Stock list: Targeted anti-cancer inhibitors list-2
GLGP 1837,CAS :1654725-02-6, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
Balovaptan ;1228088-30-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Baloxavir marboxil ;1985606-14-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Bimiralisib ;PQR309,1225037-39-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Cavosonstat ;1371587-51-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Ceclazepide;1801749-44-9 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Citarinostat ;ACY-241;1316215-12-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Wogonin，632-85-9, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
Wogonin, a natural and biologically-active flavonoid found in plants, has been reported to exhibit anticancer effects on several cancer cell types such as osteosarcoma, leukemia, breast cancer and glioma.
Wogonin, a natural and biologically-active flavonoid found in plants, has been reported to exhibit anticancer effects on several cancer cell types such as osteosarcoma, leukemia, breast cancer and glioma.
PNU-74654，113906-27-7, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
PNU-75654 disrupts the Wnt signaling pathway via inhibition of the interaction (KD50=450 nM) between β-catenin and Tcf4.
RRx-001，925206-65-1, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
RRx-001 is a novel epigenetic modulator with potential radiosensitizing activity. It inhibits glucose 6-phosphate dehydrogenase(G6PD) in human tumor cells, binds hemoglobin and drives RBC-mediated redox reactions under hypoxia.
MI-463，1628317-18-9, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
MI-463 is a potent inhibitor of Menin-MLL interaction with an IC50 value of 15.3
PNU-75654 disrupts the Wnt signaling pathway via inhibition of the interaction (KD50=450 nM) between β-catenin and Tcf4.
RRx-001，925206-65-1, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
RRx-001 is a novel epigenetic modulator with potential radiosensitizing activity. It inhibits glucose 6-phosphate dehydrogenase(G6PD) in human tumor cells, binds hemoglobin and drives RBC-mediated redox reactions under hypoxia.
MI-463，1628317-18-9, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
MI-463 is a potent inhibitor of Menin-MLL interaction with an IC50 value of 15.3
CCT196969，1163719-56-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
CCT196969 is a novel orally available, pan-RAF inhibitor with anti-SRC activity.
CCT196969 is a novel orally available, pan-RAF inhibitor with anti-SRC activity.
eFT-508 (eFT508)，1849590-01-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
eFT-508 (eFT508) is a potent and selective MNK1/2 inhibitor, potentially resulting in decreased tumor cell proliferation and tumor growth.
eFT-508 (eFT508) is a potent and selective MNK1/2 inhibitor, potentially resulting in decreased tumor cell proliferation and tumor growth.
KRIBB11，342639-96-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
KRIBB11 abolishes the heat shock-induced luciferase activity with an IC50 of 1.2 μM. It is an inhibitor of the transcription factor Heat Shock Factor 1 (HSF1).
KRIBB11 abolishes the heat shock-induced luciferase activity with an IC50 of 1.2 μM. It is an inhibitor of the transcription factor Heat Shock Factor 1 (HSF1).
SAR-020106，1184843-57-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
SAR-020106 is an ATP-competitive, potent, and selective CHK1 inhibitor with an IC50 of 13.3 nM.
SAR-020106 is an ATP-competitive, potent, and selective CHK1 inhibitor with an IC50 of 13.3 nM.
VPS34 inhibitor 1 (Compound 19, PIK-III analogue)，1383716-46-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM.
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM.
OTS514，1338540-63-8(free base), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
OTS514 is a highly potent TOPK(T-LAK cell-originated protein kinase) inhibitor with an IC50 value of 2.6 nM.
OTS514 is a highly potent TOPK(T-LAK cell-originated protein kinase) inhibitor with an IC50 value of 2.6 nM.
BP-1-102，1334493-07-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
BP-1-102 is a potent, orally bioavailable and selective STAT3 inhibitor, binds Stat3 with an affinity Kd of 504 nM and blocks Stat3-phospho-tyrosine (pTyr) peptide interactions and Stat3 activation at 4-6.8 μM.
BP-1-102 is a potent, orally bioavailable and selective STAT3 inhibitor, binds Stat3 with an affinity Kd of 504 nM and blocks Stat3-phospho-tyrosine (pTyr) peptide interactions and Stat3 activation at 4-6.8 μM.
LY3039478，1421438-81-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
LY3039478是一种有效的Notch抑制剂，IC50为0.41 nM。
GSK583，1346547-00-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
GSK583是一种高度有效的、选择性的RIP2激酶抑制剂，IC50为5 nM。
LCI699(Osilodrostat)，928134-65-0, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
LCI699(Osilodrostat)是有效的11β-hydroxylase抑制剂，11β-hydroxylase是催化皮质醇合成的最后一步。
ARQ 092，1313883-00-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
ARQ 092是新型的、具有口服生物活性的、选择性的AKT抑制剂，在晚期实体肿瘤中具有较好的、可调控的安全性。
S49076，1265965-22-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
S49076是一种新型的、有效的MET, AXL/MER和FGFR1/2/3抑制剂，IC50低于20 nM。
Capsazepine，138977-28-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Capsazepine是capsaicin的拮抗剂，是TRPV1的拮抗剂。
EPZ020411，1700663-41-7(free base), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
praliciguat;1628730-49-3 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
quilseconazole;1340593-70-5 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
relacorilant ;1496510-51-0 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
rislenemdaz;808732-98-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
solriamfetol ;178429-62-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
tapinarof;79338-84-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
teslexivir ;1075798-37-6 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
EPZ020411是有效的、选择性的PRMT6小分子抑制剂，IC50为10 nM。
1400W，214358-33-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
1400W是iNOS的抑制剂，与iNOS缓慢、紧密地结合，具有选择性。
TAK-063,1238697-26-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
TAK-063是新型的、选择性的PDE10A抑制剂，IC50为0.30 nM。
Danshensu，76822-21-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Danshensu(丹参素)，是一种传统中药中的中草药，具有潜在的抗肿瘤和抗血管生成的效果。
UNC0638，1255580-76-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
UNC0638是一种有效的选择性的组蛋白赖氨酸甲基转移酶（HMTase）抑制剂，作用于G9a和GLP，IC50分别为< 15 nM和19 nM，有效且选择性地作用于多种表观遗传和非表观遗传靶点。
Monastrol，329689-23-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Monastrol是一种具有细胞透性的kinesin-5(KIF11)小分子抑制剂，kinesin-5(KIF11)可保持半纺锤体的分离状态。
Psoralen,66-97-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Psoralen是一种天然存在的呋喃香豆素，插入DNA中抑制其合成及细胞分裂。
Acoziborole，Oxaborole，SCYX-7158，CAS：1266084-51-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Acrizanib,CAS:1229453-99-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Aprocitentan ,ACT-132577,1103522-45-7 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
timapiprant ;OC000459;851723-84-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
tinostamustine ;EDO-S101;1236199-60-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
tropifexor;1383816-29-2 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
tulrampator;1038984-31-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
voxelotor ;GBT 440;1446321-46-5, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Atelocantel ,1370540-16-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Atogepant ,1374248-81-3 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
nM.
Importazole，662163-81-7, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
Importazole is a small molecule inhibitor of the transport receptor importin-β specifically blocking importin-β-mediated nuclear import.
SH5-07 (SH-5-07)，1456632-41-9, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
SH5-07 is a robust hydroxamic acid-based STAT3 inhibitor, which induce antitumor cell effects in vitro and antitumor response in vivo against human glioma and breast cancer models.
SH5-07 is a robust hydroxamic acid-based STAT3 inhibitor, which induce antitumor cell effects in vitro and antitumor response in vivo against human glioma and breast cancer models.
UK-371804 HCl，256476-36-5, HPLC 99%, NMR, LCMS is ok, stock more than 10g.
UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin).
UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin).
Azeloprazole;E-3710;Z-215;CAS:955095-45-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Balipodect,TAK-063,1238697-26-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Delpazolid;1219707-39-7 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
Derazantinib;1234356-69-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
dezapelisib;1262440-25-4, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
dorzagliatin ;1191995-00-2 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
dotinurad;1285572-51-1, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
eltanexor ;KPT-8602;1642300-52-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
empesertib ;1443763-60-7 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
etrasimod ;APD334;1206123-37-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
firuglipel ;1371591-51-3, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
THZ1，1604810-83-4(free base), HPLC 99%, NMR, LCMS is ok, stock more than 20g.
THZ1是共价的CDK7抑制剂，对位于经典的激酶结构域外端的半胱氨酸残基具有结合能力，对CDK7选择性高。
SRT2183，1001908-89-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
SRT2183是sirtuin蛋白亚型SIRT1的小分子激活剂。
AZD3293 (LY3314814)，1383982-64-6, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
AZD3293(LY3314814)是BACE抑制剂。
Fruquintinib;HMPL-013;1194506-26-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
imarikiren;TAK-272;1202265-63-1 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
itanapraced;CHF5074;749269-83-8 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
lanabecestat ;AZD3293;1383982-64-6 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
landipirdine;1000308-25-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
lanifibranor;IVA-337;927961-18-0 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
mavacamten;1642288-47-8 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
midomafetamine ;42542-10-9 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
miransertib ;ARQ-092;1313881-70-7, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
mitapivat;1260075-17-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
mocravimod ;KRP 203;509092-16-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
molibresib ;GSK 525762A;1260907-17-2, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
neflamapimod VX-745;209410-46-8, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
nemiralisib;GSK2269557;1254036-71-9, HPLC 99%, NMR, LCMS is ok, stock more than 20g.
olodanrigan;EMA401;1316755-16-4 , HPLC 99%, NMR, LCMS is ok, stock more than 20g.
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