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執大象，天下往，往而無害，安平泰
WEB: www.eosmedchem.com
EMAIL: info@eosmedchem.com; eosmedchem@gmail.com; eosmedchem@qq.com
TEL: 0086-531-69905422
GMP PLANT: No. 37, Yulong Road, Qufu City, Shandong Province.
Description: Pifithrin-alpha is a p53 inactivator. It also has neuroprotective activity against strokes.
Name: Pifithrin-alpha
CAS#: 63208-82-2
Chemical Formula: C16H19BrN2OS
Exact Mass: 366.0401
Molecular Weight: 367.3
Elemental Analysis: C, 52.32; H, 5.21; Br, 21.75; N, 7.63; O, 4.36; S, 8.73
Synonym: Pifithrin-alpha; Pifithrin alpha; PFT-alpha; PFTalpha; PFT alpha;
IUPAC/Chemical Name: 2-(2-Imino-4,5,6,7-tetrahydro-1,3-benzothiazol-3-yl)-1-(4-methylphenyl)ethanone;hydrobromide
InChi Key: HAGVCKULCLQGRF-UHFFFAOYSA-N
InChi Code: InChI=1S/C16H18N2OS.BrH/c1-11-6-8-12(9-7-11)14(19)10-18-13-4-2-3-5-15(13)20-16(18)17;/h6-9,17H,2-5,10H2,1H3;1H
SMILES Code: CC1=CC=C(C(CN2C(SC3=C2CCCC3)=N)=O)C=C1.[H]Br
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility: Soluble in DMSO
Shelf Life: >2 years if stored properly
Drug Formulation: This drug may be formulated in DMSO
Stock Solution Storage: 0 - 4 C for short term (days to weeks), or -20 C for long term (months).
Harmonized System Code: 293490
REFERENCES
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