Small Molecule Stock List-9.27

2017 China CPHI: E1M35

EOS Med Chem, Medchem is Big

執大象，天下往，往而無害，安平泰

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CEP-28122, 1022958-60-6, (1S,2S,3R,4R)-3-[5-chloro-2-((S)-1-methoxy-7-morpholin-4-yl-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-ylamino)pyrimidin-4-ylamino]bicyclo[2.2.1]hept-5-ene-2-carboxylic acid amide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GDC-0980, RG 7422 , 1032754-93-0, (S)-1-(4-((2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxypropan-1-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

LDK378, Ceritinib, 1032900-25-6, 5-chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

VS-4718 CT-VS4718 PND-1186, SR 2516  , 1061353-68-1, 2-(2-(2-methoxy-4-morpholinophenylamino)-5-(trifluoromethyl)pyridin-4-ylamino)-N-methylbenzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Defactinib  VS-6063, PF-04554878, 1073154-85-4, N-methyl-4-(4-((3-(N-methylmethylsulfonamido)pyrazin-2-yl)methylamino)-5-(trifluoromethyl)pyrimidin-2-ylamino)benzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Pyridostatin, 1085412-37-8, 4-(2-aminoethoxy)-N2,N6-bis(4-(2-aminoethoxy)quinolin-2-yl)pyridine-2,6-dicarboxamide trihydrochloride, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK2126458, Omipalisib, 1086062-66-9, 2,4-difluoro-N-(2-methoxy-5-(4-(pyridazin-4-yl)quinolin-6-yl)pyridin-3-yl)benzenesulfonamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK-923295, 1088965-37-0, 3-chloro-N-((2S)-1-(2-(dimethylamino)acetamido)-3-(4-(8-((S)-1-hydroxyethyl)-2,3-dihydroimidazo[1,2-a]pyridin-2-yl)phenyl)propan-2-yl)-4-isopropoxybenzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

ASP3026, 1097917-15-1, N2-(2-(isopropylsulfonyl)phenyl)-N4-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)-1,3,5-triazine-2,4-diamine, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

D- Luciferin Potassium salt, 115144-35-9, potassium (S)-2-(6-hydroxybenzo[d]thiazol-2-yl)-4,5-dihydrothiazole-4-carboxylate, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AMG-337, 1173699-31-4, (R)-6-(1-(8-fluoro-6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)ethyl)-3-(2-methoxyethoxy)-1,6-naphthyridin-5(6H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AP26113,Brigatinib, 1197953-54-0, 5-chloro-N4-(2-(dimethylphosphoryl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

IPI-145, INK 1197, Duvelisib , 1201438-56-3, (S)-3-(1-(9H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1(2H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GLPG0634 analog, Filgotinib analog, 1206101-20-3 , N-(5-(4-((6-cyanopyridin-3-yl)methoxy)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

LEE-011, Ribociclib, 1211441-98-3, 7-cyclopentyl-N,N-dimethyl-2-(5-(piperazin-1-yl)pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Alpelisib, BYL-719, 1217486-61-7, (S)-N1-(4-methyl-5-(2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl)thiazol-2-yl)pyrrolidine-1,2-dicarboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK2256098, 1224887-10-8, 2-(5-chloro-2-(1-isopropyl-3-methyl-1H-pyrazol-5-ylamino)pyridin-4-ylamino)-N-methoxybenzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK2334470 , 1227911-45-6, ((3S,6R)-1-(6-(3-amino-1H-indazol-6-yl)-2-(methylamino)pyrimidin-4-yl)-6-methylpiperidin-3-yl)(piperidin-1-yl)methanone, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GS-9973, Entospletinib, 1229208-44-9, 6-(1H-indazol-6-yl)-N-(4-morpholinophenyl)imidazo[1,2-a]pyrazin-8-amine, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

HA130, 1229652-21-4, (Z)-3-((4-((3-(4-fluorobenzyl)-2,4-dioxothiazolidin-5-ylidene)methyl)phenoxy)methyl)phenylboronic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

A-1155463, 1235034-55-5, 2-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)-5-(3-(4-(3-(dimethylamino)prop-1-ynyl)-2-fluorophenoxy)propyl)thiazole-4-carboxylic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

RN486, 1242156-23-5, 6-cyclopropyl-8-fluoro-2-(2-(hydroxymethyl)-3-(1-methyl-5-(5-(4-methylpiperazin-1-yl)pyridin-2-ylamino)-6-oxo-1,6-dihydropyridin-3-yl)phenyl)isoquinolin-1(2H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

, 1256577-71-5, 6,6-dimethyl-8-(4-morpholinopiperidin-1-yl)-11-oxo-6,11-dihydro-5H-benzo[b]carbazole-3-carbonitrile, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GDC-0032, Taselisib; RG-7604, 1282512-48-4, 2-(4-(2-(1-isopropyl-3-methyl-1H-1,2,4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)-1H-pyrazol-1-yl)-2-methylpropanamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

NVP-CGM097, 1313363-54-0, (S)-1-(4-chlorophenyl)-7-isopropoxy-6-methoxy-2-(4-(methyl(((1r,4r)-4-(4-methyl-3-oxopiperazin-1-yl)cyclohexyl)methyl)amino)phenyl)-1,2-dihydroisoquinolin-3(4H)-one hydrochloride, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

NVP-CGM097, 1313363-54-0, (S)-1-(4-chlorophenyl)-7-isopropoxy-6-methoxy-2-(4-(methyl(((1r,4r)-4-(4-methyl-3-oxopiperazin-1-yl)cyclohexyl)methyl)amino)phenyl)-1,2-dihydroisoquinolin-3(4H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK126, 1346574-57-9, (S)-1-sec-butyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

CNDAC HCl salt, 134665-72-8, (2R,3S,4S,5R)-2-(4-amino-2-oxopyrimidin-1(2H)-yl)-4-hydroxy-5-(hydroxymethyl)tetrahydrofuran-3-carbonitrile hydrochloride, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

HM71224, Olmutinib, 1353550-13-6, N-(3-(2-(4-(4-methylpiperazin-1-yl)phenylamino)thieno[3,2-d]pyrimidin-4-yloxy)phenyl)acrylamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

GSK2636771, 1372540-25-4, 2-methyl-1-(2-methyl-3-(trifluoromethyl)benzyl)-6-morpholino-1H-benzo[d]imidazole-4-carboxylic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

BAY-1082439; BAY 2439, 1375469-38-7, (R)-N-(8-(2-hydroxy-3-morpholinopropoxy)-7-methoxy-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl)-2-methylnicotinamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

M2698, 1379545-95-5, (S)-4-(2-(azetidin-1-yl)-1-(4-chloro-3-(trifluoromethyl)phenyl)ethylamino)quinazoline-8-carboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

CEP-37440, 1391712-60-9, (S)-2-(5-chloro-2-(6-(4-(2-hydroxyethyl)piperazin-1-yl)-1-methoxy-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-ylamino)pyrimidin-4-ylamino)-N-methylbenzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

ACP196 (Acalabrutinib), 1420477-60-6, (S)-4-(8-amino-3-(1-but-2-ynoylpyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AZD9291, Osimertinib; Mereletinib, 1421373-65-0, N-(2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methoxy-5-(4-(1-methyl-1H-indol-3-yl)pyrimidin-2-ylamino)phenyl)acrylamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AZ5104, 1421373-98-9, N-(5-(4-(1H-indol-3-yl)pyrimidin-2-ylamino)-2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methoxyphenyl)acrylamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

A-1331852, 1430844-80-6, 6-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-(1-(adamantylmethyl)-5-methyl-1H-pyrazol-4-yl)picolinic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AG-221, Enasidenib, 1446502-11-9, 2-methyl-1-(4-(6-(trifluoromethyl)pyridin-2-yl)-6-(2-(trifluoromethyl)pyridin-4-ylamino)-1,3,5-triazin-2-ylamino)propan-2-ol, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AZD3965, 1448671-31-5, (S)-5-(4-hydroxy-4-methylisoxazolidine-2-carbonyl)-1-isopropyl-3-methyl-6-((5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)methyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

BLU9931, 1538604-68-0, N-(2-(6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-ylamino)-3-methylphenyl)acrylamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

LY-294002, 154447-36-6 , 2-morpholino-8-phenyl-4H-chromen-4-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

EPZ011989, 1598383-40-4, N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl((1r,4r)-4-((2-methoxyethyl)(methyl)amino)cyclohexyl)amino)-2-methyl-5-(3-morpholinoprop-1-ynyl)benzamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

LY-3177833, 1627696-51-8, (R)-3-(5-fluoropyrimidin-4-yl)-3-methyl-6-(1H-pyrazol-4-yl)isoindolin-1-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

A-1210477, 1668553-26-1, 7-(5-((4-(4-(N,N-dimethylsulfamoyl)piperazin-1-yl)phenoxy)methyl)-1,3-dimethyl-1H-pyrazol-4-yl)-1-(2-morpholinoethyl)-3-(3-(naphthalen-1-yloxy)propyl)-1H-indole-2-carboxylic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

IPI-549, 1693758-51-8, (S)-2-amino-N-(1-(8-((1-methyl-1H-pyrazol-4-yl)ethynyl)-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl)ethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Aprepitant, 170729-80-3, 3-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-(4-fluorophenyl)morpholino)methyl)-1H-1,2,4-triazol-5(4H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Mirabegron, 223673-61-8, (R)-2-(2-aminothiazol-4-yl)-N-(4-(2-(2-hydroxy-2-phenylethylamino)ethyl)phenyl)acetamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AVN944 (VX-944) , 297730-17-7, (R)-1-cyanobutan-2-yl (S)-1-(3-(3-(3-methoxy-4-(oxazol-5-yl)phenyl)ureido)phenyl)ethylcarbamate, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

IC-87114, 371242-69-2, 2-((6-amino-9H-purin-9-yl)methyl)-5-methyl-3-o-tolylquinazolin-4(3H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

AS 605240, 648450-29-7, (Z)-5-(quinoxalin-6-ylmethylene)thiazolidine-2,4-dione, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Elvitegravir, 697761-98-1, (S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-methylbutan-2-yl)-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

PCI-27483, 871266-63-6, (S)-2-(2-(5-(5-carbamimidoyl-1H-benzo[d]imidazol-2-yl)-2',6-dihydroxy-5'-sulfamoylbiphenyl-3-yl)acetamido)succinic acid, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Trametinib (GSK1120212，JTP 74057), 871700-17-3, N-(3-(3-cyclopropyl-5-(2-fluoro-4-iodophenylamino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7-tetrahydropyrido[4,3-d]pyrimidin-1(2H)-yl)phenyl)acetamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

BGJ-398,NVP-BGJ398,Infigratinib, 872511-34-7, 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-(4-(4-ethylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)-1-methylurea, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

PIK-293 , 900185-01-5  , 2-((4-amino-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)-5-methyl-3-o-tolylquinazolin-4(3H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

NVP-BKM120, 944396-07-0, 5-(2,6-dimorpholinopyrimidin-4-yl)-4-(trifluoromethyl)pyridin-2-amine, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

Decernotinib,VX-509, 944842-54-0, (R)-2-(2-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-ylamino)-2-methyl-N-(2,2,2-trifluoroethyl)butanamide, HPLC 99%, NMR, LCMS is ok, stock more than 10g.

MK-1775, AZD1775， , 955365-80-7, 2-allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6-(4-(4-methylpiperazin-1-yl)phenylamino)-1H-pyrazolo[3,4-d]pyrimidin-3(2H)-one, HPLC 99%, NMR, LCMS is ok, stock more than 10g.