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗系统性萎缩症的髓过氧物酶抑制剂。

AZD-3759;CAS号1626387-80-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌的表皮生长因子受体抑制剂。

AZD-4547;CAS号1394854-62-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体肿瘤的纤维母细胞生长因子受体抑制剂。

AZD-5069;CAS号878385-84-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗头颈癌的趋化因子CXCR2受体配体。

AZD-5363,CAS号1143532-39-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌的AKT激酶抑制剂。

AZD-6738;CAS号1352226-97-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体肿瘤的ATR丝氨酸/苏氨酸激酶抑制剂。

AZD-7325; AZ-7325 CAS号942437-37-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗自闭症谱系障碍(ASD)的GABA受体激动剂。

AZD-8529;CAS号877145-53-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗烟瘾的代谢型谷氨酸受体第二亚型(mGluR2)阳性变构调节剂。

Bafetinib;CNS-9; INNO-406; NS-187
CAS号 859212-16-1(Bafetinib), 859212-17-2(Bafetinib Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性淋巴细胞白血病的Bcr-Abl/Fyn/Lyn激酶抑制剂。

BAL-101553;CAS号1263384-43-5(BAL 101553) 1387574-54-0(BAL 101553), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗晚期实体瘤的微管减稳剂。

Barasertib;AZD-1152 CAS号722543-31-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗难治性弥漫大 B 细胞淋巴瘤的极光激酶抑制剂。

Bardoxolone Methyl;RTA-402; NSC-713200; TP-155C; Methyl-CDDO; MethylCDDO
CAS号218600-53-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性肾脏疾病及肺动脉高血压的NF-kB抑制剂。

Basimglurant Sulfate;RG-7090; RO-4917523
CAS号 802906-73-6(Basimglurant) 1034442-21-1(RG-7090), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗重度抑郁症的代谢性谷氨酸受体第5亚型拮抗剂。

Basmisanil;RG-1662; RO-5186582 CAS号1159600-41-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗唐氏综合症的α5亚型-γ-氨基丁酸受体拮抗剂。

Batefenterol Succinate;GSK-961081; GSK-961081D; TD-5959; 961081
CAS号 743461-65-6(Batefenterol) 945905-37-3(Batefenterol succinate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性阻塞性肺病的β2-肾上腺素受体激动剂和毒蕈碱受体拮抗剂。

BAY-85-8501;CAS号1161921-82-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗支气管扩张的白细胞弹性蛋白酶抑制剂。

F-13640; NLX-112
CAS号208110-64-9(Befiradol) 208110-65-0(Befiradol Fumarate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗帕金森病患者中因药物引起运动障碍的5-羟色胺受体激动剂。

ESP-55016; ETC-1002;CAS号738606-46-7(Bempedoic acid), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗高胆固醇血症与高血压的腺苷酸活化蛋白激酶激动剂与ATP-柠檬酸裂解酶抑制剂。

PGL-5001; AS-602801 CAS号848344-36-5(Bentamapimod), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗女性子宫内膜异位的JNK1激酶抑制剂。

Besifovir;ANA-380; LB-80380; PMCDG dipivoxil CAS号441785-26-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乙肝感染的逆转录酶抑制剂。

BGP-15;CAS号66611-37-8(BGP 15) 66611-38-9(NP 51), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗Ⅱ型糖尿病及杜氏肌萎缩症的胰岛素增敏剂。

BGT-226; NVP-BGT-226; NVPBGT-226 CAS号915020-55-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗晚期实体瘤的磷脂酰肌醇3-激酶抑制剂。

BI-2536;CAS号755038-02-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌、非霍奇金淋巴瘤及急性髓系白血病的plk-1抑制剂。

BIIB-021; CNF-2024; CF-1983 mesylate
CAS号 848695-25-0(BIIB 021) 1225041-97-3(BIIB-021), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胃肠道间质肿瘤和实体瘤的热休克蛋白90抑制剂。

Birinapant;NSC-756502; TL-32711 CAS号1260251-31-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.一种潜在的治疗骨髓增生异常综合征,卵巢癌和慢性乙肝的凋亡抑制蛋白抑制剂。

BIT-225;CAS号917909-71-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙型肝炎和艾滋病的核衣壳p7蛋白 (NCp7)锌指结构抑制剂。

Bitopertin;R-1678; RG-1678; RO-4917838 CAS号845614-11-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗强迫症的甘氨酸转运体1型抑制剂。

BMS-754807;CAS号1001350-96-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗乳腺癌的胰岛素样生长因子1受体拮抗剂。

BMS-833923; XL-139 CAS号1059734-66-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗基底细胞母斑综合征的SMO受体拮抗剂。

BMS-911543;CAS号1271022-90-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗骨髓纤维化的酪氨酸蛋白激酶2(JAK2)抑制剂。

BMS-919373;CAS号1272353-82-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗阵发性心房颤动的钾离子通道阻滞剂。

BMS-986020; AM-152; BMS-986202 CAS号1257213-50-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗特发性肺纤维化的溶血磷脂酸1型受体拮抗剂。

BN-82451; BN-82451B CAS号335242-75-6, 663172-95-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗亨廷顿氏舞蹈症的环氧化酶抑制剂。

BNC-105; BNC-105P CAS号945772-45-2(BNC-105), 945771-96-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗肾细胞癌、胸膜间皮瘤与卵巢癌的微管蛋白聚合抑制剂。

BQ-788;CAS号 156161-89-6(BQ-788), 173326-37-9(BQ-788 Free), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗高血压的内皮素受体拮抗剂。

Brigatinib;AP-26113
CAS号1197953-54-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗ALK阳性非小细胞肺癌的ALK与EGFR抑制剂。

PNU-166196; PNU-166196A
CAS号 203258-60-0(Brostallicin), 203258-38-2(Brostallicin Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌、软组织肉瘤、脂肪肉瘤的DNA小沟结合剂。

Cabotegravir;GSK-1265744; GSK-1265744A; GSK-744; S-265744; S-265744 LAP; S
CAS号1051375-10-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗艾滋病感染的整合酶抑制剂。

GSK-962040; CAS号 923565-21-3(Camicinal) 923565-22-4(Camicinal Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗糖尿病性胃轻瘫的胃动素受体激动剂。

CI-1033;CAS号 289499-45-2(Canertinib dihydrochloride) 267243-28-7(Canertinib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.一种潜在的治疗非小细胞肺癌及乳腺癌的表皮生长因子受体抑制剂。

Capmatinib;INC-280; INCB-028060; INCB-28060 CAS号1029712-80-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌,恶性胶质细胞瘤,黑色素瘤,肝癌和乳头状肾上皮细胞癌的肝细胞生长因子受体抑制剂。

JNJ-10234094; RWJ-333369; YKP-509 CAS号194085-75-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.

CHF-4226; TA-2005CAS号147568-66-9(Carmoterol), 137888-11-0(Carmoterol Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性阻塞性肺疾病(COPD)和哮喘的肾上腺素β2受体激动剂。

CC-220;CAS号1323403-33-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗全身性红斑狼疮的药物。

CCX-168;CAS号1346623-17-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗抗中性粒细胞胞质抗体(ANCA)相关血管炎的C5过敏毒素趋化因子受体拮抗剂。

Cebranopadol hemicitrate;GRT-6005
CAS号863513-92-2(Cebranopadol Hemicitrate),863513-91-1(Cebranopadol), HPLC 99%, NMR, LCMS is ok, stock more than 20g.

CEP-9722;CAS号916574-83-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体瘤,非小细胞肺癌和卵巢癌的聚腺苷二磷酸核糖聚合酶抑制剂。

Cerdulatinib;PRT-062070; PRT-2070
CAS号1198300-79-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性淋巴细胞白血病(CLL)和非霍奇金B细胞淋巴瘤(NHL)的脾酪氨酸激酶(Syk)和janus激酶(JAK)双重抑制剂。

CFG-920;CAS号1260006-20-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗去势抵抗性前列腺癌的17α羟化酶抑制剂。

CG-200745; HDCG-0745 CAS号936221-33-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体肿瘤的组蛋白去乙酰化酶抑制剂。

CG-400549; CG-0549 CAS号934628-27-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗急性细菌性皮肤和皮肤结构感染的酰基载体蛋白还原酶抑制剂。

CHF-5074; CSP-1103 CAS号749269-83-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗轻度认知功能损害(MCI)的γ-分泌酶调节剂。

CHF-6001;CAS号1239278-59-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗哮喘与慢性阻塞性肺病(COPD)的磷酸二酯酶4型抑制剂。

Cimicoxib;UR-8880 CAS号265114-23-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗重度抑郁症的环氧化酶抑制剂。

Cinepazide mesylate CAS号88197-48-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗脑血管疾病的药物。

CNS-5161;CAS号160754-76-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗糖尿病性神经病变的N-甲基-D-天冬氨酸受体拮抗剂。

COTI-2;CAS号1039455-84-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗卵巢癌与头颈部鳞状细胞癌的P53基因调节剂与AKT2抑制剂。

CPI-613; BBOA, CAS号95809-78-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗小细胞肺癌(SCLC)、骨髓增生异常综合征(MDS)与胰腺癌的AEMD药物。

CR-4056;CAS号1004997-71-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.

ARO-002-26; CP-868596-26; CP-86859626; ARO-00226. CAS号670220-88-9(Crenolanib), 670220-93-6(Crenolanib Besylate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗急性髓系白血病和胃肠道间质肿瘤的血小板衍生生长因子受体(PDGFR)抑制剂。

Cutamesine Hydrochloride;AGY-94806; SA-4503; Msc-1
CAS号165377-43-5(Cutamesine),165377-44-6(SA 4503), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗重度抑郁症及中风的乙酰胆碱释放增强剂及西格玛受体激动剂。

BEZ-235; NVP-BEZ-235; NVPBEZ-235
CAS号915019-65-7(Dactolisib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌、肾细胞癌、膀胱癌和前列腺癌的磷脂酰肌醇-3-羟激酶抑制剂。

GSK-1325756; GSK-1325756B; 1325756
CAS号954126-98-8(Danirixin), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性阻塞性肺病的CXC2趋化因子受体拮抗剂。

PHA-739358;CAS号827318-97-8(Danusertib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.一种潜在的治疗实体瘤和慢性粒细胞白血病的多靶点激酶抑制剂。

APO-866; FK-866; K-22.175
CAS号658084-64-1(Daporinad), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗B细胞慢性淋巴细胞白血病,皮肤T细胞淋巴瘤和黑色素瘤的烟酰胺磷酸核糖基转移酶(NMPRTase)抑制剂。


GSK-1278863; GSK-1278863A; 1278863
CAS号960539-70-2(Daprodustat), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性肾病引起贫血症的低氧诱导因子脯氨酰基羟化酶抑制剂。

DB-959Na; T-3D-959; T-3D959
CAS号1257641-15-8(DB-959) 1258076-66-2(DB-959Na), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗阿尔兹海默症的过氧化物酶体增殖物活化受体激动剂。

PF-04554878; PF-4554878; VS-6063;CAS号1073154-85-4(Defactinib),1073160-26-5(Defactinib Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌和胸膜间皮瘤的局部粘着斑激酶抑制剂。

BIIB-050; KNS-760704; SND-919CL-2X; SND-919CL2X;CAS号
908244-04-2(Dexpramipexole Dihydrochloride Monohydrate)
104632-28-2(Dexpramipexole), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗阿尔茨海默病(AD)、嗜酸性粒细胞增多症(HES)和嗜酸细胞性慢性鼻窦炎的多巴胺受体激动剂。

DG-041;CAS号861238-35-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗外周动脉硬化的前列腺素EP3受体拮抗剂。

DG-051;CAS号929916-05-2(DG-051),929915-58-2(DG 051), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的预防心肌梗塞的白三烯A4水解酶(LTA4H)抑制剂。

BIBR-796; BIRB-0796; BIRB-796 BS. CAS号285983-48-4(Doramapimod), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗类风湿性关节炎、牛皮癣和克罗恩病的p38MAP激酶和肿瘤坏死因子-α抑制剂。

E-3710; Z-215;CAS号955095-45-1, 955095-47-3(E-3710), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胃食管反流病的质子泵抑制剂。

E-6005;CAS号947620-48-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗过敏性皮炎的磷酸二酯酶-4抑制剂。

E-7449;CAS号1140964-99-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体瘤和B细胞恶性肿瘤的聚腺苷二磷酸核糖聚合酶抑制剂。

E-7820; NSC-719239; ER-68203-00; ER-6820300
CAS号289483-69-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗结直肠癌的α2-整合素受体抑制剂。

Efatutazone hydrochloride; CS-7017; RS-5444
CAS号223132-37-4(Efatutazone), 1048002-36-3(Efatutazone hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗甲状腺癌与脂肉瘤的过氧化物酶体增殖物活化受体-γ(PPARγ)激动剂。

STA-4783;CAS号488832-69-5(Elesclomol), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗女性生殖系统癌症的热休克蛋白70诱导剂。

DU-28853;CAS号98224-03-4(Eltoprazine), 98206-09-8(Eltoprazine Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗治疗注意力不足过动症(ADHD),运动障碍与认知障碍的5-羟色胺拮抗剂。

Endoxifen;CAS号112093-28-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌的雌激素受体拮抗剂。

5-EU; 776C-85; ADH-300004; GW-776; 5EU CAS号59989-18-3(Eniluracil), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗转移性乳腺癌和其它实体肿瘤的二氢嘧啶脱氢酶抑制剂。

ENMD-2076; ENMD-981693
CAS号934353-76-1(ENMD-2076 Free) 1453868-32-0(ENMD-2076), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌,卵巢癌,软组织肉瘤的VEGFR抑制剂和Aurora激酶抑制剂。

GS-9973;CAS号
1648797-46-9(Entospletinib Dimesylate), 1229208-44-9(Entospletinib, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的用于治疗慢性淋巴细胞白血病和急性髓系白血病的脾络氨酸激酶抑制剂。

Entrectinib;NMS-E-628; RXDX-101  ; NMSE-628;
CAS号1108743-60-7(Entrectinib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌和结肠癌的多重激酶抑制剂。

INCB-024360; INCB-24360
CAS号1204669-58-8(Epacadostat), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗女性生殖系统癌症,黑色素瘤和脊髓发育不良的吲哚胺2,3-双加氧酶抑制剂。

JNJ-42756493;CAS号1346242-81-6(Erdafitinib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗膀胱癌和肝癌的纤维母细胞生长因子受体抑制剂。

ESN-364;CAS号1629229-37-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗子宫肌瘤和多囊卵巢综合征的速激肽NK3拮抗剂。

AGI-001; MT-102 CAS号26328-11-0((S)-(-)-Pindolol), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗癌症相关恶病质的β-肾上腺素受体拮抗剂。

EHT-0202; EHT-202 CAS号51022-77-6(Etazolate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种用于治疗与阿尔茨海默病相关的认知功能障碍的磷酸二酯酶4/γ-氨基丁酸受体双靶点抑制剂。

Ezatiostat); TER-199; TLK-199,CAS号 168682-53-9(Ezatiostat) 286942-97-0(Ezatiostat Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗骨髓增生异常综合征与严重慢性中性粒细胞减少症的谷胱甘肽S-转移酶P1抑制剂。

BMN-195; SMTC-1100; VOXC-1100 CAS号945531-77-1(Ezutromid), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗杜式肌营养不良症的utrophin蛋白活化剂。

FE-106483; VA-106483; VT-483 CAS号347887-36-9(Fedovapagon), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗夜尿症的血管加压素受体激动剂。

QAW-039;CAS号 872365-14-5(Fevipiprant), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗哮喘,过敏性皮炎和过敏性鼻炎的前列腺素D2受体拮抗剂。

FG-2216; YM-311 CAS号223387-75-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗贫血症的低氧诱导因子脯氨酰羟化酶抑制剂。

AM-803; GSK-2190915; 2190915
CAS号936350-00-4(Fiboflapon), 1196070-26-4(Fiboflapon Sodium), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗哮喘的5-脂氧合酶抑制剂。

G-146034; GLPG-0634 CAS号1206161-97-8(Filgotinib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗风湿性关节炎和克罗恩病的蛋白酪氨酸激酶抑制剂。

JP-1730;CAS号150586-72-4(MPV 1730 Hydrochloride), 150586-58-6(Fipamezole), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗帕金森病运动障碍的α2-肾上腺素受体拮抗剂。

HM-101;CAS号 341524-89-8(Fispemifene), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗性腺机能减退的选择性雌激素受体调节剂。

ATx-08-001; FK-614; ATx-08001
CAS号193012-35-0(FK-614) NPS-005; SJP-0035, HPLC 99%, NMR, LCMS is ok, stock more than 20g.

CAS号515138-06-4(Fonadelpar), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗角膜疾病的过氧化物酶体增殖物活化受体激动剂。

EXEL-2880; XL-880; GSK-1363089; GSK-089; 1363089
CAS号849217-64-7(Foretinib), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌和非小细胞肺癌的VEGFR-2激酶和c-Met激酶的抑制剂。

PF-04171327; PF-4171327
CAS号1044535-58-1(Fosdagrocorat), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗类风湿性关节炎的糖皮质激素受体 (GR) 调制器。

Gandotinib; LY-2784544
CAS号1229236-86-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗骨髓及外骨髓增殖(MPD)的Janus激酶2(JAK2)抑制剂。

GDC-0810; ARN-810; RG-6046
CAS号1365888-06-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗晚期或转移性乳腺癌的选择性雌激素受体失稳剂。

GZ-452; Genz-682452;CAS号 1401090-53-6, 1629063-78-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗法布瑞氏病的葡糖神经酰胺合成酶抑制剂。

GSK-2140944; 2140944
CAS号1075236-89-3(Gepotidacin), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗细菌性皮肤和皮肤结构感染和淋病的DNA拓扑异构酶II抑制剂。

GET-73;CAS号202402-20-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗酒精依赖的代谢性谷氨酸受体-5别构调节剂。

ITF-2357;CAS号 497833-27-9(Givinostat) 199657-29-9(Givinostat Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗幼年特发性关节炎、骨髓增生性疾病、慢性淋巴细胞白血病和真性红细胞增多的组蛋白去乙酰化酶(HDAC)抑制剂。

GKT-137831;CAS号1218942-37-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗糖尿病性肾病的NOX抑制剂。

PF-04449913;CAS号1095173-27-5(Glasdegib)
一种潜在的治疗骨髓增生异常综合征,慢性粒细胞白血病和急性骨髓性白血病的SMO拮抗剂。

GLPG-0974;CAS号1391076-61-1
一种潜在治疗溃疡性结肠炎的游离脂肪酸受体2(FFAR2)拮抗剂。

ER-396901-08; E-7050; Golvatinib; ER-39690108
CAS号928037-13-2(Golvatinib) 1007601-96-8(Golvatinib tartrate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗头颈癌、肝癌(HCC)与实体瘤的c-Met和VEGFR-2抑制剂。

PF-00734200; PF-734200;CAS号869490-23-3(Gosogliptin), 869490-47-1(Gosogliptin Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗2型糖尿病的二肽基肽酶-4(DPP-4)抑制剂。

AAT-007; CJ-023423; CJ-23423; MR-10A-7; RQ-00000007; RQ-7; MR-10A7 CAS号415903-37-6(Grapiprant), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性疼痛和骨关节炎的前列腺素EP4受体拮抗剂。

GS-9620;CAS号1228585-88-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乙肝的Toll样受体7抑制剂。

GSK-163090; 163090;CAS号
844903-58-8(GSK-163090 Free), 844903-52-2(GSK-163090), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗重度抑郁症的5-羟色胺拮抗剂。

GSK-2269557; 2269557 CAS号1254036-71-9 1254036-77-5(GSK-2269557), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗慢性阻塞性肺疾病(COPD)和哮喘的磷脂酰肌醇-3-羟激酶δ抑制剂。

GSK-2330672; 2330672 CAS号1345982-69-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗2型糖尿病的回肠胆汁酸转运体抑制剂。

GSK-239512;CAS号720691-69-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗复发-缓解型多发性硬化症(RRMS)的组胺H3受体拮抗剂。

GSK-2636771;CAS号1372540-25-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体肿瘤的磷脂酰肌醇-3-羟激酶抑制剂。

GSK-2894512; CAS号 79338-84-4(WBI-1001), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗过敏性皮炎和牛皮癣的非甾体类抗炎药物。

GSK-525762; GSK-525762A; I-BET-762; IBET-762 CAS号1260907-17-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗恶性肿瘤的溴结构域蛋白抑制剂。

GSK-598809;CAS号 863680-46-0(GSK-598809) 863766-31-8(GSK-598809), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的控制烟瘾的多巴胺D3受体拮抗剂。

GSK-805; GSK-2336805; JNJ-56914845 CAS号1256390-53-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙型肝炎的丙肝病毒NS5A抑制剂。

GTx-011; GBT-440 CAS号1446321-46-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗镰刀状贫血病的镰状血红蛋白调节器。

GW-501516; GW-516; GSK-516CAS号317318-70-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.一种潜在的治疗血脂异常的过氧化物酶体增殖物活化受体-δ激动剂。

GW-876167; BVT-933; PNU-183933; PRX-00933 CAS号313658-33-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗肥胖的5-羟色胺2C激动剂。

HT-0712; IPL-455903 CAS号617720-02-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗年龄相关性记忆障碍(AAMI)的磷酸二酯酶4型抑制剂。

F-351; Hydronidone CAS号851518-71-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.一种潜在治疗肝纤维化的非甾体类抗炎药(NSAIDs)。

Icaritin  (阿克拉定);SNG-162; SGIC-162CAS号118525-40-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗肝癌的MAPK与ERK抑制剂。
Ifetroban;BMS-180291 CAS号143443-90-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗肝肾综合征(HRS)与呼吸障碍的前列腺素TP受体拮抗剂。
Ilorasertib;ABT-348 CAS号1227939-82-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗实体瘤的极光激酶/血管内皮生长因子受体激酶双靶点抑制剂。

Imeglimin;EMD-387008 CAS号775351-65-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗Ⅱ型糖尿病的腺苷酸活化蛋白激酶激活剂。

Imexon;AOP-990001; BM-06002 CAS号59643-91-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胰腺癌,肺癌及黑色素瘤的核苷二磷酸还原酶抑制剂。

Imidol Hydrochloride  (盐酸艾咪朵尔)
CAS号 172041-16-6(Imidol) 1606174-14-4(Imidol Hydrochloride), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗HBV感染的药物。

Implitapide;AEGR-427; BAY-13-9952; BAY-139952 CAS号177469-96-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗高胆固醇症的微粒体甘油三酯转运蛋白(MTTP)抑制剂。

INCB-39110; INCB-039110 CAS号1334298-90-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗非小细胞肺癌和胰腺癌的Jak1抑制剂。

Indisulam;E-7070; ER-35744 CAS号165668-45-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗急性髓性白血病及高危骨髓增生异常综合征的碳酸酐酶抑制剂。

Indoximod;NSC-721782; D-1MT; NLG-8189 CAS号110117-83-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗乳腺癌、前列腺癌、恶性脑瘤、胰腺癌与黑色素瘤的吲哚胺2,3-二加氧酶(IDO)抑制剂。

Infigratinib;BGJ-398; NVP-BGJ-398; NVPBGJ-398 CAS号872511-34-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胆管癌,恶性胶质瘤,白血病,黑色素瘤和实体肿瘤的磷脂酰肌醇-3-羟激酶抑制剂。

Ipatasertib Dihydrochloride;GDC-0068; RG-7440
CAS号1001264-89-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗胃癌,三阴性乳腺癌和前列腺癌的Akt激酶抑制剂。

Irosustat;BN-83495; STX-64; 667-Coumate; 667Coumate, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌的碳酸酐酶/酰硫酸酯酶抑制剂。

CAS号288628-05-7 Iroxanadine;BRX-005; BRX-235 CAS号276690-58-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗动脉粥样硬化的丝裂原活化蛋白激酶P38抑制剂。

Isatoribine  (沙托立宾) ANA-245; ICN-10146; NARI-10146 CAS号122970-40-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙型肝炎的Toll样受体-7激动剂。

Ispinesib mesylate; CK-0238273; SB-715992
CAS号 336113-53-2(Ispinesib) 514820-03-2(Ispinesib mesylate), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗乳腺癌的纺锤体驱动蛋白(KSP)抑制剂。

Ispronicline;AZD-3480; TC-1734; RJR-1734
CAS号252870-53-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗阿尔兹海默症的α4β2烟碱型受体激动剂。

Istaroxime;Debio-0614; PST-2744; ST-2744
CAS号203737-93-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗心脏衰竭的钠离子/钾离子ATP酶抑制剂。

Itriglumide;CR-2945
CAS号201605-51-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗消化性溃疡,消化不良,胃食管反流疾病(GERD)的缩胆囊素受体拮抗剂。

ITX-5061;CAS号 1252679-52-9(ITX-5061) 848144-15-0(ITX-5061 free), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丙肝的scavenger B1受体拮抗剂。
JNJ-42847922;MIN-202; JNJ-922 CAS号1293281-49-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗伴失眠的重度抑郁症的食欲肽受体-2拮抗剂。

JNJ-872;VRT-0928787; VX-787; JNJ-63623872 CAS号1629869-44-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗甲型流感的病毒蛋白抑制剂。

K-134; OPC-33509 CAS号189362-06-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗动脉粥样硬化的磷酸二酯酶3抑制剂。
KAF-156;CAS号1261113-96-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗疟疾的抗疟药。

KD-025;SLx-2119 CAS号911417-87-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗牛皮癣的rho激酶2抑制剂。

KD-026;SLx-4090 CAS号913541-47-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗2型糖尿病、高脂血症与高甘油三酯血症的微粒体甘油三酯转移蛋白抑制剂。

KNF-299;KRP-203 CAS号 509088-69-1(KRP 203), 509092-16-4(KRP 203), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗移植排斥、自身免疫疾病的1-鞘氨醇磷酸酯受体拮抗剂。

KX-01;KX-2-391; KXO-1; KX-2391
CAS号897016-82-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌,前列腺癌,胃癌以及急性髓性白血病的Src激酶抑制剂。

LCL-161;CAS号1005342-46-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌,多发性骨髓瘤和骨髓纤维化的凋亡抑制蛋白抑制剂。

Lemborexant;E-2006 CAS号1369764-02-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗失眠症的食欲肽受体拮抗剂。

Leteprinim Potassium;AIT-082; SPI-205
CAS号 138117-50-7(Leteprinim) 192564-13-9(Leteprinim potassium), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗帕金森病、脊髓损伤与化疗所致外周神经病的神经营养因子。

LGH-447;PIM-447 CAS号1210608-43-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗多发性骨髓瘤的激酶抑制剂。

LGK-974;WNT-974 CAS号1243244-14-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗结直肠癌的porcupine抑制剂。

Linsitinib;ASP-7487; OSI-906; OSI-906AA CAS号867160-71-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗转移性前列腺癌、胃肠道间质瘤(GISTs)与尤文氏肉瘤的胰岛素样生长因子1受体与胰岛素受体拮抗剂。

Lonafarnib;EBP-994; SCH-066336; Sch-66336 CAS号193275-84-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗丁型肝炎的法尼基转移酶抑制剂。

Lorediplon;GF-015535-00; GF-01553500 CAS号917393-39-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗失眠症的γ-氨基丁酸(GABA)受体平衡药物。

Lucitanib  (德立替尼);AL-3810; CO-3810; E-3810; S-80881 CAS号1058137-23-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗乳腺癌、非小细胞肺癌、小细胞肺癌和实体瘤的血管生成抑制剂。

Luminespib;AUY-922; NVP-AUY-922 CAS号747412-49-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗非小细胞肺癌、胃癌、结肠直肠癌、胰腺癌、淋巴瘤、多发性骨髓瘤的抑制剂。

LX-1031;CAS号945976-76-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗肠易激综合征(IBS)的色胺酸羟化酶-1(TPH1)抑制剂。

LX-7101;CAS号1192189-69-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗原发性开角型青光眼及眼压过高的LIM域结构蛋白/Rho激酶2抑制剂。

LY-2090314;CAS号603288-22-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗胰腺癌的糖原合成酶激酶3β (GSK-3β) 抑制剂。

LY-2456302;CERC-501; LY-DMPF; LYDMPF CAS号1174130-61-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗药物依赖与滥用及治疗抑郁症的kappa-阿片受体拮抗剂。

LY-2874455;CAS号1254473-64-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在治疗晚期癌症的成纤维细胞生长因子受体(FGFR)抑制剂。

LY-2940094;CAS号 1307245-86-8(LY-2940094 Free) 1307245-87-9(LY-2940094), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗重度抑郁症及酒精中毒的孤啡肽受体拮抗剂。

LY-3039478;CAS号1421438-81-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
一种潜在的治疗急性T-细胞成淋巴细胞白血病或T-细胞成淋巴细胞淋巴瘤的notch信号通路抑制剂。



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