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2017年6月8日星期四

EOS Building block June 9th


 81237-69-6 5-bromo-1,2,3,4-tetrahydroisoquinoline

864373-47-7
oxetane-2-carboxylic acid
[1000343-69-0]6-Bromo-5-methyl-1H-indazole
[1000932-73-9](2,3-Dihydro-1H-indol-3-ylmethyl)-carbamic acid tert-butyl ester
[1002334-12-4]1-Phenyl-1H-pyrazole-4-boronic acid pinacol ester
[1017781-45-1]3-(4-tert-Butoxycarbonylamino-phenyl)-3-oxo-propionic acid ethyl ester
[1017781-46-2]3-(2-tert-Butoxycarbonylamino-phenyl)-3-oxo-propionic acid ethyl ester
[1017781-47-3]3-(3-tert-Butoxycarbonylamino-phenyl)-3-oxo-propionic acid ethyl ester
[1020966-78-2]4-Bromo-benzofuran-3-one
[1022961-12-1]2-Amino-3-chloro-5-fluoro-benzoic acid
[102735-84-2]5-Chloro-1H-indazole-3-carbaldehyde
[103030-70-2]5-Methoxy-1,2,3,4-tetrahydro-isoquinoline
[1033194-55-6(Benzenesulfonyl-isopropyl-amino)-acetic acid
[105174-97-8]3-Bromo-isoxazole-5-carboxylic acid ethyl ester
[105174-97-8]3-Bromo-isoxazole-5-carboxylic acid ethyl ester
[1064194-10-0]tert-Butyl 3-bromoazetidine-1-carboxylate 
[1092350-92-9][4-(2-Amino-ethyl)-cyclohexyl]-carbamic acid tert-butyl ester
[110234-68-9]4,4,4-Trifluoro-3-oxo-butyronitrile
[110928-44-4]4-Hydroxymethyl-cyclohexanecarboxylic acid methyl ester
[111454-71-8]3-Bromo-isoxazole
[1123169-43-6]7-Bromo-quinazolin-4-ylamine
[1123169-45-8]6-Bromo-3,4-dihydro-2H-quinoline-1-carboxylic acid tert-butyl ester
[113283-94-6](4-Methylamino-phenyl)-carbamic acid tert-butyl ester
[1134327-91-5](5-Bromo-pyrimidin-2-yl)-acetic acid ethyl ester
[114079-50-4]2-Methylamino-propionic acid methyl ester hydrochloride
[114744-51-3]7-Bromo-1,2,3,4-tetrahydro-quinoline
[115514-66-4]4-Bromo-pyridazine
[116070-31-6]2,6-Dichloro-4-methyl-benzaldehyde
[1167418-13-4]Quinoxaline-6-boronic acid pinacol ester
[1170108-38-9]3-Boc-aminomethyl-azetidine hydrochloride
[1171047-31-6]2,6-Dimethoxy-benzamidine hydrochloride
[1176754-31-6]1-Methyl-1H-indazole-5-carboxylic acid
[1185302-13-9]2,2,2-Trifluoro-1-(3-fluoro-phenyl)-ethylamine hydrochloride
[1187928-61-5]7-Bromo-benzothiazole-2-carboxylic acid methyl ester
[1187932-85-9](R)-2-Methyl-1-pyridin-3-yl-propylamine
[1187933-07-8]3-Hydroxy-cyclopentanecarboxylic acid ethyl ester
[1211516-09-4]6-Bromo-1H-pyrazolo[4,3-b]pyridin-3-ylamine
[1216012-87-1]2-Methyl-oxazole-5-carboxylic acid
[121632-81-3]4-(2-Cbz-aminoethyl)benzoic acid
[1220039-48-4](3-Bromo-5-chloro-phenyl)-hydrazine hydrochloride
[1227270-50-9]5-Bromo-1H-indazol-6-ol
[1234710-03-2]4-(4(5)-Methyl-1H-imidazol-2-yl)-piperidine-1-carboxylic acid tert-butyl ester
[1256360-04-9][3-Methyl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-carbamic acid tert-butyl ester
[1258940-00-9](S)-3-Phenyl-piperidine hydrochloride
[1262409-43-7]4-Oxo-cyclohexanesulfonyl chloride
[1263378-30-8]3-Methyl-tetrahydro-pyran-4-ylamine
[1263378-39-7]2-Cyclopropyl-oxazole-5-carboxylic acid
[127685-30-7](S)-3-Phenyl-3-(4-trifluoromethyl-phenoxy)-propylamine hydrochloride
[128740-14-7]6-Benzyl-octahydro-pyrrolo[3,4-b]pyridine
[129477-21-0]5-Bromo-2-methyl-nicotinic acid ethyl ester
[129488-10-4]1-Boc-5-amino-indazole
[1305324-99-5]5-Iodo-1H-pyrazolo[3,4-b]pyridine
[13058-77-0]8-Chloro-[1,7]naphthyridine
[131747-45-0](4-Bromo-pyridin-2-yl)-methanol
[131747-63-2]4-Bromo-pyridine-2-carbaldehyde
[132095-53-5]5-Bromo-3,4-dihydro-1H-naphthalen-2-one
[132205-73-3]5-Amino-indan-1-carboxylic acid methyl ester hydrochloride
[13296-30-5]2-(6,6-Dimethyl-bicyclo[3.1.1]hept-2-en-2-yl)-ethylamine
[1341529-37-0]3-Cyclobutoxy-azetidine hydrochloride 
[13472-00-9]4-(2-Amino-ethyl)-phenylamine
[135484-74-1]2-Amino-6-bromo-benzaldehyde
[13623-87-5]1,2,3,4-Tetrahydro-[1,8]naphthyridine
[137069-23-9]Methyl-(2-m-tolyl-ethyl)-amine
[1375472-17-5]2,5-Dimethyl-cyclopentylamine hydrochloride
[137837-55-9]Pyrazolo[1,5-a]pyridin-3-ylamine
[138537-66-3](S)-6-(2-Methylamino-propyl)-benzo[1,3]dioxol-4-ol hydrochloride
[138614-32-1](R)-3-Phenyl-3-(4-trifluoromethyl-phenoxy)-propylamine hydrochloride
[1391436-37-5](S)-2,2,2-Trifluoro-1-(3-fluoro-phenyl)-ethylamine hydrochloride
[1391527-41-5](R)-2,2,2-Trifluoro-1-(3-fluoro-phenyl)-ethylamine hydrochloride
[13924-94-2]5-Amino-pyrazine-2-carboxylic acid methyl ester
[13958-86-6]5-Methyl-pyridine-3,4-diamine
[13993-61-8]1,2,3,4-Tetrahydro-[1,5]naphthyridine
[1400999-64-5]4-(1-Amino-cyclopropyl)-phenylamine dihydrochloride
[1402672-54-1]2-Chloro-6-methyl-benzamidine hydrochloride
[1414960-64-7](R)-5-Bromo-2,3-dihydro-benzofuran-3-ylamine hydrochloride
[1430839-87-4]2-Amino-4-fluoro-5-(4-methyl-[1,4]diazepan-1-yl)-benzoic acid
[1439-09-4]5-Bromo-4-methyl-pyrimidine
[14613-37-7]C-(1-Methyl-piperidin-3-yl)-methylamine
[146137-92-0]5-Trifluoromethyl-benzo[b]thiophene-2-carboxylic acid methyl ester
[148404-28-8]cis-5-Oxo-hexahydro-cyclopenta[c]pyrrole-2-carboxylic acid tert-butyl ester
[149965-78-6]But-3-ynyl-carbamic acid benzyl ester
[1515866-60-0]7-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazine
[152626-78-3]5-Bromo-6-methoxy-1H-indazole
[153138-05-7]2-Methyl-oxazole-5-carbaldehyde
[15540-81-5]1-Bromo-2,5-dimethyl-4-nitro-benzene
[159634-59-0]1'-Boc-3-oxo-2,3-dihydrospiro[indene-1,4'-piperidine]
[159783-22-9]3,5-Difluoro-pyridin-4-ylamine
[16205-46-2]Pyrazolo[1,5-a]pyridine-3-carboxylic acid
[1623461-06-2]6-Amino-2-bromo-3-fluoro-benzoic acid
[171346-87-5]2-(2-Phenyl-imidazo[1,2-a]pyridin-3-yl)-ethylamine
[17402-83-4]Benzo[b]thiophen-4-ylamine
[17429-00-4]3-Methoxy-cyclohexanone
[17680-55-6]7-Bromo-1,2,3,4-tetrahydro-isoquinoline
[17965-71-8]3-Bromo-[1,5]naphthyridine
[17965-78-5]3-Bromo-[1,8]naphthyridine
[180465-55-8]Spiro[indene-1,4'-piperidin]-3(2H)-one
[180975-66-0]cis-1-Boc-2,6-dimethyl-piperazine
[187658-19-1]1-(5-Fluoro-benzo[b]thiophen-3-yl)-ethanone
[194543-22-1](Tetrahydro-pyran-4-yl)-hydrazine hydrochloride
[195447-85-9]2-Methyl-4-trifluoromethyl-nicotinic acid
[19577-84-5]2-(4-Methyl-piperazin-1-ylmethyl)-aniline
[21294-14-4]2-Aminomethyl-benzylamine dihydrochloride
[214614-97-81-Boc-7-bromo-1,2,3,4-tetrahydro-quinoline
[218301-87-2]N-Boc-4-amino-3-fluoro-benzeneboronic acid
[22190-35-8]6-Bromo-1,2,3,4-tetrahydro-quinoline
[253176-93-1]3-Bromomethyl-azetidine-1-carboxylic acid tert-butyl ester
[253801-04-6]1H-Indazole-5-carbaldehyde
[25672-97-3]2-Aminomethyl-benzoic acid
[26130-49-4]3,5-Dimethoxy-benzamidine
[26673-30-3]5-Chloro-tetral-1-on
[26673-31-4]6-Chloro-tetral-1-on
[26673-32-5]7-Chloro-3,4-dihydro-2H-naphthalen-1-one
[267413-25-2]C-(1H-Indazol-5-yl)-methylamine
[281203-98-3]6-Thiophen-3-yl-1H-indazole
[2812-32-0]N,N-Dimethyl-L-valine
[30273-40-6]4-Bromo-2,5-dimethyl-phenylamine
[31434-93-2]3-(1H-Imidazol-4-yl)-propionic acid methyl ester
[316833-42-8](S)-2-amino-3-phenoxypropanoic acid
[32868-32-9]4-(2-Methylamino-ethyl)-phenylamine
[33537-99-4]6-Chloro-1,2,3,4-tetrahydro-isoquinoline
[338949-36-3]6,6a,7,8,9,10-Hexahydro-5H-pyrido[1,2-a]quinoxaline
[341-24-2]7-Fluoro-1H-indazole
[350683-67-9](4-Propylphenyl)-hydrazine hydrochloride
[35212-96-5]5-Chloro-benzo[b]thiophene-2-carboxylic acid methyl ester
[3970-37-4]1-Bromo-2-chloro-3-nitro-benzene
[3973-62-4]3-Phenyl-piperidine
[39889-94-6]2-Methyl-pyrimidin-5-ylamine
[406923-64-6]5-Fluoro-1,2,3,4-tetrahydro-isoquinoline
[406923-91-9]7-Fluoro-1,2,3,4-tetrahydro-isoquinoline
[40740-57-6]5-Fluoro-benzo[b]thiophene-3-carboxylic acid
[41110-28-5]3-Methyl-pyrazine-2-carboxylic acid
[41239-40-1]Methyl-(2-morpholin-4-yl-ethyl)-amine
[42839-04-3]Pyrimidine-4-carbonitrile
[42887-67-2]1-(2-Amino-5-methoxy-phenyl)-ethanone
[43207-78-9]7-Methoxy-1,2,3,4-tetrahydro-isoquinoline
[4363-13-7]3-Phenyl-azetidine
[4441-59-2]4-Cyclohexyl-butylamine
[4487-57-4]2,4-Dibromo-5-nitro-pyridine
[4498-69-5]6-Methyl-1H-indazole-3-carboxylic acid ethyl ester
[450416-58-7](R)-3-Phenyl-piperidine hydrochloride
[4507-84-0]3-Nitro-naphthalene-1-carboxylic acid
[485841-48-3]5-Fluoro-1H-indazole-3-carbaldehyde
[501944-79-2]2-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-oxazole
[503417-30-9]1-m-Tolyl-cyclopropylamine
[50476-72-7]4-Chloro-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester
[50675-25-7]C-(2,2-Dimethyl-tetrahydro-pyran-4-yl)-methylamine
[51984-71-5]2-Methyl-5-nitro-nicotinic acid ethyl ester
[52412-10-9]5,6-Dihydroxy-pyrimidine-4-carboxylic acid
[52516-20-8][2-(3-Chloro-phenyl)-ethyl]-methyl-amine
[53544-13-1]3-Cyano-2-oxo-propionic acid ethyl ester sodium salt
[5400-79-3]3-Oxo-cyclopentanecarboxylic acid ethyl ester
[54013-06-8]5-Amino-pyrazine-2-carboxylic acid ethyl ester
[5435-66-5]1-(3-Nitro-phenyl)-butane-1,3-dione
[54569-28-7]4-Bromo-[1,8]naphthyridine
[5465-28-1]2-Ethyl-2-phenyl-butyric acid
[55052-27-2]6-Chloro-1H-pyrrolo[2,3-b]pyridine
[5571-03-9]2-Methyl-pyrimidine-5-carboxylic acid methyl ester
[56181-39-6]5-Bromo-4-chloro-pyrimidine
[5621-13-6]2,7-Dimethyl-1H-indole
[5649-36-5]2,6-Dimethyl-1H-indole
[5708-19-0](S)-(-)-Cyclohex-3-enecarboxylic acid
[573768-09-9]4-Amino-2-chloro-3-methyl-benzonitrile
[57631-11-5]5-Bromo-3-trifluoromethyl-1H-indazole
[5763-55-3]2-Cyclopentyl-ethylamine
[5780-66-5]Pyrazine-2-carbaldehyde
[58123-57-2]C-Quinolin-5-yl-methylamine
[59123-22-7]2-amino-3-phenoxypropanoic acid
[59123-23-8](R)-2-amino-3-phenoxypropanoic acid
[59128-15-3](6-Bromo-imidazo[1,2-a]pyridin-2-yl)-acetic acid
[59376-81-7]5-Chloro-1,2,3,4-tetrahydro-naphthalen-1-ylamine
[5938-16-9]4-(4-Methoxy-phenyl)-pyridine
[59489-71-3]5-Bromo-pyrazin-2-ylamine
[6004-60-0]1-Cyclopentyl-ethanone
[62150-46-3]4-Bromo-pyridine-2-carboxylic acid amide
[624-97-5]2-Methyl-pent-4-en-2-ol
[63155-11-3]Pyrimidin-2-yl-acetic acid ethyl ester
[651059-70-0]2-Methyl-oxazole-5-carboxylic acid methyl ester
[6558-66-3]7-Methyl-imidazo[1,2-a]pyrimidine
[6786-30-7]3,4-Dihydro-2H-benzo[b]oxepin-5-one
[6914-76-7]1-Methyl-cyclopropanecarboxylic acid
[69383-60-4]5-Bromo-2,4-dimethyl-phenylamine
[70060-12-7]5-Fluoro-benzo[b]thiophene
[717843-56-6]3-Bromo-2-methoxy-5-methyl-pyridine
[73075-43-1]5-chloro-1,2,3,4-tetrahydroisoquinoline
[73792-08-2]4-Amino-2-fluoro-benzoic acid methyl ester
[74213-24-4]1,1-Dibromoformaldoxime
[7498-54-6]3-tert-Butyl-benzoic acid
[76179-43-6]4,5-Diiodo-benzene-1,2-diamine
[767-70-4]7-Bromo-benzothiazole
[771454-16-1]8-Methoxy-thiochroman-3-ylamine
[775576-21-1]2-(5-Chloro-thiophen-2-yl)-ethylamine
[78917-44-9]Ethyl 3-benzofuran-2-yl-3-oxo-propionate
[82257-09-8]3-Bromo-4-methoxy-pyridine
[82771-60-6]7-Chloro-1,2,3,4-tetrahydro-isoquinoline
[836619-77-3](3-Bromo-4-fluoro-phenyl)-carbamic acid tert-butyl ester
[844891-30-1](2-Fluoro-6-formyl-phenyl)-carbamic acid tert-butyl ester
[858227-11-9]6-Methyl-1H-indazole-3-carboxylic acid methyl ester
[862723-42-0]1H-Indazole-5-boronic acid pinacol ester
[863118-41-6]6-Trifluoromethyl-benzo[b]thiophene-2-carboxylic acid methyl ester
[864771-44-8]1-Boc-1H-indalzole-5-boronic acid pinacol ester
[866848-94-4]6-Bromo-indan-1-one 1,2-ethanediol ketal
[869783-22-2]6-Thiophen-2-yl-1H-indazole-3-carboxylic acid
[871791-79-6]3-Isopropoxy-azetidine
[876716-04-0](1-Isopropyl-piperidin-4-ylmethyl)-methyl-amine
[878740-89-7]2-Pyrazin-2-yl-ethylamine dihydrochloride
[882402-12-2]C-Oxetan-2-yl-methylamine
[88491-61-6]3-Bromo-pyridazine
[885271-54-5]5-Chloro-imidazo[1,5-a]pyridine-1-carboxylic acid ethyl ester
[885271-72-7]6-Bromo-1H-indazole-3-carbaldehyde
[885271-95-4]6-Furan-2-yl-1H-indazole
[885272-17-3]6-Boc-2,6-diaza-spiro[3.5]nonane
[885272-18-4]6-(Tetrahydro-pyran-4-yl)-1H-indazole
[885272-33-3]6-(1-Methyl-piperidin-4-yl)-1H-indazole
[885272-41-3]5-Thiophen-3-yl-1H-indazole
[885272-43-5]5-Furan-2-yl-1H-indazole
[885272-45-7]5-Furan-3-yl-1H-indazole
[885278-02-4]2-(1-Boc-piperazin-4-yl-methyl)-aniline
[885278-71-7]7-Bromo-1H-indazole-3-carboxylic acid
[885279-52-7]Methyl 7-bromo-1H-indazole-3-carboxylate
[885518-46-7]6-Bromo-4-nitro-1H-indazole
[885519-21-1]6-Bromo-4-methoxy-1H-indazole
[885520-35-4]4-Bromo-6-fluoro-1H-indazole
[885693-20-9]1-Boc-5,6-dihydro-2H-pyridine-3-boronic acid pinacol ester
[886528-42-3]4-(2,2,2-Trifluoroethoxy)phenylboronic acid pinacol ester
[887576-89-8]7-Bromo-1H-indazole-3-carbaldehyde
[887583-90-6]4-Bromo-2-trifluoromethyl-pyridine
[89614-96-0]3-Amino-cyclopentanecarboxylic acid
[89891-69-0]3-Bromo-4-formyl-benzonitrile
[899900-52-8]N,N-Dimethyl-D-valine
[90348-29-1]5-Nitro-1H-indazole-3-carbonitrile
[90561-75-4]2-(4-Bromo-phenyl)-cyclopropylamine
[90766-34-0]3-Bromo-naphthalen-1-ylamine
[912773-24-1]6-Bromoimidazo[1,2-a]pyrazine
[914672-66-5]3-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-pyrazole-1-carboxylic acid tert-butyl ester
[915021-19-1]4,6-Dimethoxypyridine-3-boronic acid
[91550-08-2](S)-1-Boc-2-acetyl-pyrrolidine
[921938-63-8](4-Bromo-thiophen-3-ylmethyl)-methyl-amine
[92385-37-0]5-Chloro-quinolin-4-ylamine
[92629-13-5]2-Phenyl-oxazole-5-carbaldehyde
[935466-69-6]6-Amino-4-chloro-7-azaindole
[936829-23-1]3-Amino-2,3-dihydro-indole-1-carboxylic acid tert-butyl ester
[944142-47-6]1-(Tetrahydro-pyran-4-yl)-cyclopropylamine
[944900-52-1]2-Amino-oxazole-4-carboxylic acid
[944904-38-5]7-Fluoro-3-iodo-1H-indazole
[954238-88-1](2-Amino-5-chloro-phenyl)-carbamic acid tert-butyl ester
[954240-97-2]5,6-Dihydroxy-2-methyl-pyrimidine-4-carboxylic acid amide
[954241-13-5]5,6-Dihydroxy-2-isopropyl-pyrimidine-4-carboxylic acid amide
1000342-95-94-Bromo-6-trifluoromethyl-1H-indazole
1000931-58-71-N-Boc-octahydro-[1,5]naphthyridine
100123-25-9Ethyl 5-bromo-3-formyl-1H-indole-2-carboxylate
100123-25-9Ethyl 5-bromo-3-formyl-1H-indole-2-carboxylate
1001353-86-1(S)-1-Boc-4,4-dimethyl-pyrrolidine-2-carboxylic acid ethyl ester
1001756-21-34-Amino-6-chloro-pyridine-3-carbaldehyde
1005077-74-66-Amino-2-aza-bicyclo[2.2.1]heptane-2-carboxylic acid tert-butyl ester
1005397-62-52,6-Dimethyl-piperidin-4-one hydrochloride
1005397-64-7cis-2,6-Dimethyl-4-oxo-piperidine-1-carboxylic acid tert-butyl ester
101048-76-42-Fluoro-4-formyl-benzonitrile
1015460-59-97-Bromo-5H-pyrido[4,3-b]indole
1016167-98-8(S)-3-Isopropoxy-pyrrolidine
1017422-91-1C-(1-Methyl-1H-benzoimidazol-2-yl)-C-pyridin-3-yl-methylamine
1017423-86-7C-(1-Methyl-1H-benzoimidazol-2-yl)-C-pyridin-2-yl-methylamine
1017470-41-5C-(1-Ethyl-1H-benzoimidazol-2-yl)-C-phenyl-methylamine
1017781-53-1tert-butyl 4-(3-oxo-3-phenylpropanoyl)piperidine-1-carboxylate
1017781-98-42,5-Dimethyl-4,5,6,7-tetrahydro-oxazolo[4,5-c]pyridine
102014-40-41-Methyl-piperidin-3-one hydrochloride monohydrate
10271-85-9Isothiazole-5-carboxylic acid
10271-85-9 isothiazole-5-carboxylic acid
102732-63-8(1H-Pyrazol-3-yl)-acetic acid
10299-61-32,4-Dimethyl-1H-indole
10315-07-81-Benzyl-piperidine-4-carboxylic acid
1034769-88-45-bromo-4-chloro-1H-pyrazolo[3,4-b]pyridine
103862-63-14-Chloro-6-ethoxy-quinoline
104575-40-82-(4-Fluoro-phenyl)-4-methyl-1H-imidazole
104704-40-74-Bromo-1-methyl-isoquinoline
105174-97-83-Bromo-isoxazole-5-carboxylic acid ethyl ester
105175-00-62-(3-Bromo-isoxazol-5-yl)-ethanol
105250-16-6(2-Methyl-pyridin-4-yl)-methanol
105499-10-3(1-Methyl-2-oxo-ethyl)-carbamic acid benzyl ester
10602-00-34-Ethynyl-benzoic acid
1060801-10-6(6-Aminomethyl-pyridin-2-yl)-carbamic acid tert-butyl ester
1060806-76-94-Amino-6-methoxy-nicotinic acid
1060809-69-94-Amino-6-bromo-pyridine-3-carbaldehyde
1060809-85-94-Hydroxy-pyridine-2-carbaldehyde
1060810-09-42-Bromo-6-methyl-nicotinic acid
1060815-26-01-Pyridin-4-yl-cyclopropylamine
1065073-48-4(2-methyloxazol-5-yl)methanol
106-56-92,5-Dimethyl-morpholine
106833-79-82-Phenyl-oxazole-5-carboxylic acid
1082041-34-65-Bromo-4-methyl-1H-indazole
1083197-78-74-Trifluoromethyl-pyridine-3-carbaldehyde
1086392-24-63-Aminomethyl-2,3-dihydro-indole-1-carboxylic acid tert-butyl ester
108805-39-65-Methoxy-benzo[d]isoxazole-3-carboxylic acid 
1089340-69-13-Hydroxy-cyclobutanecarboxylic acid methylamide
1092579-78-65-bromo-4-chloro-3-iodo-1H-pyrazolo[3,4-b]pyridine
109397-72-0[4,4']Bipiperidinyl-1-carboxylic acid benzyl ester
1096936-82-1C-(1-Cyclopropyl-1H-benzoimidazol-2-yl)-C-phenyl-methylamine
1097146-30-94-Isopropoxy-piperidine hydrochloride
1099570-25-8benzyl 6-hydroxy-2-azabicyclo[2.2.1]heptane-2-carboxylate
111376-39-73-(3-Oxo-propyl)-benzonitrile
111454-71-83-Bromo-isoxazole
1118786-85-8(2-Aza-spiro[3.3]hept-6-yl)-carbamic acid tert-butyl ester hydrochloride
1118786-86-92-(Boc-amino)-6-oxo-spiro[3.3]heptane
1123169-50-54-Chloro-7-methoxy-quinoline-3-carboxylic acid methyl ester
1123169-54-97-Benzyloxy-1H-indazole-3-carbonitrile
112461-31-16-Oxa-3-aza-bicyclo[3.1.1]heptane
1130053-86-9(2R,5S)-2,5-Dimethyl-morpholine
1134327-87-94-Bocamino-1-pyridin-3-yl-butan-1-one
1134327-91-5(5-Bromo-pyrimidin-2-yl)-acetic acid ethyl ester
113707-75-8(R)-(2-Iodo-1-methyl-ethyl)-carbamic acid benzyl ester
114072-02-52-Pyrimidin-2-yl-ethanol
1147107-39-84-Difluoromethoxy-piperidine
1147557-97-86-Hydroxy-2-aza-spiro[3.3]heptane-2-carboxylic acid tert-butyl ester
1153767-91-91,8-Diaza-spiro[4.5]decane-1-carboxylic acid tert-butyl ester hydrochloride
1159821-30-32-(Tetrahydro-pyran-4-yl)-pyrimidin-4-ylamine
116129-07-82-Aza-bicyclo[2.1.1]hexane-1-carboxylic acid hydrochloride
1174028-22-85-Bromo-6-methyl-nicotinic acid methyl ester
1180112-41-71,7-Diaza-spiro[3.5]nonane-7-carboxylic acid tert-butyl ester hydrochloride
118054-57-2(1H-Pyrazol-3-yl)-acetic acid hydrochloride
1181816-12-56-Oxo-2-aza-spiro[3.3]heptane-2-carboxylic acid tert-butyl ester
1185138-23-1C-(4-Trifluoromethyl-pyridin-3-yl)-methylamine hydrochloride
1187174-14-65,7-difluoro-1,2,3,4-tetrahydroisoquinoline
1187243-09-96-Formyl-2,3-dihydro-1H-indole
1187582-59-7Ethyl 2-bromo-5-methyl-oxazole-4-carboxylate
1187929-19-62-Hydrazino-benzenesulfonamide hydrochloride
1187930-92-24-Amino-hexahydro-cyclopenta[c]pyrrole-2-carboxylic acid tert-butyl ester
1187932-43-9(R)-3-Isopropoxy-pyrrolidine
1187933-07-83-Hydroxy-cyclopentanecarboxylic acid ethyl ester
1188265-73-73-(2-Hydroxy-ethyl)-piperazine-1-carboxylic acid tert-butyl ester
118994-86-8Oxazole-5-carbaldehyde
1190862-70-45-Bromo-6-methyl-nicotinic acid ethyl ester
1192347-65-12-Methanesulfonyl-5-methoxy-benzylamine
1194374-71-45-Fluoro-2-formyl-benzoic acid methyl ester
1196155-38-02-Chloro-6-trifluoromethyl-isonicotinonitrile
1196156-67-82-Amino-6-bromo-pyridine-3-carbaldehyde
1196157-42-25,7-Dichloro-1H-pyrazolo[4,3-d]pyrimidine
1196-79-82,5-Dimethyl-1H-indole
1203566-77-1(3R,4R)-(4-Hydroxy-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
1203683-26-43-(4-Bromo-phenyl)-piperidine hydrochloride
1205544-78-01-(aminomethyl)cyclopropane-1-carbonitrile hydrochloride
1210935-33-3(R)-(1-Methyl-pyrrolidin-3-yl)-methanol
1211525-26-66-Chloro-4-phenyl-pyridin-2-ylamine
1211526-53-22-Aza-spiro[3.3]heptane-2,6-dicarboxylic acid 2-tert-butyl ester
1211567-54-23-Phenyl-oxetan-3-ylamine
1211586-09-26-Amino-2-aza-spiro[3.3]heptane-2-carboxylic acid tert-butyl ester
1211586-14-91-N-Boc-octahydro-pyrrolo[3,2-b]pyridine
1212822-72-4Octahydro-cyclopenta[c]pyrrol-4-ol
1214332-41-82,6-Difluoro-3-hydroxy-benzoic acid methyl ester
1216012-87-12-methyloxazole-5-carboxylic acid
1216012-87-12-Methyl-oxazole-5-carboxylic acid
1217047-14-73-tert-Butyl-isoxazole-4-carboxylic acid
1220039-87-15-Bromo-4-chloro-pyrimidine hydrochloride
1220039-87-15-Bromo-4-chloro-pyrimidine hydrochloride
1227269-41-1(4-Methoxy-1H-indol-6-yl)-carbamic acid tert-butyl ester
122851-60-9(3-Bromo-pyridin-2-yl)-acetonitrile
123278-03-53-Chloro-2-iodo-benzoic acid
1235440-17-11,7-Diaza-spiro[3.5]nonan-2-one
1235440-17-11,7-Diaza-spiro[3.5]nonan-2-one
1240589-57-4(6R)-Methyl-piperazin-2-one
1240598-14-42-Bromo-5-methyl-oxazole-4-carbaldehyde
1240725-66-95-Chloro-1H-pyrazolo[3,4-b]pyridine
1243243-89-12-[4-(2-Methyl-pyridin-4-yl)-phenyl]-N-(4-pyridin-3-yl-phenyl)-acetamide
1243245-69-3[4-(2-Methyl-pyridin-4-yl)-phenyl]-acetic acid
124779-00-63-Cyano-2-methyl-acrylic acid ethyl ester
1249024-78-98-Methanesulfonyl-8-aza-bicyclo[3.2.1]oct-3-ylamine
1249198-23-94-Pyrrolidin-2-yl-pyrimidin-2-ylamine
1250358-31-62,6-Bis-methoxymethyl-pyrimidin-4-ylamine
1250444-46-21-Oxo-1,2,3,4-tetrahydro-isoquinoline-8-carboxylic acid methyl ester
1251013-07-6cis-2-Boc-octahydro-pyrrolo[3,4-d]azepine
1251013-07-6cis-2-Boc-octahydro-pyrrolo[3,4-d]azepine
1253730-25-42-Oxetan-3-yl-ethylamine
1254328-26-12,3-Dimethyl-isonicotinic acid methyl ester
1255099-41-2Spiro[3.3]hept-2-ylamine
1256358-90-32-(Hydroxy)pyridine-4-boronic acid pinacol ester
1257072-34-66-Bromo-3-chloro-pyrazine-2-carbonitrile
125781-45-5(S)-4,4-Dimethyl-pyrrolidine-2-carboxylic acid ethyl ester
1260606-18-52S,3S-1-Boc-2-methyl-piperidine-3-carboxylic acid
1260783-69-4Methyl-pyrimidin-4-ylmethyl-amine hydrochloride
1260834-38-56-Nitro-1H-benzoimidazole-2-carbaldehyde
1260890-57-0(2-Boc-amino-pyridin-4-yl)-acetic acid methyl ester
1261475-16-41-Bromo-3-isocyanato-2-methyl-benzene
1263365-47-4cis-Octahydro-isoindol-5-ol
1263378-34-22-Bromo-4-fluoro-5-iodo-benzoic acid
126971-79-7tert-butyl (2-(hydroxy(pyridin-4-yl)methyl)phenyl)carbamate
127232-41-1Oxazol-5-yl-methanol
127430-46-0Hexahydro-cyclopenta[c]pyrrol-4-one hydrochloride
1277168-52-14-Boc-octahydro-pyrrolo[3,2-b]pyridine
127926-24-32-Boc-2-aza-bicyclo[2.1.1]hexane-1-carboxylic acid
128740-14-76-Benzyl-octahydro-pyrrolo[3,4-b]pyridine
1289103-14-56-Methyl-4-trifluoromethyl-pyridine-3-carbaldehyde
129295-31-46-Chloro-1H-indazole-3-carboxylic acid
129477-21-05-Bromo-2-methyl-nicotinic acid ethyl ester
1303975-05-4(R)-4,4-Dimethyl-pyrrolidine-2-carboxylic acid
13047-01-33-Bromo-tetrahydro-pyran
130658-14-94-Oxo-hexahydro-cyclopenta[c]pyrrole-2-carboxylic acid tert-butyl ester
1312760-59-06-Chloro-[1,5]naphthyridin-4-ol
131747-45-0(4-Bromo-pyridin-2-yl)-methanol
131747-60-9(2-Fluoro-pyridin-4-yl)-methanol
131747-63-24-Bromo-pyridine-2-carbaldehyde
131747-69-82-Fluoro-pyridine-4-carbaldehyde
131774-72-63-Hydrazino-benzenesulfonamide
131774-72-63-Hydrazino-benzenesulfonamide
13220-27-41-Methyl-pyrrolidin-3-ylamine
132205-76-65-Chloro-indan-1-carbonitrile
13230-03-02-Ethyl-4-nitro-1H-imidazole
132414-50-71-Benzyl-octahydro-pyrrolo[3,4-b]pyrrole
13273-53-54-Bromo-1-methyl-1H-[1,2,3]triazole
133277-08-46-Bromo-1,2,3,4-tetrahydro-naphthalen-2-ylamine hydrochloride
13373-32-52-Isopropyl-4-nitro-1H-imidazole
13374-55-51-Aza-spiro[3.5]nonane
1342158-87-51-Difluoromethoxy-2-ethynyl-benzene
1343864-38-92-Aza-spiro[4.4]nonane-4-carboxylic acid
134682-54-51,3-Dihydro-pyrrolo[3,2-c]pyridin-2-one
1350475-33-06-Methoxy-3-nitro-pyridine-2-carboxylic acid
13600-43-64-Trifluoromethyl-nicotinonitrile
13600-49-26-methyl-4-(trifluoromethyl)nicotinonitrile
13600-49-26-Methyl-4-trifluoromethyl-nicotinonitrile
13626-59-03-methoxyisoxazole-5-carboxylic acid
13626-59-03-Methoxy-isoxazole-5-carboxylic acid
136866-27-83,5-Dichloro-pyrazine-2-carbaldehyde
1369160-12-26,7-Dihydro-5H-pyrrolo[1,2-a]imidazole-6-carboxylic acid
13720-94-0ethyl 4-chloroquinoline-3-carboxylate
1373223-06-3(7-Methoxy-1-methyl-1H-indazol-5-yl)-methanol
1373223-18-7(2-Chloro-6-trifluoromethyl-pyridin-4-yl)-carbamic acid tert-butyl ester
13745-27-2(1-Methyl-1H-benzoimidazol-2-yl)-pyridin-4-yl-methanone
13745-30-7C-(1-Methyl-1H-benzoimidazol-2-yl)-C-pyridin-4-yl-methylamine
13745-30-7C-(1-Methyl-1H-benzoimidazol-2-yl)-C-pyridin-4-yl-methylamine
1374657-44-91-Hydroxymethyl-cyclobutanecarbonitrile
1375472-17-52,5-Dimethyl-cyclopentylamine hydrochloride
138163-12-94-Methylene-piperidine-1-carboxylic acid benzyl ester
138175-25-4(R)-2-Methyl-1-pyridin-2-yl-propylamine
13877-55-91,6-Dihydro-pyrazolo[4,3-d]pyrimidin-7-one
138786-65-9Methyl 2-bromomethyl-5-fluoro-benzoate
138969-57-0(2,3-Dihydro-1H-indol-2-yl)-methanol
139458-29-0C-(5-Methyl-isoxazol-4-yl)-methylamine hydrochloride
14088-84-7N1-(4-Chloro-phenyl)-ethane-1,2-diamine dihydrochloride
140927-13-5benzyl 5-oxo-2-azabicyclo[2.2.1]heptane-2-carboxylate
1410783-77-5(R)-3-Methyl-pyrrolidine-3-carboxylic acid
1414958-33-06-Oxa-3-aza-bicyclo[3.1.1]heptane hydrochloride
1414959-08-24-Phenyl-3-piperidin-4-yl-oxazolidin-2-one
1423-63-81-(5-Bromo-benzo[b]thiophen-3-yl)-ethanone
1427195-04-7C-[4-(1,1-Difluoro-ethyl)-pyrimidin-5-yl]-methylamine
1427195-21-82-Fluoro-5-iodo-4-methyl-benzoic acid methyl ester
1427195-24-16-Methoxy-3-nitro-pyridine-2-carboxylic acid methyl ester
1427195-24-16-Methoxy-3-nitro-pyridine-2-carboxylic acid methyl ester
1427203-52-8tert-butyl (R)-3-(2-methoxy-2-oxoethoxy)pyrrolidine-1-carboxylate
1437790-06-17-Fluoro-[1,5]naphthyridin-4-ol
1439-09-45-Bromo-4-methyl-pyrimidine
144222-23-1(4-Amino-butyl)-methyl-carbamic acid tert-butyl ester
145901-11-71H-Pyrrolo[2,3-b]pyridin-6-ylamine
14736-49-32-[2-(Methoxycarbonyl)phenyl]acetic acid
148136-03-24-[2-(4-Chloro-phenyl)-ethyl]-piperidine hydrochloride
14847-51-92-Bromo-5-methyl-phenol
149353-75-31-Boc-4-(4-carboxy-phenyl)-piperidine
149353-75-31-Boc-4-(4-carboxy-phenyl)-piperidine
149488-78-8(3-Fluoro-pyridin-2-yl)-acetonitrile
149649-58-1Pyrrolidin-2-ylmethyl-carbamic acid tert-butyl ester
15018-66-3Quinazolin-4-ylamine
15224-11-02-Hydroxymethyl-cyclopropanecarboxylic acid ethyl ester
153024-86-35,6,7,8-Tetrahydro-4H-thieno[2,3-c]azepine
153435-96-2Ethyl 4,6-dichloro-3-formyl-1H-indole-2-carboxylate
155058-02-97,8-Dihydro-6H-[1,6]naphthyridin-5-one
156041-33-7cis-5-Hydroxymethyl-cyclohex-2-enol
15889-32-43-Pyridin-2-yl-phenylamine
15889-32-4]3-Pyridin-2-yl-phenylamine
15901-66-3Isothiazole-5-carboxylic acid methyl ester
1601-81-6cis-2-Benzoyl-cyclopropanecarboxylic acid
1601-81-6cis-2-Benzoyl-cyclopropanecarboxylic acid
1601-82-7trans-2-Benzoyl-cyclopropanecarboxylic acid
1601-82-7trans-2-Benzoyl-cyclopropanecarboxylic acid
160809-34-74-Acetyl-piperidine-1-carboxylic acid benzyl ester
1611469-80-71-(3-Bromo-propyl)-4-octyl-benzene
1614-73-9Cyclohept-4-enecarboxylic acid
1639924-58-5(2S,5R)-2,5-dimethylmorpholin
165253-29-23-Bromomethyl-tetrahydro-furan
166526-03-04,6-Dichloro-nicotinonitrile
16778-21-54-Chloro-8-methoxy-quinoline
168038-14-0(R)-2-Methyl-morpholine hydrochloride
168072-81-92-Carboxymethyl-benzoic acid tert-butyl ester
168072-81-92-Carboxymethyl-benzoic acid tert-butyl ester
16858-56-32-Chloro-6-methyl-pyrimidine-4-carbonitrile
16880-11-83-Methoxy-isoxazole-5-carboxylic acid methyl ester
169037-38-11H-Pyrrolo[3,2-c]pyridine-2,3-dione
169789-36-0(5-Methoxy-1H-indazol-3-yl)-methanol
169789-37-15-Methoxy-1H-indazole-3-carbaldehyde
171049-35-7[4,4']Bipiperidinyl-1-carboxylic acid tert-butyl ester
171049-35-7[4,4']Bipiperidinyl-1-carboxylic acid tert-butyl ester
1710-66-3Isothiazol-5-yl-methanol
171663-13-1tert-butyl (3-bromobenzyl)carbamate
171753-74-5(2R,6R)-2,6-Dimethyl-morpholine
17231-51-53-Amino-6-bromo-pyrazine-2-carbonitrile
172733-79-83H-spiro[isobenzofuran-1,4'-piperidin]-3-one hydrochloride
172733-79-83H-spiro[isobenzofuran-1,4'-piperidin]-3-one hydrochloride
17347-32-96-Bromo-benzo[b]thiophene
17347-32-96-Bromo-benzo[b]thiophene
17607-00-04-Oxo-cycloheptanecarboxylic acid methyl ester
177-17-36-Aza-spiro[4.5]decane
177-17-36-Aza-spiro[4.5]decane
177202-83-42-Pyridin-3-yl-phenylamine
177941-16-15-Benzyloxy-1H-indazole-3-carboxylic acid
177941-17-27-Benzyloxy-1H-indazole-3-carboxylic acid
178312-48-6(4,4-Difluoro-cyclohexyl)-methanol
17841-68-8methyl 3-(aminomethyl)benzoate hydrochloride
178984-46-8(4-Chloro-quinolin-7-yl)-dimethyl-amine
17965-71-83-Bromo-[1,5]naphthyridine
17965-71-83-Bromo-[1,5]naphthyridine
17965-73-03-Bromo-[1,6]naphthyridine
17965-74-18-Bromo-[1,6]naphthyridine
17965-74-18-Bromo-[1,6]naphthyridine
17965-75-23,8-Dibromo-[1,6]naphthyridine
17965-78-53-Bromo-[1,8]naphthyridine
17965-78-53-Bromo-[1,8]naphthyridine
17965-78-53-Bromo-[1,8]naphthyridine
179898-81-83,3-Dimethyl-4-oxo-3,4-dihydro-2H-quinoline-1-carboxylic acid tert-butyl ester
179898-87-42,2-Dimethyl-4-oxo-3,4-dihydro-2H-quinoline-1-carboxylic acid tert-butyl ester
180160-47-85-Chloro-3H-spiro[isobenzofuran-1,4'-piperidin]-3-one 
180163-21-73-(2,6-Dimethyl-phenylamino)-phenol
180623-89-65-Bromo-7-chloro-1H-indole
18085-37-5methyl 1-benzylazetidine-2-carboxylate
180975-66-0cis-1-Boc-2,6-dimethyl-piperazine
181308-57-6trans-(4-Formyl-cyclohexyl)-carbamic acid tert-butyl ester
18436-71-04-Chloro-6-methyl-quinoline
184368-70-5trans-2,6-Dimethyl-4-oxo-piperidine-1-carboxylic acid tert-butyl ester
185315-52-0(3-Chloro-pyridin-2-yl)-acetonitrile
185526-66-31'-Boc-2,3-dihydrospiro[indene-1,4'-piperidine]-3-acetic acid
185527-11-1tert-Butyl 3-amino-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxylate
185692-51-72-Benzyl-hexahydro-cyclopenta[c]pyrrol-4-one
186201-60-52-Benzyl-octahydro-cyclopenta[c]pyrrol-4-ylamine
188554-13-42-Hydroxy-pyridine-4-carbaldehyde
18977-45-2Cyclopropylmethyl-methyl-amine
19036-43-23-Amino-2,2-dimethyl-propionic acid
19075-58-26-Bromo-benzo[b]thiophene-2-carboxylic acid
194804-80-32,4-Difluoro-3-hydroxy-benzoic acid methyl ester
19524-10-84-Chloro-3,5-dimethyl-pyridine
197516-58-82-Bromomethyl-6-fluoro-benzoic acid methyl ester
1975-54-85-Cyano-2-methyl-benzoic acid
198281-55-93-(4-Methyl-piperazin-1-ylmethyl)-aniline
198401-76-2(4-Trifluoromethyl-pyridin-3-yl)-methanol
198835-02-8exo-6-Hydroxy-2-aza-bicyclo[2.2.1]heptane-2-carboxylic acid tert-butyl ester
198835-06-22-Boc-5-oxo-2-aza-bicyclo[2.2.1]heptane
19983-42-76-Nitro-benzo[b]thiophene-2-carboxylic acid
201227-38-55-Bromo-1H-indazole-3-carbaldehyde
201227-38-55-Bromo-1H-indazole-3-carbaldehyde
202522-04-13-Ethyl-4-formyl-benzonitrile
20493-60-15-Bromo-3-methyl-isothiazole
205059-32-11-Ethyl-[4,4']bipiperidinyl
205444-22-02-Chloro-4-iodo-6-trifluoromethyl-pyridine
20567-67-36-Methyl-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazine
20662-83-34,5-Dimethyl-oxazole
207405-62-75-Amino-2-aza-bicyclo[2.2.1]heptane-2-carboxylic acid tert-butyl ester
207502-65-6N-[[4-[trifluoromethyl]-3-pyridinyl]carbonyl]-glycine
209256-42-82,3-Dihydro-benzofuran-4-carbaldehyde
209256-64-4Chroman-5-carboxylic acid
212184-86-65,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
213118-56-0(2-Amino-4-methoxy-phenyl)-carbamic acid tert-butyl ester
21609-70-13,4-Dihydro-2H-benzo[b]thiepin-5-one
2183-66-62-(Methylthio)pyrimidin-4-amine
219862-14-3(1,2,3,4-Tetrahydro-quinolin-3-yl)-carbamic acid tert-butyl ester
2205-98-3Spiro[2.5]octan-4-one
22061-78-52-Bromo-3-methyl-phenol
220780-57-43-Bromo-isoxazole-5-carbaldehyde
221024-31-35-Bromo-7-chloro-2,3-dihydro-1H-indole
2213-66-35-TERT-BUTYL-3-METHYLCATECHOL
22190-35-86-Bromo-1,2,3,4-tetrahydro-quinoline
222978-03-24-Bromomethyl-2-fluoro-benzonitrile
222978-03-24-Bromomethyl-2-fluoro-benzonitrile
22364-29-02-Bromo-4,5-dimethyl-phenylamine
2288-74-63,5-Dichloro-4-methoxy-pyridazine
229621-74-3Methyl-(2-p-tolyl-ethyl)-amine
23443-25-66-Methoxy-[1,5]naphthyridin-4-ol
238433-75-5(2-Phenyl-oxazol-5-yl)-methanol
239074-29-4tert-butyl ((1r,4r)-4-(hydroxymethyl)cyclohexyl)carbamate
2402-97-33-Bromo-pyridine 1-oxide
24303-64-84-Methoxy-but-2-ynoic acid
24334-19-81H-Pyrrolo[2,3-c]pyridine-2-carboxylic acid ethyl ester
24334-20-11H-Pyrrolo[2,3-c]pyridine-2-carboxylic acid
24334-20-11H-Pyrrolo[2,3-c]pyridine-2-carboxylic acid
24340-77-04-Bromo-isothiazole
24340-77-04-Bromo-isothiazole
2450-08-0Pyrimidine-4-carboxylic acid methyl ester
2469-99-03-Oxo-butyronitrile
249889-68-78-chloro-2-methoxy-1,5-naphthyridine
249889-68-78-Chloro-2-methoxy-[1,5]naphthyridine
249889-69-86-Methoxy-[1,5]naphthyridin-4-ylamine
25039-53-64-chloroisothiazole
251635-21-94-Cyclopropyl-3-oxo-butyric acid methyl ester
252004-42-51-Bromo-2,5-difluoro-4-methyl-benzene
2523-56-0cis-4-Methyl-cyclohexylamine
252372-09-11-Furan-3-yl-ethylamine
253801-04-61H-Indazole-5-carbaldehyde
255882-72-51-Boc-azetidine-2-carboxylic acid methyl ester
25712-60-11-Methyl-pyrrolidine-3-carboxylic acid 
25864-34-06-Methyl-3,5-dinitro-pyridin-2-ylamine
264254-04-8[1,4]Dioxan-2-ylmethyl-methyl-amine
264602-74-67-Bromo-4,4-dimethyl-1,2,3,4-tetrahydro-isoquinoline
265108-25-6cis-(4-Hydroxy-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
265324-26-32-Cyclopropyl-pyrimidin-4-ylamine
26673-30-35-Chloro-tetral-1-on
267413-25-2C-(1H-Indazol-5-yl)-methylamine
271-34-11H-pyrrolo[3,2-c]pyridine
273-70-1Thiazolo[5,4-c]pyridine
2746-23-83-Chloromethyl-thiophene
276252-73-4(2S,6S)-2,6-Dimethyl-morpholine
27684-84-05-Bromo-2-nitro-phenol
27772-90-34,5,6,7-Tetrahydro-benzo[d]isoxazol-3-ol
27772-90-34,5,6,7-Tetrahydro-benzo[d]isoxazol-3-ol
27784-69-6Cyclobutylidene-acetonitrile
2806-84-03-Methoxy-propionaldehyde
2806-84-03-Methoxy-propionaldehyde
28114-87-628114-87-6
2812-32-0N,N-Dimethyl-L-valine
281235-04-94-Piperidin-4-yl-benzoic acid methyl ester
28593-08-0[1,6]Naphthyridin-4-ylamine
28593-08-0[1,6]Naphthyridin-4-ylamine
286390-20-33-Oxa-6-aza-bicyclo[3.1.1]heptane
288-16-4Isothiazole
2906-60-74,4'-dithiodibutyric acid
29241-62-15-Bromo-6-chloro-nicotinic acid
29509-06-64-Methyl-3-oxo-pentanenitrile
29528-30-12-Pyridin-2-yl-phenylamine
29681-42-34-Bromo-pyridine-2-carboxylic acid methyl ester
29908-11-0[1,4]Dioxan-2-yl-methanol
30084-91-4Indan-5-carbaldehyde
30273-40-64-Bromo-2,5-dimethyl-phenylamine
30532-36-63-Pyridin-4-yl-propylamine
30721-88-16-Dimethylamino-pyridine-2-carboxylic acid
30830-27-43-Benzyloxy-cyclobutanone
3095-48-54-Amino-3,5-dimethyl-benzoic acid methyl ester
319474-35-63-Formyl-1H-indazole-6-carboxylic acid
323592-68-3(6S)-Methyl-piperazin-2-one
32385-74-32-(1H-Pyrazol-3-yl)-ethanol
324-32-32-Methyl-7-trifluoromethyl-quinoline
3261-62-94-Methylphenethylamine 
327046-67-33-Amino-4-tert-butoxycarbonylamino-benzoic acid methyl ester
32804-66-3Methyl but-3-ynoate
33036-67-8ethyl oxazole-2-carboxylate
33036-67-8Ethyl oxazole-2-carboxylate
33042-66-9Spiro[indene-1,4'-piperidine]
3308-02-92-Phenyl-pyridin-3-ol
33483-66-8(1s,4s)-4-methylcyclohexan-1-amine hydrochloride
33537-18-7Cyclopentyl-oxo-acetic acid ethyl ester
335428-62-15-Bromo-1-methyl-2,3-dihydro-1H-isoindole
34084-88-36-Nitro-benzo[b]thiophene-2-carboxylic acid methyl ester
341-24-27-Fluoro-1H-indazole
3413-28-34-(4-Fluoro-phenoxy)-piperidine
34486-22-12-Chloro-6-trifluoromethyl-pyridin-4-ylamine
346599-63-14-Chloro-5H-pyrrolo[2,3-d]pyrimidin-6(7H)-one
3469-63-45-Metoxy-1H-pyrrolo[2,3-c]pyridine-2-carboxylic acid ethyl ester
351003-02-65-Bromo-2-methyl-nicotinic acid
351003-02-65-Bromo-2-methyl-nicotinic acid
351456-45-65-Chloro-3-iodo-1H-indazole
3528-45-82-(4-Methoxy-benzyl)-2H-pyrazol-3-ylamine
354587-75-04-Trifluoromethyl-thiazole-2-carbaldehyde
361389-86-83-Methyl-indan-1-ylamine
362670-09-5(2-Amino-5-methoxy-phenyl)-carbamic acid tert-butyl ester
36635-66-2[1-Phenyl-1-tosyl]methyl isocyanide
36856-91-42-Bromo-quinoxaline
36982-56-6(2-Bromo-ethyl)-cyclopropane
37444-46-5Pyridazin-3-yl-methanol
37466-89-02,3-Diaminoanisol
37949-03-45,6,8,9-Tetrahydro-benzocyclohepten-7-one
37949-03-45,6,8,9-Tetrahydro-benzocyclohepten-7-one
380-41-62,2-Difluoro-3-hydroxy-propionic acid ethyl ester
38076-78-72-Amino-5-methylnicotinonitrile
38275-55-75-Fluoro-pyrimidine-2-carbonitrile
38275-61-55-Chloro-pyrimidine-2-carboxylic acid
38778-05-14-Phenoxy-benzenethiol
3912-37-6Isothiazole-4-carbonitrile
391680-79-85,6-Dihydroxy-2-thiophen-2-yl-pyrimidine-4-carboxylic acid
393553-44-11H-Indazole-3,4-dicarboxylic acid 4-methyl ester
3951-89-17-Bromo-1,2,3,4-tetrahydro-benzo[b]azepin-5-one
396133-32-71,2,2-trimethylpiperazine
396730-55-51,2,3,6-Tetrahydro-pyridin-3-ol hydrochloride
3973-62-43-Phenyl-piperidine
39889-94-62-Methyl-pyrimidin-5-ylamine
39959-51-82-Iodo-benzylamine
40018-10-83-Oxo-3-(2-trifluoromethyl-phenyl)-propionitrile
402-17-52-Nitro-5-trifluoromethyl-phenol
40397-90-81-Chloro-3-isocyanato-2-methyl-benzene
40605-42-33-Chloro-but-2-en-1-ol
40990-53-24-Methoxy-1H-indole-6-carboxylic acid
41110-28-53-Methyl-pyrazine-2-carboxylic acid
41172-57-0Methyl 5-methyl-1,3-oxazole-4-carboxylate
4133-35-16-Bromo-3,4-dihydro-1H-naphthalen-2-one
4160-75-21-Cyclopropyl-propan-2-one
420786-53-4(4-Hydroxy-phenyl)-piperidin-4-yl-methanone
42450-36-21-Isobutyl-piperidin-4-ylamine
426266-77-5C-(5-Chloro-pyrimidin-2-yl)-methylamine
42858-39-9Ethyl bicyclo[2.2.2]oct-5-ene-2-carboxylate
4295-04-94-Chloro-6-methoxy-quinoline
4315-14-44,5-Dimethyl-2-nitro-benzoic acid
439811-37-71-Boc-4-(4-bromo-benzoyl)-piperidine
4487-50-74-Nitro-pyridin-2-ylamine
4576-90-3Isothiazole-3-carboxylic acid
4664-00-0Pyrrolo[3,4-b]pyridine-5,7-dione
473416-12-5methyl 1H-indazole-5-carboxylate
473416-12-5Methyl 1H-indazole-5-carboxylate
474656-47-84-(1H-Pyrazol-3-yl)-morpholine
478375-40-53-Bromo-5-methyl-benzoic acid methyl ester
48108-93-62-(2-Amino-ethyl)-phenylamine
4919-40-84-Amino-3,5-dimethyl-benzoic acid 
4934-99-03-Hydroxy-cyclobutanecarboxylic acid methyl ester
4934-99-03-Hydroxy-cyclobutanecarboxylic acid methyl ester
5025-59-22-Iodo-6-methoxy-benzaldehyde
50386-65-7Chroman-5-ylamine
50476-72-74-Chloro-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl ester
50564-59-53-Chloro-piperidine 
50593-68-53-chloro-6-nitro-1H-indazole
50675-23-5(2,2-Dimethyl-tetrahydro-pyran-4-yl)-methanol
51015-29-3 6-Methyl-1-tetralone
51532-07-12-Bromo-[1,5]naphthyridine
51532-07-12-Bromo-[1,5]naphthyridine
518047-31-95,6-Dihydroxy-pyrimidine-4-carboxylic acid methyl ester
5190-68-14-Chloro-quinazoline
51907-18-75,6-Dihydro-[2]pyrindin-7-one
51907-18-75,6-Dihydro-[2]pyrindin-7-one
521979-97-5(R)-4-Phenyl-3-piperidin-4-yl-oxazolidin-2-one hydrochloride
521979-98-6(S)-4-Phenyl-3-piperidin-4-yl-oxazolidin-2-one hydrochloride
52320-59-95-Ethyl-isoxazole-3-carboxylic acid
52378-64-0(3-Bromo-pyridin-2-yl)-methanol
52378-64-0(3-Bromo-pyridin-2-yl)-methanol
52412-10-95,6-Dihydroxy-pyrimidine-4-carboxylic acid
5242-57-9Isothiazole-5-carbaldehyde
52516-20-8[2-(3-Chloro-phenyl)-ethyl]-methyl-amine
5335-05-7Chloromethyl benzoate
53821-72-02-Nitro-malonaldehyde sodium salt monohydrate
54015-04-21-(p-tolyl)guanidine hydrochloride
54237-53-56-Bromo-pyrazin-2-ylamine
54752-50-07-Trifluoromethyl-3,4-dihydro-2H-naphthalen-1-one
54752-50-07-Trifluoromethyl-3,4-dihydro-2H-naphthalen-1-one
55052-27-26-Chloro-1H-pyrrolo[2,3-b]pyridine
55314-30-22,4-Dimethyl-nicotinic acid
55698-67-48-Hydroxy-quinoline-4-carboxylic acid
55755-17-4/125470-40-63-Methylphenethylamine
56105-19-2Cyclopropyl-acetaldehyde
5638-60-8[1,4]Oxazepane
5649-36-52,6-Dimethyl-1H-indole
5649-36-52,6-Dimethyl-1H-indole
56621-98-85-Amino-pyrimidine-2-carboxylic acid
56633-75-1(S)-Pyrrolidin-2-yl-acetic acid
56700-66-4tert-butyl cyclobutylcarbamate
56723-86-53-Methoxy-5-(trifluoromethyl)benzalderhyde
5709-98-8(R)-(+)-Cyclohex-3-enecarboxylic acid
57174-62-61-Aza-spiro[3.4]octane
57260-70-5tert-butyl 4-benzylpiperazine-1-carboxylate
5763-55-32-Cyclopentyl-ethylamine
5780-66-5Pyrazine-2-carbaldehyde
5780-66-5Pyrazine-2-carbaldehyde
58088-72-52-Methyl-1-pyridin-2-yl-propylamine
586330-18-9tert-butyl 3-iodo-6-nitro-1H-indazole-1-carboxylate
59128-15-3(6-Bromo-imidazo[1,2-a]pyridin-2-yl)-acetic acid
591-55-9Pyrimidin-5-ylamine
59193-77-03-Amino-2,2-dimethyl-propionic acid ethyl ester
59215-41-74-Piperazin-1-yl-quinazoline
5964-97-4N-(4-Chloro-phenyl)-guanidine hydrochloride
59660-30-9(4-Methyl-4H-[1,2,4]triazol-3-yl)-methanol
60170-83-4Pyridazine-3-carbaldehyde
60307-26-8(R)-2-(1-Methyl-pyrrolidin-2-yl)-ethanol
604010-24-42,6-Dimethyl-4-oxo-piperidine-1-carboxylic acid tert-butyl ester
611226-36-94-Hydroxy-pyridine-2-carboxylic acid methylamide
612499-04-4C-(5-Bromo-thiophen-2-yl)-methylamine
61266-70-4oxetan-2-ylmethanol
6127-17-96-Chloro-2-methyl-1H-indole
612833-66-61-Benzyloxy-4-bromo-2-iodo-benzene
61319-97-94-Chloro-2-methyl-[1,5]naphthyridine
61350-65-0(R)-Pyrrolidin-2-yl-acetic acid
615568-24-62,3-Dihydro-[1,4]dioxino[2,3-b]pyridine-6-carbaldehyde
61810-78-4(S)-2-(1-Methyl-pyrrolidin-2-yl)-ethanol
62150-46-34-Bromo-pyridine-2-carboxylic acid amide
62222-38-25,6-Dihydroxy-2-phenyl-pyrimidine-4-carboxylic acid
62482-32-05-Chloro-quinoline-4-carboxylic acid
627527-23-51-Bromo-3-methoxy-5-trifluoromethyl-benzene
6281-32-9Quinolin-4-yl-methanol
63126-47-6(S)-2-Methoxymethyl-pyrrolidine
6314-43-8C-Benzo[b]thiophen-2-yl-methylamine 
63200-54-42,4-Dichloro-5H-pyrrolo[3,2-d]pyrimidine
63910-32-73,4-Dichloro-5-methoxy-pyridazine
63927-22-08-Bromo-isoquinoline
64132-13-4(1H-Indazol-3-yl)-methanol
64145-51-33-Phenyl-cyclopentanone
643069-40-38-Bromo-5-methoxy-1H-quinolin-4-one
643069-46-94-Bromo-5-methoxy-quinoline
64330-46-71-Benzyl-1,5-dihydro-pyrrol-2-one
64330-46-71-Benzyl-1,5-dihydro-pyrrol-2-one
64403-25-43-Methyl-4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridine
650141-20-12,6-Dimethyl-pyridine-3-carbaldehyde
650141-20-12,6-Dimethyl-pyridine-3-carbaldehyde
651059-70-0methyl 2-methyloxazole-5-carboxylate
651059-70-02-Methyl-oxazole-5-carboxylic acid methyl ester
65326-33-21-(2-Amino-pyridin-3-yl)-ethanone
65340-74-17-Bromo-quinolin-4-ylamine
65783-21-3N-(4-Fluoro-phenyl)-guanidine
66500-55-81,4-Dioxa-spiro[4.5]decane-8-carboxylic acid
6684-39-56-Chloro-pyridine-3-sulfonyl chloride
669050-69-51H-Indazole-6-carbaldehyde
67120-38-16-Chloro-indan-1-ylamine
67120-39-25-Chloro-indan-1-ylamine
67221-50-54-Amino-1H-pyrazole-3-carboxylic acid amide
672948-03-7Oxazole-2-carboxylic acid
675185-27-0(R)-1-Boc-2-acetyl-pyrrolidine
677304-83-5Benzothiazole-7-carboxylic acid
677304-83-5Benzothiazole-7-carboxylic acid
6786-30-73,4-Dihydro-2H-benzo[b]oxepin-5-one
679433-91-15-Bromo-8-methoxy-isoquinoline
68776-58-9Isoxazole-4-carbonitrile
68776-62-5Pyridazine-4-carbonitrile
69135-98-4trans-2,6-Dimethyl-4-oxo-piperidine
697299-86-8C-(4-Bromo-thiazol-2-yl)-methylamine
698-24-86-Methyl-1H-indazole
698-26-05-Chloro-1H-indazole
70315-70-73-iodo-6-nitro-1H-indazole
71278-11-04-Amino-1-pyridin-3-yl-butan-1-one
713-09-7Ethyl 1H-indazole-6-carboxylate
71322-99-12-Methyl-piperidin-4-one
717134-47-9Methyl 6-chloro-1H-indazole-3-carboxylate
718595-36-92-Bromo-1-(4-chloro-pyridin-2-yl)-ethanone
72754-06-42-Bromo-[1,6]naphthyridine
73870-28-74-Bromomethyl-quinoline hydrobromide
74213-24-41,1-Dibromoformaldoxime
74417-44-01-Bromomethyl-isoquinoline
749256-90-42-Chloro-4-methyl-6-trifluoromethyl-pyridine
75366-10-81-Bromo-2-bromomethyl-3-methyl-benzene
766557-40-85,6-Dihydroxy-2-pyridin-2-yl-pyrimidine-4-carboxylic acid
767-70-47-Bromo-benzothiazole
7681-84-7Tetrahydro-furan-2-carbaldehyde
77029-01-76-Methoxy-naphthalene-1-carbonitrile
77156-85-54-Chloro-7-methoxy-quinoline-3-carboxylic acid ethyl ester
771580-70-2C-(4-Trifluoromethyl-pyridin-3-yl)-methylamine
771580-70-2C-(4-Trifluoromethyl-pyridin-3-yl)-methylamine
77168-85-55-Chloro-6-methyl-pyrazine-2-carboxylic acid methyl ester
774531-95-25,8-Dihydro-6H-quinolin-7-one
79069-50-4(S)-(1-Methyl-2-oxo-ethyl)-carbamic acid tert-butyl ester
79578-98-61-Methyl-1H-imidazol-4-ylamine
796090-23-82-Chloro-6-trifluoromethyl-isonicotinic acid
796090-23-82-chloro-6-(trifluoromethyl)isonicotinic acid
800401-67-65-Chloro-1H-pyrrolo[2,3-c]pyridine-2-carboxylic acid ethyl ester
809273-70-9(4-Oxo-cyclohexylmethyl)-carbamic acid tert-butyl ester
81445-44-5(S)-2-Benzyloxy-propionaldehyde
822-54-8Isothiazole-4-carbaldehyde
82261-42-54-Pyridin-3-yl-phenylamine
822-82-2Isothiazole-4-carboxylic acid
822-82-2Isothiazole-4-carboxylic acid
82353-55-7(R)-(1-Methyl-2-oxo-ethyl)-carbamic acid benzyl ester
82353-56-8(R)-(1-Methyl-2-oxo-ethyl)-carbamic acid tert-butyl ester
82357-92-4isothiazol-5-amine hydrochloride
82668-50-6(1H-Pyrazol-3-yl)-acetic acid ethyl ester
82683-51-0spiro[4.5]decane-7,9-dione
83101-12-64-(3-Hydroxy-propyl)-benzonitrile
84025-81-0(R)-2-Methoxymethyl-pyrrolidine
84200-06-63-Pyridin-4-yl-propionitrile
846036-96-2(4-Amino-6-chloro-pyridin-3-yl)-methanol
847801-92-72-Chloro-1H-pyrrolo[2,3-c]pyridine-3-carbaldehyde
849475-89-45,6-Dihydroxy-2-pyridin-2-yl-pyrimidine-4-carboxylic acid methyl ester
862129-72-44-Methanesulfonyl-cyclohexanone
86499-35-63-Amino-1,3,4,5-tetrahydro-benzo[b]azepin-2-one
865887-11-26-Benzyloxy-1H-indazole-3-carboxylic acid
865887-17-8Ethyl 5-benzyloxy-1H-indazole-3-carboxylate
866782-59-48-Fluoro-3-iodo-quinoline
867130-58-36-Oxo-1,6-Dihydropyridazine-4-Carboxylic Acid
870632-89-6trans-(4-Hydroxy-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
870632-91-0(3S,4S)-(4-Hydroxy-pyrrolidin-3-yl)-carbamic acid tert-butyl ester
87121-89-93-Oxo-cyclobutanecarboxylic acid ethyl ester
871507-79-82,8-Dibromo-quinoline
872018-40-16-Bromo-3-methyl-2H-isoquinolin-1-one
873924-08-49-Oxo-3-aza-spiro[5.5]undecane-3-carboxylic acid tert-butyl ester
873924-08-49-Oxo-3-aza-spiro[5.5]undecane-3-carboxylic acid tert-butyl ester
875755-36-57-chloro-1,2,3,4-tetrahydronaphthalen-1-amine
875781-17-25-Bromo-1H-pyrazolo[3,4-b]pyridine
87673-88-91-Methyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine
87673-88-91-Methyl-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine
878158-18-0methyl 5,6-dihydroxy-2-methylpyrimidine-4-carboxylate
878649-59-32-Benzyl-5,6-dihydroxy-pyrimidine-4-carboxylic acid
879883-54-24-Piperidin-4-ylmethyl-piperidine-1-carboxylic acid tert-butyl ester
879883-60-01-Ethyl-4-piperidin-4-ylmethyl-piperidine
884004-48-22-amino-4-chloronicotinaldehyde
885223-72-35-Bromo-6-methyl-1H-indazole
885266-91-11-(2-Amino-pyridin-4-yl)-ethanol
885269-76-1Ethyl 3-(1H-indazol-3-yl)-3-oxo-propionate
885269-93-2(4-Acetyl-2-bromo-phenyl)-carbamic acid tert-butyl ester
885271-15-86-bromo-8-methoxy-2H-chromene-3-carbaldehyde
885271-72-76-bromo-1H-indazole-3-carbaldehyde
885272-94-6Ethyl 6-bromo-1H-indazole-3-carboxylate
885273-36-92-Methyl-4,5,6,7-tetrahydro-oxazolo[4,5-c]pyridine
885273-50-7C-[3-(3-Chloro-phenyl)-isoxazol-5-yl]-methylamine
885273-54-13-m-Tolyl-isoxazole-5-carbaldehyde
885273-61-0Ethyl 5-bromo-3-(2-carboxy-vinyl)-1H-indole-2-carboxylate
885274-77-1Piperidine-4-carboxylic acid 4-chloro-benzylamide
885275-59-26-Chloro-3-iodo-imidazo[1,2-a]pyridine
885276-99-32-Amino-6-methyl-pyridine-3-carbaldehyde
885276-99-32-Amino-6-methyl-pyridine-3-carbaldehyde
885277-01-02-Chloro-4-(2,2,2-trifluoro-ethoxy)-pyridine
885278-10-42-Isopropoxy-pyridine-3-carbaldehyde
885278-33-1           6-fluoro-1H-indazole-3-carbonitrile
885278-42-2Methyl 6-bromo-1H-indazole-3-carboxylate
885278-62-6Methyl 5-benzyloxy-1H-indazole-3-carboxylate
885278-65-9Methyl 7-benzyloxy-1H-indazole-3-carboxylate
885279-23-2Ethyl 6-chloro-1H-indazole-3-carboxylate
885279-78-73,5-Dibromo-2,4-dihydroxybenzoic acid methyl ester
885280-91-12-(5-Methoxy-pyridin-2-yl)-phenylamine
885281-16-33-Phenyl-5,6,7,8-tetrahydro-imidazo[1,2-a]pyrazine
88536-11-24-Propoxy-piperidine
885520-35-44-Bromo-6-fluoro-1H-indazole
885520-35-44-Bromo-6-fluoro-1H-indazole
886364-28-94-N-Boc-8-fluoro-1,2,3,5-tetrahydro-benzo[e][1,4]diazepine
886371-24-0C-(3-Trifluoromethyl-pyridin-2-yl)-methylamine
886779-69-7tert-butyl 3-(trifluoromethyl)piperazine-1-carboxylate
887579-62-65-Cyano-nicotinic acid
88982-87-04-Chloro-isothiazole-5-carboxylic acid
891183-50-9(S)-4,4-Dimethyl-pyrrolidine-2-carboxylic acid
891782-63-15-Boc-amino-pyrazine-2-carboxylic acid
89315-56-05,7-dichloro-1,2,3,4-tetrahydroisoquinoline
893411-52-4Spiro[2.5]octane-5,7-dione
89446-67-34-Bromo-7-trifluoromethyl-quinoline
894779-32-97-Methoxy-1-methyl-1H-indazole-5-carboxylic acid ethyl ester
89581-38-45-Bromo-pyrimidine-2-carboxylic acid methyl ester
89793-12-4Ethyl 2-chloro-pyrimidine-5-carboxylate
89892-95-53-Bromomethyl-cyclobutanecarboxylic acid methyl ester
89892-95-53-Bromomethyl-cyclobutanecarboxylic acid methyl ester
89942-70-12-Methyl-pyridine-3,5-dicarboxylic acid
899900-52-8N,N-Dimethyl-D-valine
90001-34-64-Bromo-[1,5]naphthyridine
90109-74-35,6-Dihydroxy-2-methyl-pyrimidine-4-carboxylic acid
90348-29-15-Nitro-1H-indazole-3-carbonitrile
90417-53-15-Methoxy-1H-indazole-3-carboxylic acid
908334-04-34-Bromo-indan-1-one 1,2-ethanediol ketal
90874-56-92,5-Dimethyl-2,3-dihydro-1H-indole
909717-95-9ethyl 4-methoxypyrazolo[1,5-a]pyridine-3-carboxylate
911389-21-48-Chloro-2-methyl-[1,5]naphthyridine
914225-72-24-tert-Butyl-5-chloro-2-hydroxy-benzaldehyde
916056-76-35-Amino-pyrimidine-2-carboxylic acid ethyl ester
916902-55-1(1H-Indazol-6-yl)-methanol
918644-73-29-Hydroxy-3-aza-spiro[5.5]undecane-3-carboxylic acid tert-butyl ester
918644-73-29-Hydroxy-3-aza-spiro[5.5]undecane-3-carboxylic acid tert-butyl ester
91973-39-6(2-Amino-phenyl)-pyridin-4-yl-methanone
92385-37-05-Chloro-quinolin-4-ylamine
92635-33-11H-Pyrrolo[2,3-c]pyridine-2,3-dione
930-42-74-Bromo-3-methyl-isothiazole
93074-72-74-Amino-quinoline-3-carboxylic acid ethyl ester
934-59-85-nitropyridin-3-amine
935466-69-66-Amino-4-chloro-7-azaindole
935466-69-66-Amino-4-chloro-7-azaindole
936940-63-52-Methyl-2H-[1,2,3]triazol-4-ylamine
938439-54-43-Amino-6-methoxy-pyridine-2-carboxylic acid methyl ester
939793-21-21,7-Diaza-spiro[4.5]decane-7-carboxylic acid tert-butyl ester
944896-64-4imidazo[1,2-a]pyrimidine-6-carboxylic acid
944898-72-0C-(1H-Indazol-4-yl)-methylamine
944899-22-37-Benzyloxy-3-iodo-1H-indazole
944900-19-0imidazo[1,2-a]pyrimidin-6-amine
944904-38-57-Fluoro-3-iodo-1H-indazole
944905-56-02-Pyrrolidin-2-yl-pyrimidine
945953-48-02-Pentyl-6,7-dihydro-5H-benzo[b]thiophen-4-one
95206-97-66-Isopropyl-2-methyl-pyrimidin-4-ylamine
954238-84-7(2-Amino-6-methoxy-phenyl)-carbamic acid tert-butyl ester
954239-25-96-Benzyloxy-1H-indazole-3-carboxylic acid methyl ester
954240-14-32,8-Diaza-spiro[5.5]undecane-2-carboxylic acid tert-butyl ester
954240-84-72-(2-Amino-pyridin-3-yl)-ethanol
954240-93-85,6-Dihydroxy-pyrimidine-4-carboxylic acid amide
954241-01-15,6-Dihydroxy-2-isopropyl-pyrimidine-4-carboxylic acid methyl ester
954241-05-55,6-Dihydroxy-2-isopropyl-pyrimidine-4-carboxylic acid
954241-13-55,6-Dihydroxy-2-isopropyl-pyrimidine-4-carboxylic acid amide
960294-14-81-Boc-1,7-Diaza-spiro[4.5]decane
96037-97-21-Cyclopropyl-4-oxo-cyclohexanecarbonitrile
98437-43-55-Bromo-2,4-dihydroxybenzoic acid methyl ester
99207-32-6(4-Hydroxy-butyl)-methyl-carbamic acid tert-butyl ester
na3-Methyl-6-nitro-2H-isoquinolin-1-one
na4-Isopropyl-oxazole-2-carboxylic acid ethyl ester
na3-(4-Methanesulfonyl-phenyl)-piperidine hydrochloride
na(S)-2-Methyl-1-pyridin-2-yl-propylamine dihydrochloride
na4,4-Dimethyl-pyrrolidine-2-carboxylic acid ethyl ester
na3-(3-Methanesulfonyl-phenyl)-piperidine hydrochloride
none2-Iodo-1-methanesulfonyl-4-methoxy-benzene
7-bromo-2,5-bis(phenylsulfonyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
4-((tert-butoxycarbonyl)amino)cyclopent-2-ene-1-carboxylic acid
2-(trifluoromethyl)piperazine
tert-butyl isoxazol-5-ylcarbamate
methyl (1r,4r)-4-((tert-butoxycarbonyl)amino)cyclohexane-1-carboxylate
9-bromo-5H-indeno[1,2-c]pyridine
4-methoxypyrazolo[1,5-a]pyridine-3-carboxylic acid
7-bromo-2-(phenylsulfonyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
tert-butyl (2-tosyl-2-azaspiro[3.3]heptan-6-yl)carbamate
2-chloro-6-(trifluoromethyl)nicotinamide
(R)-(4,4-dimethylpyrrolidin-2-yl)methanol
9-bromo-2-(phenylsulfonyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
tert-butyl 4-(3-(4-bromophenyl)-3-oxopropanoyl)piperidine-1-carboxylate
ethyl (R)-4,4-dimethylpyrrolidine-2-carboxylate
(S)-(Pyrrolidin-3-yloxy)-acetic acid methyl ester tosylate
benzyl 5-hydroxy-2-azabicyclo[2.2.1]heptane-2-carboxylate
(1s,4s)-N-benzyl-4-methylcyclohexan-1-amine
5-methoxy-2-(methylsulfonyl)benzonitrile
4-amino-4H-pyrazole-3-carboxamide
4-chloro-7-iodoquinoline
tert-butyl (S)-3-(2-methoxy-2-oxoethoxy)pyrrolidine-1-carboxylate
(R)-(Pyrrolidin-3-yloxy)-acetic acid methyl ester tosylate
6-fluoro-1,2,3,4-tetrahydroisoquinoline-1-carboxylic acid
tert-butyl 2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxylate
ethyl 5-nitropyrimidine-2-carboxylate
(4,4-dimethylcyclohexyl)methanediol
ethyl 6,8-dioxospiro[3.5]nonane-5-carboxylate
1-(6-chloro-4-iodo-1H-indazol-1-yl)ethan-1-one
N-methylcyclopropanecarboxamide
1H-pyrazolo[4,3-d]pyrimidin-7-ol
1H-pyrazolo[4,3-d]pyrimidin-7-ol
2-Iodo-1-methanesulfonyl-4-methoxy-benzene
(R)-4,4-Dimethyl-pyrrolidine-2-carboxylic acid ethyl ester
3-Methoxymethyl-cyclobutylamine
8-chloro-1,3,4,5-tetrahydro-2H-benzo[b]azepin-2-one
8-chloro-2,3,4,5-tetrahydro-1H-benzo[b]azepine
6-chloro-1,2,3,4-tetrahydronaphthalen-1-amine
7-chloro-1,3,4,5-tetrahydro-2H-benzo[b]azepin-2-one
7-chloro-2,3,4,5-tetrahydro-1H-benzo[b]azepine
6-chloro-1,3,4,5-tetrahydro-2H-benzo[b]azepin-2-one
6-chloro-2,3,4,5-tetrahydro-1H-benzo[b]azepine

Rucaparib Intermediate 1082040-43-4 , I am very yellow

Until now, most of China supply Rucaparib Intermediate 1082040-43-4 is dark, but my product is yellow.

Little impurity you could see below pic.

EOS Med Chem produce 1082040-43-4 to be China biggest.
1082040-43-4 99%, NMR, MS, COA is OK.
1082040-43-4  Size batch could be 100kg.

COA, MSDS, HPLC MORE THAN 98%, NMR, MS is ok




2017年6月7日星期三

Sugammadex sodium Intermediates, biggest supplier 343306-79-6 53784-84-2

NMR-SUGAMMADEX, 343306-71-8, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

Sugammadex sodium is an agent for reversal of neuromuscular blockade by the agent rocuronium in general anaesthesia. It is the first selective relaxant binding agent (SRBA). Sugammadex is a modified γ-cyclodextrin, with a lipophilic core and a hydrophilic periphery. This gamma cyclodextrin has been modified from its natural state by placing eight carboxyl thio ether groups at the sixth carbon positions. These extensions extend the cavity size allowing greater encapsulation of the rocuronium molecule.

We have 100g in stock, attaching NMR


53784-84-2, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.
, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.




Sugammadex sodium Intermediates, biggest supplier 343306-79-6 , assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

http://www.eosmedchem.com/343306-79-6.html 

Name: Sugammadex sodium 
CAS#: 343306-79-6 (sodium salt) 
Chemical Formula: C72H104Na8O48S8 
Exact Mass: 
Molecular Weight: 2177.9742 

Elemental Analysis: C, 39.71; H, 4.81; Na, 8.44; O, 35.26; S, 11.78

Sugammadex sodium Intermediates: OCTAKIS(6-CHLORO-6-DEOXY)-GAMMA-CYCLODEXTRIN (CAS NO.173094-60-5, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

)
http://www.eosmedchem.com/173094-60-5.html

Sugammadex sodium Intermediates: OCTAKIS(6-BROMO-6-DEOXY)-GAMMA-CYCLODEXTRIN (CAS NO.53784-84-2, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

)
http://www.eosmedchem.com/53784-84-2.html

Sugammadex sodium Intermediates: OCTAKIS(6-IODO-6-DEOXY)-GAMMA-CYCLODEXTRIN (CAS NO.168296-33-1, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

)
http://www.eosmedchem.com/168296-33-1.html

We could supply all of them.


HPLC 99%+, NMR, MS, COA, MSDS is ok.










2017 China CPHI: E1M35
EOS Med Chem, Medchem is Big
執大象,天下往,往而無害,安平泰
網址www.eosmedchem.com 
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住所: Diaozhen Chemical Industrial Park, Jinan City, China
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QQ: 2393923585

Related CAS #: 343306-71-8 (free form)   343306-79-6 (sodium salt)  
Synonym: Org25969; Org-25969; Org 25969; 361LPM2T56; Sugammadex; trade name: Bridion. Sugammadex sodium
IUPAC/Chemical Name: 6A,6B,6C,6D,6E,6F,6G,6H-octakis-S-(2-Carboxyethyl)-6A,6B,6C,6D,6E,6F,6G,6H-octathio-γ-cyclodextrin sodium salt
InChi Key: KMGKABOMYQLLDJ-LHCKBTHCSA-F
InChi Code: InChI=1S/C72H112O48S8.8Na/c73-33(74)1-9-121-17-25-57-41(89)49(97)65(105-25)114-58-26(18-122-10-2-34(75)76)107-67(51(99)43(58)91)116-60-28(20-124-12-4-36(79)80)109-69(53(101)45(60)93)118-62-30(22-126-14-6-38(83)84)111-71(55(103)47(62)95)120-64-32(24-128-16-8-40(87)88)112-72(56(104)48(64)96)119-63-31(23-127-15-7-39(85)86)110-70(54(102)46(63)94)117-61-29(21-125-13-5-37(81)82)108-68(52(100)44(61)92)115-59-27(19-123-11-3-35(77)78)106-66(113-57)50(98)42(59)90;;;;;;;;/h25-32,41-72,89-104H,1-24H2,(H,73,74)(H,75,76)(H,77,78)(H,79,80)(H,81,82)(H,83,84)(H,85,86)(H,87,88);;;;;;;;/q;8*+1/p-8/t25?,26?,27?,28?,29?,30?,31?,32?,41-,42-,43-,44-,45-,46-,47-,48-,49-,50-,51-,52-,53-,54-,55-,56-,57+,58+,59+,60+,61+,62+,63+,64+,65+,66+,67+,68+,69+,70+,71+,72?;;;;;;;;/m0......../s1
SMILES Code: O[C@H]1[C@H](O)[C@H](O[C@@H]2[C@@H](O)[C@H](O)[C@H](O[C@@H]3[C@@H](O)[C@H](O)[C@H](O[C@@H]4[C@@H](O)[C@H](O)[C@H](O[C@@H]5[C@@H](O)[C@H](O)[C@H](O6)C(CSCCC(O[Na])=O)O5)C(CSCCC(O[Na])=O)O4)C(CSCCC(O[Na])=O)O3)C(CSCCC(O[Na])=O)O2)C(CSCCC(O[Na])=O)O[C@@H]1O[C@H]7[C@@H](O)[C@H](O)[C@@H](O[C@H]8[C@@H](O)[C@H](O)[C@@H](O[C@H]9[C@@H](O)[C@H](O)C6OC9CSCCC(O[Na])=O)OC8CSCCC(O[Na])=O)OC7CSCCC(O[Na])=O

1: Takazawa T, Mitsuhata H, Mertes PM. Sugammadex and rocuronium-induced anaphylaxis. J Anesth. 2016 Apr;30(2):290-7. doi: 10.1007/s00540-015-2105-x. Epub 2015 Dec 8. Review. PubMed PMID: 26646837; PubMed Central PMCID: PMC4819478.
2: Abad-Gurumeta A, Ripollés-Melchor J, Casans-Francés R, Espinosa A, Martínez-Hurtado E, Fernández-Pérez C, Ramírez JM, López-Timoneda F, Calvo-Vecino JM; Evidence Anaesthesia Review Group. A systematic review of sugammadex vs neostigmine for reversal of neuromuscular blockade. Anaesthesia. 2015 Dec;70(12):1441-52. doi: 10.1111/anae.13277. Review. PubMed PMID: 26558858.
3: Ledowski T. Sugammadex: what do we know and what do we still need to know? A review of the recent (2013 to 2014) literature. Anaesth Intensive Care. 2015 Jan;43(1):14-22. Review. PubMed PMID: 25579285.
4: Partownavid P, Romito BT, Ching W, Berry AA, Barkulis CT, Nguyen KP, Jahr JS. Sugammadex: A Comprehensive Review of the Published Human Science, Including Renal Studies. Am J Ther. 2015 Jul-Aug;22(4):298-317. doi: 10.1097/MJT.0000000000000103. Review. PubMed PMID: 25299638.
5: Jahr JS, Miller JE, Hiruma J, Emaus K, You M, Meistelman C. Sugammadex: A Scientific Review Including Safety and Efficacy, Update on Regulatory Issues, and Clinical Use in Europe. Am J Ther. 2015 Jul-Aug;22(4):288-97. doi: 10.1097/MJT.0000000000000092. Review. PubMed PMID: 25299637.
6: de Boer HD, Shields MO, Booij LH. Reversal of neuromuscular blockade with sugammadex in patients with myasthenia gravis: a case series of 21 patients and review of the literature. Eur J Anaesthesiol. 2014 Dec;31(12):715-21. doi: 10.1097/EJA.0000000000000153. Review. PubMed PMID: 25192270.
7: Tsur A, Kalansky A. Hypersensitivity associated with sugammadex administration: a systematic review. Anaesthesia. 2014 Nov;69(11):1251-7. doi: 10.1111/anae.12736. Epub 2014 May 22. Review. PubMed PMID: 24848211.
8: Luxen J, Trentzsch H, Urban B. [Rocuronium and sugammadex in emergency medicine: requirements of a muscle relaxant for rapid sequence induction]. Anaesthesist. 2014 Apr;63(4):331-7. doi: 10.1007/s00101-014-2303-1. Review. German. PubMed PMID: 24595442.
9: Fuchs-Buder T, Meistelman C, Raft J. Sugammadex: clinical development and practical use. Korean J Anesthesiol. 2013 Dec;65(6):495-500. doi: 10.4097/kjae.2013.65.6.495. Epub 2013 Dec 26. Review. PubMed PMID: 24427454; PubMed Central PMCID: PMC3888841.
10: Dubois PE, Mulier JP. A review of the interest of sugammadex for deep neuromuscular blockade management in Belgium. Acta Anaesthesiol Belg. 2013;64(2):49-60. Review. PubMed PMID: 24191526.
11: Van Gestel L, Cammu G. Is the effect of sugammadex always rapid in onset? Acta Anaesthesiol Belg. 2013;64(2):41-7. Review. PubMed PMID: 24191525.
12: Schaller SJ, Fink H. Sugammadex as a reversal agent for neuromuscular block: an evidence-based review. Core Evid. 2013;8:57-67. doi: 10.2147/CE.S35675. Epub 2013 Sep 25. Review. PubMed PMID: 24098155; PubMed Central PMCID: PMC3789633.
13: Nag K, Singh DR, Shetti AN, Kumar H, Sivashanmugam T, Parthasarathy S. Sugammadex: A revolutionary drug in neuromuscular pharmacology. Anesth Essays Res. 2013 Sep-Dec;7(3):302-6. doi: 10.4103/0259-1162.123211. Review. PubMed PMID: 25885973; PubMed Central PMCID: PMC4173552.
14: Karalapillai D, Kaufman M, Weinberg L. Sugammadex. Crit Care Resusc. 2013 Mar;15(1):57-62. Review. PubMed PMID: 23432503.
15: Øberg E, Claudius C. [Possible clinical potential in reverting muscular block with sugammadex in anaesthesia and surgery]. Ugeskr Laeger. 2013 Feb 11;175(7):428-32. Review. Danish. PubMed PMID: 23402253.
16: Della Rocca G, Di Marco P, Beretta L, De Gaudio AR, Ori C, Mastronardi P. Do we need to use sugammadex at the end of a general anesthesia to reverse the action of neuromuscular bloking agents? Position Paper on Sugammadex use. Minerva Anestesiol. 2013 Jun;79(6):661-6. Epub 2012 Nov 29. Review. PubMed PMID: 23192221.
17: Stair C, Fernandez-Bustamante A. Sugammadex, the first selective relaxant binding agent for neuromuscular block reversal. Drugs Today (Barc). 2012 Jun;48(6):405-13. doi: 10.1358/dot.2012.48.6.1813474. Review. PubMed PMID: 22745926.
18: Baldo BA, McDonnell NJ, Pham NH. The cyclodextrin sugammadex and anaphylaxis to rocuronium: is rocuronium still potentially allergenic in the inclusion complex form? Mini Rev Med Chem. 2012 Jul;12(8):701-12. Review. PubMed PMID: 22512555.
19: Fuchs-Buder T, Meistelman C, Schreiber JU. Is sugammadex economically viable for routine use. Curr Opin Anaesthesiol. 2012 Apr;25(2):217-20. doi: 10.1097/ACO.0b013e32834f012d. Review. PubMed PMID: 22157200.
20: Baldo BA, McDonnell NJ, Pham NH. Drug-specific cyclodextrins with emphasis on sugammadex, the neuromuscular blocker rocuronium and perioperative anaphylaxis: implications for drug allergy. Clin Exp Allergy. 2011 Dec;41(12):1663-78. doi: 10.1111/j.1365-2222.2011.03805.x. Epub 2011 Jul 7. Review. PubMed PMID: 21732999.

2017年6月6日星期二

Ozanimod 1306760-87-1 biggest supplier

Ozanimod Intermediates, biggest supplier.

HPLC 99%+, NMR, MS, is ok
R 1306763-30-3, TERT-BUTYL N-[(1R)-4-CYANO-2,3-DIHYDRO-1H-INDEN-1-YL]CARBAMATE, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.

S 1306763-31-4, (S)-tert-butyl (4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate, assay 99% in GMP plant, C-GMP standard, now COA, NMR, HPLC, MS is ok.


We could produced it in GMP plant, all document is ready to you.

Batch size, 1-5kg.

NMR, HPLC 99, MS, COA, MSDS is ok.

We could produced it in GMP plant, all document is ready to you.

Batch size, 1-5kg.

NMR, HPLC 99, MS, COA, MSDS is ok.






2017年6月4日星期日

World Biggest GMP supplier: Crisaborole; AN2728, 906673-24-3



Crisaborole; AN2728 906673-24-3 Inter:
1) 2-Bromo-5-hydroxy-benzaldehyde,CAS:2973-80-0,Appearance: white solidHPLC,1H NMR 98%+;
2)4-(4-Bromo-3-formyl-phenoxy)-benzonitrile,CAS: 906673-54-9,Appearance: white solidHPLC,1H NMR 98%+;
3)4-(4-Bromo-3-hydroxymethyl-phenoxy)-benzonitrile,CAS:906673-45-8,Appearance: white solidHPLC,1H NMR 98%+;
4) 4-(4-bromo-3-(1,3-dioxolan-2-yl)phenoxy)benzonitrile,CAS#:1217366-74-9,外观:白色至类白色固体,HPLC,1H NMR 98%+;
1-萘酮-6-位衍生物
5)6-Amino-3,4-dihydro-1(2H)-naphthalenone ;6-氨基-1,2,3,4-四氢-1-萘酮,CAS:3470-53-9;外观:浅黄棕色固体,HPLC,1H NMR 98%+ 
6)6-Chloro-1-tetralone,6-氯-3,4-二氢-2H-1-萘酮,CAS: 26673-31-4;外观:浅黄色油状物,HPLC,1H NMR 97%+
7)6-碘-3,4-二氢-2H-1-萘酮,CAS: 26673-31-4;外观:白色至类白色固体,HPLC,1H NMR 97%+
CarfilzomibPR171中间体:

8
(S)-4-(tert-Butoxycarbonylamino)-2,6-dimethyl-1-hepten-3-one
CAS: 247068-81-1Appearance: white solidHPLC,1H NMR 99%+;
9CAS:247068-82-2,tert-butyl ((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-yl)carbamate,Appearance: white solidHPLC,1H NMR 98%+;
10)CAS:247068-85-5 Appearance: white solidHPLC,1H NMR 98%+;